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N-[2-(pyridin-3-yl)ethyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(quinolin-3-ylmethyl)amine
3-(5-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)propanoic acid
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)-3-methylpyridin-2-amine
9-(2,6-difluorobenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]methyl}quinolin-4-ol
N-{1-[1-(dimethyl-1,3-thiazole-5-carbonyl)piperidin-4-yl]-2-(3-methoxyphenyl)ethyl}-N,1-dimethyl-1H-pyrazole-3-carboxamide
3-{[(5,6-dimethylpyrimidin-4-yl)amino]methyl}-N-methylbenzamide
4-ethyl-3-{1-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)acetyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
N,N-bis(1,3-oxazol-4-ylmethyl)-4-(pyrrolidin-1-ylmethyl)benzamide
8-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-3-methyl-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
(1S,3R)-N-(2-ethoxyethyl)-3-(3-fluoro-4-methylbenzenesulfonamido)cyclopentane-1-carboxamide
2-{[3-(1H-imidazol-1-yl)propyl](pyridin-4-ylmethyl)amino}-2-(2-methoxy-5-methylphenyl)acetic acid
2-{1-[(3-methoxyphenyl)methyl]-4-[(1-methyl-1H-indol-3-yl)methyl]piperazin-2-yl}ethan-1-ol
[3-(cyclopropylmethyl)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-3-yl]methanol
5-methyl-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-1,3-oxazole-4-carboxamide
1-cyclopentyl-N-[(2-ethoxypyridin-3-yl)methyl]-5-oxopyrrolidine-3-carboxamide
(2-chloro-6-fluorophenyl)({4-[(1-methyl-1H-pyrazol-4-yl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl})methanol
(1S,5R)-N,N-dimethyl-7-oxo-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-(ethylamino)-N-[3-(1H-imidazol-1-yl)propyl]-5-(pyrrolidine-1-sulfonyl)benzamide
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)cyclopropanecarboxamide
(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-6-({6-methylimidazo[1,2-a]pyridin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane
2-(naphthalen-2-yloxy)-1-(thiomorpholin-4-yl)propan-1-one
N-cyclopentyl-N'-{[2-(1H-imidazol-1-yl)pyridin-3-yl]methyl}ethanediamide
1-[4-(4-fluorophenyl)oxane-4-carbonyl]-3-propylpiperidine-3-carboxylic acid
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(2-methoxyphenyl)propanamide
5-methoxy-2-({4-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}methyl)pyridin-4-ol
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-3-(2-methoxyphenyl)propanamide
3-({4-[(3-fluorophenyl)methyl]piperazin-1-yl}methyl)-3-hydroxy-1-methylpiperidin-2-one
5-[4-(3-phenylpropyl)-1,4-diazepane-1-carbonyl]pyrazin-2-ol
1-{1-[(4-ethylphenyl)methyl]piperidin-3-yl}-4-(4-methoxyphenyl)piperazine
2-(methylsulfanyl)-5-{[3-(4-phenoxybenzoyl)piperidin-1-yl]methyl}pyrimidine
N-(1-{1-[(6-ethoxyquinolin-2-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)acetamide
2-({5-[(4-hydroxyphenyl)methyl]-4-(pyridin-3-yl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
1-[2-(3-fluorophenyl)ethyl]-N-[(2-methyl-1H-indol-5-yl)methyl]-6-oxopiperidine-3-carboxamide
1-{[(2R,5S)-5-[(3,4-dimethoxyphenyl)methyl]oxolan-2-yl]methyl}-4-methyl-1,4-diazepane
(2S,4R)-1-(2,2-diphenylethyl)-N-methyl-4-({[2-(prop-2-en-1-yloxy)phenyl]methyl}amino)pyrrolidine-2-carboxamide
N-(furan-2-ylmethyl)-N-methyl-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
2-[(4aS,7aR)-4-ethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-(furan-2-ylmethyl)acetamide
(2R,3R,6R)-3-(4-methoxyphenyl)-5-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
4-(cyclopropylmethyl)-3-(propan-2-yl)-1-[4-(1H-pyrazol-4-yl)butanoyl]-1,4-diazepan-5-one
1-ethyl-4-[2-(2-phenylethyl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[3-chloro-4-(1H-1,2,4-triazol-1-yl)phenyl]-3-[2-(2-hydroxyethoxy)ethyl]urea
3-{2-[(1S,4S)-2-azabicyclo[2.2.1]heptan-2-yl]-2-oxoethyl}-4-[(3-methylphenyl)methyl]piperazin-2-one
1-[1-(1H-imidazol-1-yl)butan-2-yl]-3-[1-(4-methoxyphenyl)-3-methyl-1H-pyrazol-5-yl]urea
5-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-N-methyl-N-[2-(1H-pyrazol-4-yl)ethyl]pyridin-2-amine
2-(4-methylphenoxymethyl)-N-[(1-methylpyrrolidin-3-yl)methyl]furan-3-carboxamide
5-(4-{[(5-ethyl-2-methylpyrimidin-4-yl)amino]methyl}piperidin-1-yl)-2-methyl-2,3-dihydropyridazin-3-one
2-cyclopropyl-N-(2-fluorophenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide