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N-[(5-fluoro-2-methylphenyl)methyl]-2-(3-methoxyphenoxymethyl)-1,3-oxazole-4-carboxamide
(5-{[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]methyl}-2-(propan-2-yloxy)phenyl)methanol
N-[(2-{4-[(methylcarbamoyl)amino]phenyl}phenyl)methyl]propanamide
2-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-1-(morpholin-4-yl)ethan-1-one
3,3-dimethyl-1-[(6-methylpyridin-2-yl)methyl]-4-(morpholin-4-ylmethyl)piperidin-4-ol
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
(3S,4R)-1-[2-(morpholin-4-yl)ethyl]-4-phenylpyrrolidine-3-carboxylic acid
4-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-1-oxaspiro[4.5]decan-2-one
2-amino-6-(3,5-difluorophenyl)-4-(1-ethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
1-{[2-(butan-2-ylsulfanyl)pyrimidin-5-yl]methyl}-4-(pyridin-2-ylmethyl)-1,4-diazepane
7-(cyclobutylmethyl)-2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide
4-(4-chlorophenyl)-1-[(3R,5R)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]butan-1-one
4-[4-(3,5-difluorophenyl)-1H-1,2,3-triazol-1-yl]-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidine
3-[3-(1H-imidazol-2-yl)piperidin-1-yl]-6-methylpyridazine
5-[4-(2,3-dimethylphenyl)piperazine-1-carbonyl]-1-[(2-fluorophenyl)methyl]piperidin-2-one
1-cyclopentyl-5-oxo-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrrolidine-3-carboxamide
1-(2,3-dihydro-1H-inden-2-yl)-4-{1-[2-(morpholin-4-yl)ethyl]-1H-1,2,3-triazole-4-carbonyl}-1,4-diazepane
1,3-dimethyl-8-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2-phenylacetamide
1-(2-{7,7-dimethyl-4-oxo-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-2-yl}ethyl)piperidine-3-carboxamide
6-methoxy-1-methyl-2-[4-(thian-4-yl)piperazine-1-carbonyl]-1H-indole
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4,4-difluoropiperidine
methyl 4-[2-amino-3-cyano-5-methyl-6-(4-methylphenyl)pyridin-4-yl]-1H-pyrazole-3-carboxylate
12-[3-ethyl-4-(propan-2-yl)piperazine-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-5-methyl-2-phenyl-1H-imidazole-4-carboxamide
N-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-1-{[3-(trifluoromethyl)phenyl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-methyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
2-methyl-2-[4-(morpholin-4-yl)-2-{[2-(pyrrolidin-1-yl)ethyl]amino}pyrimidin-5-yl]propanoic acid
N-(3-methoxypropyl)-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-[2-(ethanesulfonyl)ethyl]-4-methyl-3-phenyl-1H-pyrazole-5-carboxamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[4-methyl-6-(methylamino)pyrimidin-2-yl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[2-(dimethylamino)ethyl]-3,4-dimethyl-N-[(5-methylthiophen-2-yl)methyl]benzamide
1-[(2-methyl-1H-imidazol-4-yl)methyl]-3-[2-(methylsulfanyl)benzoyl]piperidine
2-(dimethylamino)-N-[3-(4-methoxyphenoxy)propyl]-N,4-dimethylpyrimidine-5-carboxamide
dimethyl[(4-{1-[2-(pyridin-2-yl)ethyl]piperidin-2-yl}phenyl)methyl]amine
(2S,4R)-4-amino-N,N-diethyl-1-[2-(3-methoxyphenoxy)acetyl]pyrrolidine-2-carboxamide
1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-{2-[3-(naphthalen-1-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}morpholine
(2S,4R)-4-amino-N-ethyl-1-[2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetyl]pyrrolidine-2-carboxamide
N-benzyl-2-(6-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carboxamide
8-(4-chloro-2-hydroxybenzoyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
[(6,7-dimethyl-1H-1,3-benzodiazol-2-yl)methyl][2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amine
5-oxo-1-(propan-2-yl)-N-{[3-(trifluoromethoxy)phenyl]methyl}pyrrolidine-3-carboxamide
2-[5-(oxolan-3-yl)-4-phenyl-1H-imidazol-1-yl]acetic acid
1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}-3-(1,2-oxazolidin-2-yl)propan-1-one
9-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-2-(2-methoxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[(2-{[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]methyl}phenyl)methyl]pyrrolidin-2-one
2-cyclopropyl-8-{[5-(3-fluorophenyl)-1,3,4-oxadiazol-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one