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5-({2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-1-yl]ethyl}sulfanyl)-1H-1,2,3-triazole
3-ethoxy-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
N-methyl-N-(1,3-thiazol-2-ylmethyl)-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
methyl 3-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]benzoate
2-{1-[(2,4-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-(propan-2-yl)acetamide
N-(4-{[2-(3-fluorophenyl)azepan-1-yl]methyl}phenyl)acetamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(2-methoxypyridine-3-carbonyl)pyrrolidin-3-yl]methanol
4-[1-(3-methylphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
1-[1-(1-aminocyclopropanecarbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
2,7,8-trimethyl-N-[1-(1-methyl-1H-1,2,4-triazol-5-yl)propyl]quinoline-4-carboxamide
1-(4-benzoylpiperazin-1-yl)-2-(ethanesulfonyl)propan-1-one
N4-[(2,4-dimethoxyphenyl)methyl]-N2,N2-dimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N-(1,1-dioxo-1λ6-thian-4-yl)-N,2,3,6-tetramethylquinoline-4-carboxamide
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-{2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}morpholine
3-(3,5-dimethylphenyl)-N-(pyridin-2-ylmethyl)propanamide
(2S,4S)-4-amino-N-ethyl-1-[3-(3-methyl-1H-pyrazol-1-yl)propanoyl]pyrrolidine-2-carboxamide
4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]-1-[3-(pyridin-2-yl)azetidin-1-yl]butan-1-one
1-methyl-1'-[3-(1-methylpiperidin-3-yl)propanoyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
9-methoxy-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
ethyl 4-[5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-amido]piperidine-1-carboxylate
N-{[1-(2-chloropyridine-4-carbonyl)piperidin-3-yl]methyl}-2-(2-methoxyphenoxy)acetamide
(3R)-3-cyclopropyl-4,4-dimethyl-1-(1-methyl-4-phenylpiperidine-4-carbonyl)pyrrolidin-3-ol
2-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]quinoline
N-methyl-N'-(4-methylphenyl)-N-(pyrazin-2-ylmethyl)propanediamide
N-[(4-{[(2-fluorophenyl)methyl]amino}-8-methylquinazolin-2-yl)methyl]-2,3-dihydro-1,4-benzodioxine-6-sulfonamide
1-[3-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(morpholin-4-yl)phenyl]ethan-1-one
N-[(5-fluoro-2-methylphenyl)methyl]-1-(2-methylpropyl)-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[2-(cyclohexylsulfanyl)ethyl]-5-ethyl-1,3,4-oxadiazol-2-amine
(3R,5S)-N-(2,3-dihydro-1H-inden-5-yl)-5-(piperidine-1-carbonyl)-1-(pyridin-4-ylmethyl)piperidine-3-carboxamide
4-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}-3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazole
2-ethyl-N-[3-(pyridin-3-yloxy)propyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
[(1-cyclohexylpiperidin-3-yl)methyl][(3,5-difluorophenyl)methyl](pyridin-3-ylmethyl)amine
4-{4-ethyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}-1-(3-methoxypropyl)piperidine
3,4-difluoro-N-(1-hydroxybutan-2-yl)-N-(pyridin-2-ylmethyl)benzamide
N-(2,4-dimethoxyphenyl)-3-[1-(thiolan-3-yl)piperidin-4-yl]propanamide
2-methyl-4-(3-{9-methyl-3,9-diazaspiro[5.6]dodecane-3-carbonyl}phenyl)butan-2-ol
2-{5-methyl-4-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(5-methylfuran-2-yl)pyrimidine
methyl 4-({4-[(2E)-4-methylpent-2-en-1-yl]-7-oxo-1,4-diazepan-1-yl}methyl)benzoate
(1R,2R,4R)-N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)bicyclo[2.2.1]hept-5-ene-2-carboxamide
4-hydroxy-N-methyl-2-(4-methylphenyl)-N-[1-(pyridin-3-yl)ethyl]pyrimidine-5-carboxamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]quinoxaline-6-carboxamide
(2S)-3-methyl-2-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)butanamide
8-fluoro-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]quinoline-2-carboxamide
N-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
2-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]-1H-imidazol-2-yl}-8-methoxyquinoline
3-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}urea
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]cycloheptanecarboxamide
3-cyclopropyl-1-[(3-methoxyphenyl)methyl]-5-[1-(1H-1,2,4-triazol-1-yl)ethyl]-1H-1,2,4-triazole
(3aR,5S,6S,7aS)-2-{4H-thieno[3,2-b]pyrrole-5-carbonyl}-octahydro-1H-isoindole-5,6-diol