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2-[4-({[3-(4-fluorophenyl)oxolan-3-yl]methyl}amino)phenyl]acetonitrile
4-methoxy-N-(1-{1-[(2-oxo-1,3-oxazolidin-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)benzamide
2-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
1-[2-(1H-imidazol-1-yl)propyl]-4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1H-1,2,3-triazole
3-[1-(6,7-dimethoxy-4-methylquinolin-2-yl)piperidin-3-yl]propanamide
1-{1-[(2-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(3-methoxyphenyl)piperazine
methyl 2-[(2,3-dihydro-1H-inden-5-yl)sulfamoyl]-6-[(2E)-2-methylbut-2-enoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4,6-dimethyl-3-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
5-(1-methyl-5-phenyl-1H-pyrrol-2-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2,2,3-trimethylbut-3-en-1-one
3-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(2,4-dimethoxyphenyl)propanamide
5-cyano-N,4-dimethyl-6-oxo-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}-1,6-dihydropyridine-3-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]-2-(3,4-dimethylphenoxy)ethan-1-one
N-(2H-1,3-benzodioxol-5-yl)-8-(2-methoxyethyl)-9-oxo-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-(2,6-dimethylphenyl)-3-({[1-(furan-2-yl)ethyl](methyl)amino}methyl)benzamide
N-{[1-(dimethylamino)cycloheptyl]methyl}-4-hydroxy-2-phenylpyrimidine-5-carboxamide
1-[1-(2-amino-2-methylpropanoyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)piperidine-3-carboxamide
4-[(4aS,8aR)-1-butyl-2-oxo-decahydro-1,6-naphthyridin-6-yl]-4-oxobutane-1-sulfonamide
1-{4-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carbonyl]-3,5-dimethyl-1H-pyrrol-2-yl}ethan-1-one
3-ethyl-N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-4-methyl-1H-pyrazole-5-carboxamide
7-(2,1,3-benzoxadiazol-4-ylmethyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
6-ethoxy-2-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]quinoline
N-[1-(2-methanesulfonylethyl)piperidin-4-yl]-3-phenyl-1H-pyrazole-4-carboxamide
N4,N4-dimethyl-N6-[2-(pyridin-2-yl)ethyl]pyrimidine-4,6-diamine
N-[(5-methylthiophen-2-yl)methyl]-2-(morpholin-2-yl)-N-(pyridin-4-ylmethyl)acetamide
N-methyl-3-(4-methyl-1,3-thiazol-5-yl)-N-[2-(phenylsulfanyl)ethyl]propanamide
2-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
1-(3-cyanophenyl)-3-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}urea
2-(dimethyl-1,2-oxazol-4-yl)-1-[9-hydroxy-7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethan-1-one
1-{5,6-dimethylthieno[2,3-d]pyrimidin-4-yl}-N-[(2-methyl-1,3-thiazol-4-yl)methyl]piperidin-4-amine
(4-{[(5-ethyl-2-methylpyrimidin-4-yl)(methyl)amino]methyl}oxan-4-yl)methanol
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]pyrrolidin-2-one
4-[4-(hydroxymethyl)-1H-1,2,3-triazol-1-yl]-N-(2-phenylphenyl)piperidine-1-carboxamide
1-[3-(2-oxopyrrolidin-1-yl)propyl]-5-[2-({[3-(trifluoromethyl)phenyl]methyl}amino)ethyl]pyrrolidin-2-one
2-[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
5-oxo-1-[2-(4-phenylpiperidin-1-yl)ethyl]pyrrolidine-3-carboxylic acid
N-[(1S,2R,4R)-bicyclo[2.2.1]heptan-2-yl]-5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carboxamide
N-[2-(dimethylamino)ethyl]-2-methyl-N-[(5-methylthiophen-2-yl)methyl]-1,3-thiazole-4-carboxamide
[(3-{[1-(3-chlorobenzoyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(2-phenylethyl)amine
3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)-N-[1-(thiophen-3-yl)propan-2-yl]propanamide
N4-cyclopropyl-6-(3-fluorophenyl)pyrimidine-2,4-diamine
3-(1H-indol-6-yl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
N-ethyl-6-methyl-5-[5-(4-methylphenyl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine-2-carboxamide
5-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
N-[(6-chloropyridin-3-yl)methyl]-N-methyl-3-(1-methylpiperidin-2-yl)propanamide
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridine-3-carboxamide
3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]-4-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-one
{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]methylamine
2-(2-aminoethyl)-N-methyl-N-[2-(pyrrolidin-1-ylmethyl)propyl]quinazolin-4-amine
1-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)amino}ethyl)-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide