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3-(2H-1,3-benzodioxol-5-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
1,3-dimethyl-N-(2,2,2-trifluoroethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
6-[4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
4-{[5-methyl-2-(2-methylphenyl)-1,3-oxazol-4-yl]methyl}-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
3-(4-{4-[(4-benzylpiperidin-1-yl)methyl]phenoxy}piperidine-1-carbonyl)pyridine
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-(3-methoxypiperidin-1-yl)pyridine-3-carboxamide
methyl 5-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
N-(diphenylmethyl)-1-methyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(2-methylphenoxy)-1-(6-methylpyridazin-3-yl)piperidine-4-carboxylic acid
N-[3-(1H-imidazol-2-yl)propyl]-2-methylthieno[3,2-d]pyrimidin-4-amine
N-cyclopropyl-4-{[2-(3-methylphenyl)ethyl]sulfamoyl}benzamide
4-[(1-acetylpiperidin-4-yl)oxy]-3-methoxy-N-[1-(pyridin-3-yl)propan-2-yl]benzamide
(1S,5R)-6-(2-methoxypyridine-4-carbonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-ethyl-1-[(3-methoxyphenyl)methyl]-5-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[3-(naphthalen-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propanoic acid
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[(5-methylthiophen-2-yl)methyl](pyridin-4-ylmethyl)amine
3-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}pyridine
3-(2,5-dimethoxyphenyl)-1-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-1-methylurea
2-[5-(ethylsulfanyl)thiophene-2-carbonyl]-7-(2-hydroxyethyl)-2,7-diazaspiro[4.5]decan-6-one
1-cyclopentyl-6-oxo-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidine-3-carboxamide
3-{2-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]propyl}pyridine
2-{4-[(4-methoxy-2,5-dimethylphenyl)methyl]-1-methylpiperazin-2-yl}ethan-1-ol
3-(3-chlorophenyl)-N-(5-acetamido-2-methoxyphenyl)pyrrolidine-1-carboxamide
2-[3-(dimethylamino)propyl]-9-[2-(3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-cyclopentyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[(2-methylphenyl)methyl]propanamide
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetic acid
2-{3-[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]phenyl}-5-methyl-1,3,4-thiadiazole
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}piperidin-4-amine
3-{1-[(trimethyl-1H-pyrazol-4-yl)sulfonyl]piperidin-3-yl}benzoic acid
5-(2,6-difluorophenoxymethyl)-N-[3-(methylsulfanyl)propyl]-1,2-oxazole-3-carboxamide
(2S)-3-({4-[4-(2-chlorophenyl)piperidin-4-yl]pyrimidin-2-yl}amino)propane-1,2-diol
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-6-(piperidin-4-yl)pyrimidin-4-amine
2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)-N-methylethane-1-sulfonamide
N-(1-methoxypropan-2-yl)-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-benzyl-8-phenylmethanesulfonyl-2,8-diazaspiro[4.5]decan-3-one
2-[1-(1H-1,3-benzodiazol-2-ylmethyl)pyrrolidin-3-yl]benzoic acid
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(5-ethyl-1,2,4-oxadiazol-3-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
4-(1-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}piperidin-4-yl)thiomorpholine
N-{[7-(2-methoxy-2-phenylacetyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-2-phenoxyacetamide
5-methanesulfonyl-2-methyl-N-(oxan-4-yl)pyrimidin-4-amine
2-{4-cyclobutyl-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-(2-fluorophenyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(6-ethoxypyridin-3-yl)methyl]-4-(pyrrolidin-3-yl)piperazine
7-(2-cyclohexylethyl)-6-oxo-N-(propan-2-yl)-2,7-diazaspiro[4.5]decane-2-carboxamide
1-{3-[4-(2-methoxyphenyl)piperazin-1-yl]piperidin-1-yl}-5-phenylpentan-1-one
1-[2-methyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-(2-methylbutan-2-yl)urea
3-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-4,5,6,7-tetrahydro-1,2-benzoxazole
3-(3-hydroxy-3-methylbutyl)-N-{[4-(5-methyl-1,2,4-oxadiazol-3-yl)phenyl]methyl}benzamide