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1-cyclopentyl-N-ethyl-4-oxo-5-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazine-1-carbonyl}-1,4-dihydropyridine-3-carboxamide
N-{[4-amino-6-(dimethylamino)-1,3,5-triazin-2-yl]methyl}-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
2-(3-chlorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
5-chloro-3-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
1-[(3-chlorophenyl)methyl]-4-(oxolan-3-ylmethyl)piperazine
1-[5-(oxolan-2-yl)thiophene-2-carbonyl]-2-phenylpyrrolidine
2-({3-[3-(4-methanesulfonylphenyl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-propylacetamide
(2R)-2-acetamido-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}butanamide
4-{3-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]propoxy}benzamide
8-(2-amino-6-methylpyrimidin-4-yl)-2-[(3,5-difluorophenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
2-(cyclopropylmethyl)-9-[(2-ethylpyrimidin-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-2-oxo-1,2-dihydroquinazoline-4-carboxamide
2-{5-methyl-2-oxo-4-[(3,4,5-trimethoxyphenyl)methyl]piperazin-1-yl}benzonitrile
2-(2-fluoro-4-methylphenyl)-N,N-dimethylpyridine-3-carboxamide
2-{1-[3-(5-methylfuran-2-yl)butyl]azetidin-3-yl}pyridine
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-(pyridine-3-carbonyl)pyrrolidin-3-yl]methanol
4-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonane-7-carbonyl]-1,2-dihydroisoquinolin-1-one
N-(1H-imidazol-2-ylmethyl)-6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-amine
5-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]pyridine-2-carbonitrile
3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-N-{[3-(trifluoromethyl)phenyl]methyl}propanamide
4-{[2-(4-fluorophenyl)azetidin-1-yl]methyl}-3,5-dimethyl-1H-pyrazole
6-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]pyridine-3-carbonitrile
N-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,3-dihydro-1H-indene-5-carboxamide
3-[(4aR,7aS)-4-(4-methylpiperazine-1-carbonyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
(4aS,7aR)-1-(2-methoxyquinoline-4-carbonyl)-4-methyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[2-(pyridin-3-yl)-4-{[2-(pyrrolidin-1-yl)ethyl]amino}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
(1s,4s)-4-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]cyclohexan-1-ol
1-{2-[2-(2-methyl-1,3-oxazol-4-yl)-1H-imidazol-1-yl]propyl}-1H-indole
N-{1-[1-(cyclohex-1-ene-1-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
6-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}-2H-1,3-benzodioxole-5-carboxamide
4-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-1-[(3-fluorophenyl)methyl]piperazin-2-one
2-(dimethyl-1,2-oxazol-4-yl)-N-{2-[2-(thiophen-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}acetamide
(4aS,8aR)-6-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-1-(3-hydroxypropyl)-decahydro-1,6-naphthyridin-2-one
2-[1-(3-methylbutyl)-4-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperazin-2-yl]ethan-1-ol
1-(2-hydroxyethyl)-5-[(3-hydroxyphenyl)methyl]-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-[(3-fluorophenyl)methyl]-1-(1-phenyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one
1-[(2-fluorophenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,4-diazepane
2-methyl-5-(propan-2-yl)-N-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
5-{3-[4-(2,3-dihydro-1H-inden-2-yl)piperazin-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
[(3R,4R)-1-(2-methoxypyridine-4-carbonyl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzamide
2-methoxy-5-oxo-6-{3-[(pyridin-3-yl)amino]propyl}-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
N-[(1-methylpyrrolidin-3-yl)methyl]-2-[4-(methylsulfanyl)phenyl]acetamide
3-cyclopropyl-1-(4-{2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}phenyl)urea
2-cyclopropyl-5-{4-[(4-methylphenyl)methyl]-3-oxopiperazine-1-carbonyl}-3,4-dihydropyrimidin-4-one
N-[(3S,5S)-1-cyclopentyl-5-(ethylcarbamoyl)pyrrolidin-3-yl]pyridine-3-carboxamide
5-(2-ethylphenyl)-4-(4-methylphenyl)-2-(4-methylpiperazin-1-yl)pyrimidine