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1-(1-benzylpiperidin-4-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]piperidine-3-carboxamide
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
4-chloro-5-{[4-(5,6-dimethylpyrimidin-4-yl)piperazin-1-yl]methyl}-N,N-dimethyl-1,3-thiazol-2-amine
2-amino-4-(3,4-dimethylphenyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
11-(2,1-benzoxazole-3-carbonyl)-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
[4-(2-methyl-1,2,3,4-tetrahydroisoquinoline-3-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
1-cyclopentanecarbonyl-N-[3-(4-fluorophenyl)propyl]piperidine-4-carboxamide
3-(5-methyl-1H-pyrazol-1-yl)-1-[(2R,3R,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]propan-1-one
N-[(3S,4R)-1-(3,4-difluorobenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
3-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)-1-{[1,2,4]triazolo[4,3-a]pyridin-8-yl}urea
1-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-3-[(dimethylamino)methyl]pyrrolidin-3-ol
methyl 1-[(3R,5S)-5-{[2-(3-chlorophenyl)ethyl]carbamoyl}-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
6-[(1R,3S)-1-hydroxy-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonane-7-carbonyl]-2-methyl-2,3-dihydropyridazin-3-one
3-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-1-[1-(1-phenylethyl)-1H-pyrazol-5-yl]urea
5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
3-chloro-N-{[1-(furan-2-ylmethyl)piperidin-3-yl]methyl}pyridine-4-carboxamide
4-ethyl-1-methyl-3-({1-[3-(pyrazin-2-yl)propanoyl]piperidin-4-yl}methyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[1-(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)azetidin-3-yl]-3,5-dimethyl-1H-pyrazole
(3aR,6aR)-2-(2-chlorobenzoyl)-5-(2-methoxyethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-ethyl-4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}pyrimidine
4-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-2-(pyridin-3-yl)morpholine
1-(2-methyl-1,3-thiazole-5-carbonyl)-3-(2-methylphenoxymethyl)piperidine
1-{3-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-oxopropyl}pyrrolidin-2-one
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-N-methyl-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
(2S,4S)-4-amino-1-[3-(2-chlorophenyl)propanoyl]-N-ethylpyrrolidine-2-carboxamide
N-(1-benzylpyrrolidin-3-yl)-3-[1-(thian-4-yl)piperidin-4-yl]propanamide
2-[4-(1-butyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-5-chlorophenol
4-(5-{[(2-methoxyethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoic acid
2-methoxy-4-[2-({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}amino)ethyl]phenol
[1-(1-benzofuran-2-ylmethyl)-4-[(2-chlorophenyl)methyl]piperidin-4-yl]methanol
dimethyl[2-(4-{octahydro-1H-pyrido[1,2-a]piperazin-2-ylmethyl}phenoxy)ethyl]amine
1-(5-methylpyridine-3-carbonyl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
7-[(3,4-difluorophenyl)methyl]-2-(2,3-dihydro-1H-inden-2-yl)-2,7-diazaspiro[4.5]decan-6-one
2-(2-methoxyphenoxy)-N-({1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]piperidin-3-yl}methyl)acetamide
methyl (2S)-1-{2-[(2-ethoxyphenyl)carbamoyl]ethyl}pyrrolidine-2-carboxylate
5-cyclohexaneamido-N-cyclohexyl-1-(2-methoxyethyl)-N-methyl-1H-1,3-benzodiazole-7-carboxamide
4-methoxy-N-{[1-(4-methylphenyl)pyrrolidin-3-yl]methyl}cyclohexane-1-carboxamide
2-(dimethyl-1,3-thiazol-5-yl)-1-(4-methanesulfonyl-1,4-diazepan-1-yl)ethan-1-one
2-propyl-8-(thiophen-3-ylmethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-methyl-4-({2-[3-(1H-pyrazol-1-yl)phenoxy]phenyl}methyl)piperazine
5-(4-methanesulfonylphenyl)-1,3-benzothiazol-2-amine
2-[3-(1H-pyrazol-3-yl)phenyl]benzene-1-sulfonamide
N-cyclopentyl-2-[4-methyl-6-(pyrrolidine-1-carbonyl)-3,4-dihydro-2H-1,4-benzoxazin-2-yl]acetamide
N-[(3-methyl-7-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(methylsulfanyl)benzamide
1-(4-chlorophenyl)-N-{[1-(3-phenylprop-2-yn-1-yl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
1-[3-(2-fluorophenoxymethyl)piperidin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-(oxolane-3-carbonyl)piperidine
2-(azepan-1-yl)-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]acetamide
(7R,8aS)-7-[(6-ethylpyrimidin-4-yl)amino]-2-methyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione