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1-[2-(3-methylphenyl)ethyl]-3-phenylpyrrolidin-3-ol
3-cyclohexyl-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-1H-pyrazole-4-carboxamide
N-benzyl-N-(2-hydroxyethyl)-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
1-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]-4-(1H-pyrrole-2-carbonyl)piperazine
3-(3-methylthiophene-2-carbonyl)-1-(thian-4-yl)piperidine
7-(3-chloro-4-hydroxybenzoyl)-2-(pyridin-3-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(3,4-dichlorophenyl)-4-[3-(1H-imidazol-1-yl)propyl]morpholine
1-{2-[benzyl(ethyl)carbamoyl]ethyl}piperidine-3-carboxamide
(3aS,6aS)-1-oxo-5-(4-phenylbutanoyl)-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(4-fluorophenyl)-N-{2-[4-(propan-2-yloxy)phenyl]ethyl}-1,2,4-triazin-3-amine
1-ethyl-N-{2-[2-(2-methoxyphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-1H-pyrazole-4-carboxamide
2,8-dimethyl-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}-[1,2,4]triazolo[1,5-a]pyridine
3-[(5-cyclopropyl-1,3,4-oxadiazol-2-yl)methyl]-7-methoxy-2,3,4,5-tetrahydro-1H-3-benzazepine
1-{6-methylthieno[2,3-d]pyrimidin-4-yl}-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]piperidin-4-amine
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propan-1-one
5-({[1-(4-methoxyphenyl)cyclopentyl]methyl}carbamoyl)-1H-imidazole-4-carboxylic acid
3-methoxy-5-{4-[2-(methylsulfanyl)ethyl]piperazine-1-carbonyl}benzoic acid
N-[(1-cyclohexylpiperidin-3-yl)methyl]-3-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)propanamide
N-(2,3-dihydro-1H-inden-2-yl)-2-(pyrrolidin-3-yl)benzamide
2-[(2S,5R)-2,5-dimethylpiperazin-1-yl]-4-(2,6-dimethylpyridin-3-yl)pyrimidine
N,N-dimethyl-4-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]piperazine-1-carboxamide
2-acetyl-7-(2-cyclohexylethyl)-2,7-diazaspiro[4.5]decan-6-one
5-benzyl-4-[2-(dimethylamino)acetyl]-1-(3-methoxyphenyl)piperazin-2-one
2-{4-[2-(trifluoromethoxy)phenyl]-1H-pyrazol-1-yl}propanamide
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-5-methylthiophene-2-carboxamide
2-[2-(butan-2-yl)phenoxy]-N-methyl-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]acetamide
3-(1-methylpiperidin-2-yl)-N-[2-(1H-pyrrol-1-yl)ethyl]propanamide
(3aS,6aR)-5-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-3-(pyridin-2-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
(1R,5S,6S)-6-({4-[4-cyclopropyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-3-azabicyclo[3.1.0]hexane
methyl 2-[3-oxo-4-(1,3-thiazol-2-ylmethyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetate
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-N-(2,3-dihydro-1H-inden-1-yl)-1,3-oxazole-4-carboxamide
2-{2-[(3R,4R)-3-[(4-ethylpiperazin-1-yl)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
6-fluoro-2-({[3-(propan-2-yloxy)propyl]amino}methyl)quinolin-4-ol
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-6-(thiophen-3-yl)pyridine-3-carboxamide
2-[4-(2-fluorophenyl)piperazin-1-yl]-4-(pyridin-4-yl)pyrimidine
4-({methyl[(4-methyl-1H-imidazol-2-yl)methyl]amino}methyl)benzoic acid
N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-1H-indazole-3-carboxamide
2-{[3-(2-fluorophenyl)pyrrolidin-1-yl]methyl}-8-methoxyquinoline
1-{2-oxo-2-[2-(trifluoromethyl)morpholin-4-yl]ethyl}-1H-indole-3-carboxamide
(3aS,7aR)-2-[(6-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}-1-phenylpiperazine-2-carboxylic acid
7-methyl-2-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}-2,7-diazaspiro[4.5]decan-6-one
5-{[4-(diphenylmethyl)piperazin-1-yl]methyl}-N,N-dimethylpyrimidin-2-amine
1-[(2-methyl-1,3-thiazol-4-yl)methyl]-4-[(2-methyl-1-benzothiophen-3-yl)methyl]piperazine
1-[4-(1-hydroxy-3-methylbutyl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
(2S,4R)-1-[2-(2,3-difluorophenyl)acetyl]-4-(dimethylamino)pyrrolidine-2-carboxylic acid
2-[3-(4-benzyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridin-3-ol
4,6-dimethyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-(3-fluoropyridin-2-yl)-2-(6-methoxynaphthalen-2-yl)morpholine
N,N,6-trimethyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine