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N-methyl-N-(1-{5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}pyrrolidin-3-yl)acetamide
1-methyl-8-[(5-methylthiophen-2-yl)methyl]-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[(3R,4S)-4-cyclopropyl-1-[(methylcarbamoyl)methyl]pyrrolidin-3-yl]-3-methoxy-4-methylbenzamide
1-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carbonyl}-1,4-diazepane
(5S)-5-[({[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(pyridin-4-ylmethyl)amino)methyl]pyrrolidin-2-one
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
methyl 3-[(furan-2-ylformamido)methyl]-5-(2-phenylacetamido)benzoate
2-{4-[(1-ethyl-1H-pyrazol-4-yl)methyl]-1-(thiophen-3-ylmethyl)piperazin-2-yl}ethan-1-ol
(2S)-1-(pyrazine-2-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]pyrrolidine-2-carboxamide
2-(3-hydroxypropyl)-9-[4-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
1-(butan-2-yl)-N-(furan-2-ylmethyl)-4-oxo-5-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1,4-dihydropyridine-3-carboxamide
1-[(2-chloro-4-fluorophenyl)methyl]-N-methyl-N-[(5-phenyl-1H-pyrazol-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
methyl 2-[ethyl(2-methylprop-2-en-1-yl)sulfamoyl]-6-(3-methoxybenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-3-fluoro-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
5-[(1-butyl-3-methyl-1H-1,2,4-triazol-5-yl)methyl]-2-ethyl-6-methyl-3,4-dihydropyrimidin-4-one
3-[(dimethylamino)methyl]-1-[3-(4-hydroxyphenyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-ol
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(2,4-dioxo-1,3-diazinan-1-yl)benzamide
5-{[(4-methylphenyl)methyl]amino}-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
4-[(3S)-3-ethylmorpholine-4-carbonyl]-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-2,3-dihydro-1H-isoindol-1-one
4-(2-chlorophenyl)-3-[1-(1H-pyrazol-1-yl)ethyl]-4H-1,2,4-triazole
1-ethyl-4-[(4-methyl-6-phenylpyrimidin-2-yl)methyl]piperazine-2,3-dione
N-{[3-methyl-7-(9-methyl-9H-carbazole-3-carbonyl)-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}methanesulfonamide
1-cyclohexanecarbonyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrrolidine-2-carboxamide
N-methyl-3-(piperidin-3-yl)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}benzamide
N-ethyl-N-[2-(phenylsulfanyl)ethyl]quinoxaline-5-carboxamide
1-(4-acetylpiperazin-1-yl)-2-{4-[(2E)-3-phenylprop-2-en-1-yl]morpholin-3-yl}ethan-1-one
1-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-(naphthalen-2-yl)piperazine
N-[(1S,2S)-1-amino-2,3-dihydro-1H-inden-2-yl]-5-(2-chlorophenyl)furan-2-carboxamide
3-[3-(2-methoxyphenyl)-1,2,4-oxadiazol-5-yl]-N-[3-(morpholin-4-yl)propyl]propanamide
2-[(5-{[propyl(pyridin-3-ylmethyl)amino]methyl}pyrimidin-2-yl)amino]acetic acid
3-[2-(ethylsulfanyl)ethyl]-1-[3-(4-methylpiperidine-1-carbonyl)phenyl]urea
2-[(3,5-difluorophenyl)methyl]-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-(2-chlorophenyl)-2-{[1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}ethan-1-ol
[5-({cyclopentyl[(3-methylthiophen-2-yl)methyl]amino}methyl)furan-2-yl]methanol
(3aS,6aS)-N-(2H-1,3-benzodioxol-5-yl)-1-(pyridin-2-ylmethyl)-octahydropyrrolo[2,3-c]pyrrole-5-carboxamide
4-(2-amino-6-methoxypyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
2-{1-[1-(2-phenylethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
3-[1-(furan-3-carbonyl)piperidin-4-yl]-1-(pyrrolidin-1-yl)propan-1-one
N-benzyl-N-methyl-3-{[(oxan-4-yl)amino]methyl}pyridin-2-amine
dimethyl({[4-methyl-5-(1-{6-methylimidazo[2,1-b][1,3]thiazole-5-carbonyl}piperidin-4-yl)-4H-1,2,4-triazol-3-yl]methyl})amine
3-(3-hydroxy-3-methylbutyl)-N-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]benzamide
2-methoxy-N-[(4-methoxyphenyl)methyl]-N-propylpyrimidine-5-carboxamide
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(pyridin-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[3-hydroxy-3-(hydroxymethyl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
N-[2-(furan-2-yl)ethyl]-4,5,6,7-tetrahydro-2H-indazole-3-carboxamide
N-tert-butyl-5-[4-(2-chlorophenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
1-(propan-2-yl)-N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-4-carboxamide
N-(3,5-dimethoxyphenyl)-2-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}acetamide