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2-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-1,2,3,4-tetrahydroisoquinolin-4-ol
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-(pyridin-3-yl)ethan-1-one
3-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
ethyl 1-[1-(2-cycloheptyl-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl)piperidine-4-carbonyl]piperidine-2-carboxylate
1-{3-[3-(2-methylphenyl)piperidin-1-yl]-3-oxopropyl}-1,2-dihydropyridin-2-one
(2S)-2-[({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amino]-3-phenylpropanamide
2-(4-{[(3R)-3-hydroxypyrrolidin-1-yl]methyl}phenyl)-6-(2-methyl-1,3-thiazol-4-yl)-3,4-dihydropyrimidin-4-one
N-[2-(1H-imidazol-4-yl)ethyl]-4-(piperidin-1-ylmethyl)benzamide
N-ethyl-6-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)amino)-N-methylpyridine-3-carboxamide
N-(1-{[3-(4-phenylphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)acetamide
1-[(4-fluoro-3-methoxyphenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
5-cyclobutyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1,3,4-oxadiazol-2-amine
N-(1-methylpyrrolidin-3-yl)-4-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
N-(3-methoxyphenyl)-3-[1-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperidin-4-yl]propanamide
5-[1-(4-methylpentanoyl)piperidin-4-yl]-5-(pyridin-3-yl)-3-[2-(thiophen-2-yl)ethyl]imidazolidine-2,4-dione
6-hydroxy-N-[(4-methyl-1,3-thiazol-2-yl)methyl]pyridine-3-carboxamide
N-[(2-amino-1,3-thiazol-4-yl)methyl]-N'-(2,4,6-trimethylphenyl)butanediamide
N-[1-(1H-imidazol-1-yl)butan-2-yl]-2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
(2R,6R)-11-methoxy-4-(propane-2-sulfonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N-(2,5-dimethoxyphenyl)-5-[4-hydroxy-1-(pyridin-2-ylmethyl)piperidin-4-yl]-1-benzofuran-2-carboxamide
3-[({3-[3-(1H-pyrazol-3-yl)phenyl]phenyl}methyl)amino]propan-1-ol
{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amine
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(3-fluorophenyl)ethan-1-one
1-[(4-chlorophenyl)methyl]-N-[(5-methylthiophen-2-yl)methyl]-6-oxopiperidine-3-carboxamide
(1R,9aR)-1-{[4-(thiophen-2-yl)-1H-imidazol-1-yl]methyl}-octahydro-1H-quinolizin-1-ol
2-(4-fluorophenyl)-N-(1H-imidazol-2-ylmethyl)imidazo[1,2-a]pyridine-6-carboxamide
6-[1-(methoxymethyl)cyclobutanecarbonyl]-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine
(4aS,7aR)-N-(4-chlorophenyl)-4-(cyclopropylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-(diphenylmethyl)-4-(1-methyl-1H-imidazole-5-carbonyl)piperazine
2-ethyl-9-(1-methyl-1H-pyrazole-5-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
5-(2-methoxyphenoxymethyl)-N-methyl-N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1H-pyrazole-3-carboxamide
3-methyl-1-propyl-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
[(3R,4S)-1-[(1-ethyl-1H-indol-4-yl)methyl]-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-5-ethyl-1,3,4-oxadiazol-2-amine
1-tert-butyl-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-5-oxopyrrolidine-3-carboxamide
3-(1H-imidazol-1-ylmethyl)-1-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]piperidine
2-(adamantan-1-yl)-N-methyl-N-propylacetamide
1-ethyl-3-[(3-methoxyphenyl)methyl]-8-{[1-(pyridin-3-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(benzenesulfonyl)-N-{1,9-dioxaspiro[5.5]undecan-4-yl}propanamide
N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(4aS,7aR)-1-(furan-2-carbonyl)-4-(3-methylbutanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(3-methoxyphenyl)amino]-N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]butanamide
3-(carbamoylmethoxy)-N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methylbenzamide
N-methyl-1-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}piperidine-2-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-6-(3-fluorophenyl)pyridine-3-carboxamide
3-(1-{[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-3-carbonyl)pyridine
5-methyl-2-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyrimidin-4-amine
1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}-2-(3-methoxypropyl)piperidine
N-[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]-4-hydroxy-2-(pyridin-3-yl)pyrimidine-5-carboxamide