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2-(4-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}phenoxy)acetic acid
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]acetamide
3-{1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{[(1-{2,7-dimethylpyrazolo[1,5-a]pyrimidine-5-carbonyl}piperidin-3-yl)oxy]methyl}pyridine
1-(2-{4-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)-1H-1,3-benzodiazole
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
[5-({4-[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)furan-2-yl]methanol
2-[5-(5-propyl-1,2-oxazole-3-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
5-(3-cyclopropyl-1H-1,2,4-triazol-5-yl)-1H-indole
(1S,5R)-3-benzoyl-6-cycloheptanecarbonyl-3,6-diazabicyclo[3.2.2]nonane
N-[(2-fluorophenyl)methyl]-1-methyl-3-(2-methylpropyl)-N-propyl-1H-pyrazole-5-carboxamide
N-tert-butyl-3-[2-(furan-2-yl)-1H-imidazol-1-yl]-2-methylbenzamide
7-methyl-3-[(1-propyl-1H-imidazol-2-yl)methyl]-3,7,11-triazaspiro[5.6]dodecan-12-one
N-methyl-5-{1-[2-(methylamino)pyridine-4-carbonyl]pyrrolidin-2-yl}-N-(propan-2-yl)thiophene-2-carboxamide
N-[2-(4-methylmorpholin-2-yl)ethyl]-5-(4-methylphenyl)furan-2-carboxamide
2-{4-[2-amino-6-(methylamino)pyrimidin-4-yl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
methyl 4-({4-[(2-fluoro-4-methoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)benzoate
1-(3-ethyl-5-methyl-1,2-oxazole-4-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(4aS,8aS)-2-(2H-1,3-benzodioxol-4-ylmethyl)-decahydroisoquinolin-4a-ol
N-cyclopropyl-3-{1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-yl}propanamide
2,4-bis(propan-2-yl)-6-[4-(pyrrolidin-3-yl)piperazine-1-carbonyl]phenol
2-(2-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-2-oxoethyl)-2,3-dihydro-1H-isoindole-1,3-dione
4-{[(2R,3S,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]methyl}-2-methylphenol
4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]-N-[(1R,3S)-3-(pyrrolidine-1-carbonyl)cyclopentyl]butanamide
2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]-1-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
N-[1-(6-methylpyridin-2-yl)ethyl]-4-[(6-methylpyridin-3-yl)oxy]piperidine-4-carboxamide
4-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfonyl]-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-(2-hydroxy-2-phenylethyl)-N,5-dimethyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)(pyridin-4-ylmethyl)amine
N-[(1-ethylpiperidin-3-yl)methyl]-1-methyl-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
3-(4-hydroxyphenyl)-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]propanamide
N-[1-(2-chlorophenyl)cyclopropyl]-6-ethyl-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}furan-2-yl)-1-methyl-1H-1,3-benzodiazole
4-(4-methylpiperazin-1-yl)-6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-2-amine
1-(2,3-dihydro-1,4-benzodioxin-6-yl)-5-(2H-1,2,3-triazol-2-ylmethyl)-1H-1,2,4-triazole
N-cyclopropyl-1-[(1s,4s)-4-{[(2,5-dimethoxyphenyl)methyl]amino}cyclohexyl]-1H-1,2,3-triazole-4-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
6-(1-{[(1,3-dimethyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazol-4-yl)-N-propylpyridine-3-carboxamide
1-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(3-hydroxyphenyl)pyridine-3-carbonitrile
(1S,6R)-N-[3-(1,3-oxazol-5-yl)phenyl]-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
1-{imidazo[1,2-a]pyridine-3-carbonyl}-4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine
2-[4-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperazin-1-yl]pyridine-3-carboxamide
1-(2-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydropyridin-2-one
3-[5-({7-[(2-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}methyl)thiophen-2-yl]prop-2-yn-1-ol
[1-(5-{[(2,5-dimethylphenyl)methyl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
2-[2-({8-fluoro-1H,2H,3H,4H,5H-pyrido[4,3-b]indol-2-yl}methyl)phenoxy]acetamide
1-[(4aR,8aR)-1-(furan-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-(3-methoxyphenyl)ethan-1-one
1-[(3,4-dimethylphenyl)methyl]-4-[4-(1H-pyrazol-4-yl)butanoyl]piperazin-2-one