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4-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepine-8-carbonyl}-1-(2-methoxyphenyl)-1H-pyrazole
(4aR,7aS)-1-acetyl-4-[(4-hydroxyquinolin-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-(4-fluorophenyl)pyrrolidin-1-yl]-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propan-1-one
(4aS,7aR)-1-[(4-methylphenyl)methyl]-4-(pyridin-4-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetamide
N-cyclopropyl-2-(2-methoxyethyl)-N-(thiophen-3-ylmethyl)-1,3-benzoxazole-6-carboxamide
2-methyl-2-(4-{1H-pyrrolo[2,3-b]pyridin-4-yl}phenyl)propanamide
7-(cyclopropylmethyl)-2-(4-methyl-1H-imidazole-5-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
6-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-9H-purin-2-amine
3-methyl-1-[2-(1,3,4-oxadiazol-2-yl)phenyl]-3-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)urea
5-ethyl-2-(1-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
(3S,4S)-1-{[1-(2,4-difluorophenyl)-3-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3,4-diol
2-[(4-benzylpiperazin-1-yl)methyl]-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
(4aS,7aR)-1-[(2E)-3-phenylprop-2-en-1-yl]-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(4-methoxyphenyl)methyl]-4-[(2E)-3-phenylprop-2-en-1-yl]morpholine
1-methyl-4-{2-methyl-2-[1-methyl-3-(pyridin-3-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]propyl}piperazine
N-[4-(3-methylphenyl)phenyl]-1-(pyridine-4-carbonyl)piperidine-4-carboxamide
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-[5-oxo-2-(thiophen-2-ylmethyl)pyrrolidin-2-yl]propanamide
5-[6-hydroxy-4-(1H-1,2,3-triazol-4-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-pyrrole-3-carbonitrile
5-{[benzyl(methyl)amino]methyl}-N-{[1-(hydroxymethyl)cyclobutyl]methyl}-1,2-oxazole-3-carboxamide
2-{9-[(4-fluoro-3-methylphenyl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
1-(pent-2-yn-1-yl)-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1,4-diazepan-6-ol
2-methyl-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N3-(5-hydroxy-4,4-dimethylpentyl)-N1,N1-dimethylpiperidine-1,3-dicarboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-3-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-4-yl}propanamide
2-methoxy-N-methyl-5-[({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}carbamoyl)amino]benzamide
1-(5-chloropyridin-2-yl)-4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazine
(2S,4S)-4-amino-N-(2-methoxyethyl)-N-[(3-methoxyphenyl)methyl]-1-methylpyrrolidine-2-carboxamide
3-(1,2-dihydroacenaphthylene-5-carbonyl)-1-(furan-3-carbonyl)piperidine
3-[(1R,5R)-3-azabicyclo[3.3.1]nonan-3-ylmethyl]benzoic acid
(3aR,6aR)-2-[(2,4-dimethoxyphenyl)methyl]-5-methanesulfonyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
5-(3,5-difluorobenzoyl)-3-(phenoxymethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
[(3S,5R)-5-[(dimethylamino)methyl]-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]piperidin-3-yl]methanol
2-cyclopentyl-8-[2-(2-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(3-methoxypropyl)-4-(thiomorpholine-4-sulfonyl)benzamide
1-({3-[3-(azepan-1-yl)-2-hydroxypropoxy]phenyl}methyl)piperidine-4-carbonitrile
N-(1,3-benzoxazol-2-ylmethyl)-2-cyclohexyl-N-methyl-1,3-benzoxazole-6-carboxamide
1-ethyl-N-methyl-3-(2-methylpropyl)-N-(thian-4-yl)-1H-pyrazole-5-carboxamide
6-(3-chlorophenyl)-N-(1H-1,2,4-triazol-3-ylmethyl)imidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[(1-cyclopropyl-1H-imidazol-5-yl)methyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
4-(2,4-dichlorophenyl)-2-(methylsulfanyl)pyrimidine
1-(4-{5-cyclopropyl-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carbonyl}piperazin-1-yl)ethan-1-one
2-[4-(oxolan-2-ylmethyl)piperazin-1-yl]-1,3-benzoxazole
2-(2-aminopyrimidin-5-yl)-N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,8-dimethylquinoline-4-carboxamide
N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-5-propyl-1,2-oxazole-3-carboxamide
2-(dimethylamino)-N-({2-[(dimethylamino)methyl]phenyl}methyl)-2-(4-fluorophenyl)acetamide
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-3-methyl-4-oxo-3,4-dihydroquinazoline-7-carboxamide
2-methyl-5-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidine-1-carbonyl)pyrazine
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrazole-4-carbonyl)piperidine
N'1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N'1-methylcyclopropane-1,1-dicarboxamide