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2-[1-(2,3-dihydro-1H-inden-5-yl)-5-[5-(propan-2-yl)-1,2-oxazol-3-yl]-1H-1,2,4-triazol-3-yl]acetamide
2-benzyl-8-[2-(propylsulfanyl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3R,4R)-3-hydroxypiperidin-4-yl]-2-(2,3,4-trifluorophenyl)acetamide
1-(4-fluorobenzenesulfonyl)-3-(4-methyl-1H-pyrazol-5-yl)piperidine
5-[(2-{[3-(trifluoromethyl)phenyl]methyl}morpholin-4-yl)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-{1-[2,2-dimethyl-1-(thiophen-2-yl)cyclopropanecarbonyl]azetidin-3-yl}pyridine
2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-1-methyl-5-phenyl-1H-pyrrole
(1S,5R)-3-(pyridin-3-ylmethyl)-6-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
5-[5-(ethoxycarbonyl)-2,4-dimethyl-1H-pyrrole-3-carbonyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-({5-propyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-(trifluoromethyl)pyridin-2-amine
3-[3-(2-methoxyphenoxy)azetidine-1-carbonyl]naphthalen-2-ol
2-(2,2-diphenylethyl)-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine
1-cycloheptyl-N-[2-(2-methoxyphenyl)ethyl]-6-oxopiperidine-3-carboxamide
3-(2-ethyl-1H-imidazol-1-yl)-1-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-methoxy-N-({1-[(2E)-3-phenylprop-2-en-1-yl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrrole-3-carboxamide
2-{[5-(4-hydroxy-3-methoxyphenyl)-4-(4-methylphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
2-[4-(3-fluorophenyl)oxan-4-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-1-cyclopropanecarbonylpiperidine-4-carboxamide
2-(6-methyl-1-benzofuran-3-yl)-N-[2-(4-methylmorpholin-2-yl)ethyl]acetamide
1,5-dimethyl-4-({4-[2-(oxolan-2-yl)-5-(trifluoromethyl)-1H-1,3-benzodiazol-1-yl]piperidin-1-yl}methyl)-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
2-({4-[3-(hydroxymethyl)-8-methylquinolin-2-yl]-1H-pyrrolo[2,3-b]pyridin-6-yl}amino)acetic acid
N-[(1-{[4-(propan-2-yloxy)phenyl]methyl}piperidin-3-yl)methyl]acetamide
ethyl 4-[(4-chlorophenyl)methyl]-1-[(2-hydroxy-6-methoxyphenyl)methyl]piperidine-4-carboxylate
4-(4-methanesulfonylphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[3-(4-{[2-(1H-indol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]cyclopropanecarboxamide
1-(1-benzothiophen-2-ylmethyl)-3-[5-(benzylsulfanyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
(3S,4R)-1-(5,6-dimethoxypyrazine-2-carbonyl)-4-methylpiperidine-3,4-diol
N-(3-{4-[4-(furan-2-carbonyl)piperazin-1-yl]piperidin-1-yl}phenyl)-2-methoxybenzamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-2-(morpholine-4-carbonyl)pyridin-4-amine
2-[methyl(pyridin-2-ylmethyl)amino]-1-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]ethan-1-one
3-(3-chloro-1,2-oxazol-5-yl)-1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]propan-1-one
2-cyclopropyl-5-{2-[2-(pyrrolidin-1-yl)ethyl]piperidine-1-carbonyl}pyrimidine
7-(3-chlorophenyl)-4-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
2-(3-methoxypropyl)-8-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-2,8-diazaspiro[4.5]decan-3-one
(1R,7S)-3-[4-(2-hydroxyethyl)phenyl]-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]pyrimidine-5-carboxamide
6-{2-[3-(4-fluorophenyl)-1,2,4-oxadiazol-5-yl]ethyl}-2,3,4,5-tetrahydropyridazin-3-one
6-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine
3-[(3R,4S)-1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
2-(5-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-1H-1,3-benzodiazol-1-yl)ethan-1-ol
5-methyl-N-[(3R,5S)-1-[(5-methylfuran-2-yl)methyl]-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
2,6-dimethyl-4-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidine-1-carbonyl}quinoline
5-(2-cyclopropyl-1H-imidazol-1-yl)-1,3-diethyl-6-methyl-2,3-dihydro-1H-1,3-benzodiazol-2-one
2-phenyl-1-{1-[1-(4,6,7-trimethylquinazolin-2-yl)piperidin-4-yl]piperidin-4-yl}ethan-1-ol
N-[4-({1-tert-butyl-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl}methyl)phenyl]acetamide
3-{[4-(4-methoxypyrimidin-2-yl)piperazin-1-yl]methyl}-N-methylpyridin-2-amine
4-{4-[(dimethylamino)methyl]-1H-1,2,3-triazol-1-yl}-N-(4-methoxy-2-methylphenyl)piperidine-1-carboxamide
methyl 4-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-pyrrole-2-carboxylate