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2-{1-[(4-fluorophenyl)methyl]-4-[(2,3,4-trimethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
(5S,9aS,9bS)-2-[(3-chlorophenyl)methyl]-5-(3-methyl-1H-pyrazol-5-yl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[4-(5-methyl-1,2-oxazole-3-carbonyl)morpholin-3-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
2-(3-{[4-(6-ethylpyrimidin-4-yl)piperazin-1-yl]methyl}-1H-indol-1-yl)acetamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carboxamide
(2S)-2-amino-N-butyl-N-cycloheptyl-3-methoxypropanamide
4-methyl-7-{[4-(pyridin-3-ylmethoxy)piperidin-1-yl]methyl}-2H-chromen-2-one
1-(2-methyl-4-{[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
2,3,5,6-tetramethyl-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}benzamide
N-benzyl-6-(pyrrolidin-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
(3R,5S)-N-butyl-5-(3-fluorophenoxymethyl)-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
1-[3-(4-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-[3-benzyl-1-(4-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(2-hydroxypropyl)acetamide
1-{2-[1-(3-chloro-5-fluorobenzoyl)piperidin-2-yl]ethyl}pyrrolidin-2-one
1-acetyl-N-{3-[(4-chlorophenyl)sulfanyl]propyl}piperidine-3-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-3-[(2-methylprop-2-en-1-yl)oxy]benzamide
4-(1-benzyl-1H-pyrazol-4-yl)-1-(but-2-yn-1-yl)-1,2,3,6-tetrahydropyridine
2-{2-ethoxy-4-[(4-ethyl-3,3-dimethylpiperazin-1-yl)methyl]phenoxy}propanoic acid
1-(3-chlorophenyl)-4-{1-[2-(pyridin-2-yl)ethyl]piperidin-3-yl}piperazine
(2R,3S,6R)-5-cyclopropanecarbonyl-3-(3,5-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
(3aS,6aS)-2-methyl-5-(5-propyl-1,3,4-thiadiazol-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
(4aS,7aR)-1-[1-(2-aminoethyl)-1H-1,2,3-triazole-4-carbonyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(ethanesulfonyl)ethyl]-5-(methoxymethyl)furan-2-carboxamide
N-({5-cyclohexyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-3-(pyridin-3-yl)propanamide
3-(difluoromethoxy)-N-(1H-imidazol-2-ylmethyl)-N-methylbenzamide
4-[(5-tert-butyl-1,3,4-oxadiazol-2-yl)amino]-N-phenylpiperidine-1-carboxamide
1-ethyl-3-(3-fluoro-4-methylphenyl)-6-[1-(methylsulfanyl)propan-2-yl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
3-(furan-2-yl)-4-{5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-1-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
3-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-N-cyclopropylpropanamide
5-{5-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazol-3-yl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
1-(3-cyano-4-ethoxyphenyl)-3-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(2-methylpropyl)urea
6-(methoxymethyl)-N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]pyrimidin-4-amine
3-[4-benzyl-2-(hydroxymethyl)piperazine-1-carbonyl]-5,6-dimethyl-1,2-dihydropyridin-2-one
N3-[3-(2,4-dimethylphenoxy)propyl]-N3-methylpiperidine-1,3-dicarboxamide
{[3-(3,4-dimethylpiperazine-1-carbonyl)pyrazolo[1,5-a]pyrimidin-6-yl]methyl}diethylamine
2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
5-[1-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)pyrrolidin-2-yl]-3-methyl-1,2-oxazole
2-(4-acetylphenoxy)-1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
4-({3-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]phenyl}methyl)morpholine
8-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-methyl-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclohexyl-4-(5-ethyl-1,2,4-oxadiazol-3-yl)-1,4-diazepane
N-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-1-(2-methoxyethyl)piperidine-4-carboxamide
3-{[4-methyl-6-({2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}amino)pyrimidin-2-yl]amino}phenol
2-amino-4-methyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,3-benzothiazole-6-carboxamide
6-[3-(dimethylamino)pyrrolidin-1-yl]-N-[(4-ethyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
(1R,5S,6R)-N-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]-3-{[2-(2-methylphenyl)pyrimidin-5-yl]methyl}-3-azabicyclo[3.1.0]hexane-6-carboxamide
N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-6-(1-methyl-1H-imidazol-2-yl)pyridazin-3-amine
N-(furan-2-ylmethyl)-N,1-dimethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-(1,3-benzothiazol-2-yl)-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol