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{4-fluoro-7-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
2-(2H-1,3-benzodioxol-5-yl)-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
8-(4-cyclopentylpyrimidin-2-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-5-phenylpentane-1,5-dione
2-[3-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-4-methylphenol
N-[(1r,4r)-4-hydroxycyclohexyl]-2-{tricyclo[9.4.0.03,8]pentadeca-1(11),3(8),4,6,12,14-hexaen-2-yl}acetamide
(1S)-2-cyclohexyl-1-[3-(2-methoxyethyl)-1-propyl-1H-1,2,4-triazol-5-yl]ethan-1-amine
1-(2,1,3-benzothiadiazol-5-ylmethyl)-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
1-(2-{[2-(5-butylthiophen-2-yl)-1H-imidazol-1-yl]methyl}morpholin-4-yl)ethan-1-one
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-2,4-dimethyl-1,3-oxazole-5-carboxamide
(2R,3R)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-3-methylpentanamide
[(1-cyclopentylpiperidin-4-yl)methyl][(3-ethoxyphenyl)methyl](oxolan-2-ylmethyl)amine
7-[(2,3-difluorophenyl)methyl]-2-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-2,7-diazaspiro[4.5]decane
N-[(5-ethylpyridin-2-yl)methyl]-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
{5-fluoro-7-[6-(trifluoromethyl)-1H-1,3-benzodiazol-4-yl]-2,3-dihydro-1-benzofuran-2-yl}methanamine
4-{3-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-N-methyl-1,3-thiazol-2-amine
methyl 5-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-3H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylate
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carboxamide
1-(2-methoxyethyl)-4-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperazine
N-methyl-4-{3-[(1S,5R)-6-methyl-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-3-oxopropyl}benzene-1-sulfonamide
2-(pyridin-2-ylsulfanyl)-1-[2-(pyridin-3-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]propan-1-one
4-{[2-(4-cyclohexylpiperazine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}morpholine
2-(1-{[1-(2H-1,3-benzodioxole-5-carbonyl)piperidin-3-yl]methyl}-1H-1,2,3-triazol-4-yl)propan-2-ol
3-cyclopropyl-N-{[3-(dimethylamino)thiolan-3-yl]methyl}-1H-pyrazole-5-carboxamide
2-({4-[3-(3-methylthiophene-2-carbonyl)piperidin-1-yl]piperidin-1-yl}methyl)pyridine
1-[(1-ethyl-1H-pyrazol-4-yl)methyl]-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-(2,3-dihydro-1H-inden-2-yl)-N-phenylpiperidin-3-amine
2-(2-hydroxyacetyl)-N-(1-phenylethyl)-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
(1R,6S)-9-methyl-3-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3,9-diazabicyclo[4.2.1]nonane
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-2-methoxy-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
(4aS,8aR)-1-[2-(cyclohex-1-en-1-yl)ethyl]-6-(pyrazin-2-yl)-decahydro-1,6-naphthyridin-2-one
(3aR,6aS)-1-oxo-2-(prop-2-en-1-yl)-5-(5-propyl-1,2-oxazole-3-carbonyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(5-propyl-1,2,4-oxadiazol-3-yl)-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}-2-(4H-1,2,4-triazol-4-yl)pyridine
3-[4-(5-{[(3-fluorophenyl)carbamoyl]amino}-1H-pyrazol-1-yl)piperidin-1-yl]propanamide
4-(hydroxymethyl)-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]benzamide
1-{[3-methyl-1-(1-methyl-2-oxo-1,2-dihydroquinolin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
5-ethyl-N4-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}pyrimidine-2,4-diamine
3-(5-methylthiophen-2-yl)-N-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
4-(1-{[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]methyl}azetidin-3-yl)pyridine
2-[4-(4-cyanophenyl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
2-methyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-{1-[2-(2,5,7-trimethyl-1H-indol-3-yl)acetyl]piperidin-4-yl}pyrrolidin-2-one
1-{2-[2-(3-ethyl-1,2-oxazol-5-yl)-1H-imidazol-1-yl]ethyl}-2,3-dihydro-1H-indole
3-(azetidine-1-carbonyl)-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}benzene-1-sulfonamide
2-({5-[(N-methylmethanesulfonamido)methyl]-4-(3-methylphenyl)-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
N-({5-[(2-chloro-4-fluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-methoxyacetamide
N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2,2-diphenylacetamide