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(3R,4R)-4-[4-(2-fluorophenyl)piperazin-1-yl]-1-{[4-(methylsulfanyl)phenyl]methyl}piperidin-3-ol
(3S,4S)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-4-(propan-2-yloxy)pyrrolidin-3-ol
2-(3,4-dimethoxyphenyl)-5-fluoro-1-{1-[5-(methoxymethyl)furan-2-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
6-methyl-2-(3-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}phenyl)-3,4-dihydropyrimidin-4-one
1-[2-(1,3-benzoxazol-2-yl)ethyl]-3-(5-ethyl-1-methyl-1H-1,2,4-triazol-3-yl)urea
N-[(3-chloro-4-fluorophenyl)methyl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
(3S,4R)-4-(3-methoxyphenyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidine-3-carboxylic acid
2-(5-acetylthiophen-3-yl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-5-[(dimethylamino)methyl]furan-2-carboxamide
1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-3-(1H-imidazol-2-yl)piperidine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-5-propyl-1,2-oxazole-3-carboxamide
N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-6-(pyridin-3-yl)pyridine-3-carboxamide
(3S,4S)-3-hydroxy-4-{[6-(propan-2-yl)pyrimidin-4-yl]amino}-1λ6-thiolane-1,1-dione
5-(2-ethylpiperidine-1-carbonyl)-1-[(5-methylfuran-2-yl)methyl]-4-oxo-N-(prop-2-en-1-yl)-1,4-dihydropyridine-3-carboxamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-2-(4-phenylphenyl)acetamide
5-{[3-hydroxy-2-oxo-1-(2-phenylethyl)piperidin-3-yl]methyl}-N-methyl-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[1-(2-methoxyphenyl)ethyl]-N-methyl-2-{8-methyl-3-oxo-2,8-diazaspiro[4.5]decan-2-yl}acetamide
4-{3-[2-(2-fluorophenyl)ethyl]piperidine-1-carbonyl}-2-methyl-1H-1,3-benzodiazole
2-{1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]piperidin-3-yl}-6,7-dimethoxy-1,2,3,4-tetrahydroisoquinoline
2-[(3,4-difluorophenyl)methyl]-8-[(1-methyl-1H-imidazol-5-yl)methyl]-2,8-diazaspiro[4.5]decan-3-one
benzyl[(4-methyl-1,3-thiazol-5-yl)methyl](pyridin-4-ylmethyl)amine
1-[6-ethyl-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-N-[2-(pyridin-2-yl)ethyl]piperidin-4-amine
[2-(1H-imidazol-1-yl)ethyl](methyl)[(2E)-3-phenylprop-2-en-1-yl]amine
(2r,4r)-2-[(2R,3S,6R)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-5,7-diazaspiro[3.4]octane-6,8-dione
N-cyclopropyl-1-{1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]piperidin-4-yl}piperidine-3-carboxamide
3-chloro-5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2-dihydropyridin-2-one
4-(4-methanesulfonylphenoxymethyl)-5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazole
4-(1-phenyl-1H-pyrazol-4-yl)-N-[4-(1H-pyrazol-1-yl)butan-2-yl]pyrimidin-2-amine
5-(2-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-oxoethyl)imidazolidine-2,4-dione
1-{4-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]piperidin-1-yl}-2-methylpropan-1-one
2-(3-hydroxypropyl)-9-[3-(4-methylphenyl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(5-methoxypyridin-3-yl)-1H-pyrazol-1-yl]acetamide
3-methyl-N-{2-[2-(oxolan-3-yl)-1H-imidazol-1-yl]ethyl}pyridin-4-amine
1-[2-(4-chlorophenyl)quinoline-4-carbonyl]-4-ethyl-1,4-diazepan-5-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-methylpropanamide
1-(1-methylpiperidin-4-yl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperidine-3-carboxamide
2-methoxy-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-N-[(5-methylthiophen-2-yl)methyl]-N-(prop-2-en-1-yl)acetamide
N,1-dimethyl-N-[2-(oxan-4-yl)ethyl]-6-(propan-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
methyl[3-(phenylsulfanyl)propyl]{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}amine
4-methoxy-N-({4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)benzamide
{[2-(methoxymethyl)-4-methyl-1,3-thiazol-5-yl]methyl}({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl})amine
N-(2-ethoxyethyl)-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-benzyl-8-(2-methyl-1H-pyrrole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
(3S)-4-[6-(benzylamino)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]-1,3-dimethylpiperazin-2-one
N-(2,6-dimethylphenyl)-3-[2-(2-methoxyphenoxy)acetamido]benzamide
1-(5-propyl-1,2,4-oxadiazol-3-yl)-4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidine
2-(dimethyl-1,2-oxazol-4-yl)-2-{methyl[(5-propyl-1H-pyrazol-3-yl)methyl]amino}acetic acid
N-[phenyl(pyridin-2-yl)methyl]-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
1-[2-(5-amino-1H-1,2,4-triazol-3-yl)ethyl]-5-methyl-5-phenylpiperidin-2-one