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1-(3-cyanophenyl)-3-{[1-(methoxymethyl)cyclopentyl]methyl}urea
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1-(pyridine-2-carbonyl)piperidin-4-amine
4-[6-(morpholin-4-yl)pyrimidin-4-yl]-2-(trifluoromethyl)morpholine
4'-[2-(propan-2-ylsulfanyl)ethyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
5-butyl-1-(3-chlorophenyl)-4-(1,3-thiazole-4-carbonyl)piperazin-2-one
N-methyl-5-{1H-pyrrolo[2,3-b]pyridin-4-yl}furan-2-carboxamide
N-[1-(3-phenylpropyl)piperidin-3-yl]quinoxalin-2-amine
3-{2-[1-(4-methylpiperazine-1-carbonyl)piperidin-2-yl]ethyl}phenol
2-(2,5-dioxoimidazolidin-1-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
N-(1-methanesulfonylpiperidin-4-yl)-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
(3R,4S)-1-[(2,6-difluoro-4-methoxyphenyl)methyl]-3,4-dimethylpiperidin-4-ol
N-(2-fluorophenyl)-3-{1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperidin-3-yl}propanamide
(3aS,7aR)-5-methyl-2-[2-(trifluoromethyl)benzoyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-(2-ethylpyridine-4-carbonyl)piperidin-3-ol
N-{5-[(9aS)-octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl]-2-methylphenyl}cyclopropanecarboxamide
(3S,4R)-1-(cyclopropylmethyl)-N,N-dimethyl-4-(4-methylphenyl)pyrrolidin-3-amine
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-N-methyl-2-(2-oxoazonan-1-yl)acetamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[1-(oxan-4-yl)piperidin-3-yl]piperazine
8-[(2S,4R)-4-hydroxypyrrolidine-2-carbonyl]-2-[(3-methoxyphenyl)methyl]-2,8-diazaspiro[4.5]decan-3-one
N-(adamantan-2-ylmethyl)-1-[2-(1,1-dioxo-1λ6-thiolan-3-yl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-3-carboxamide
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-[(2-methylphenyl)sulfanyl]piperidine
N-(4-methoxyphenyl)-1-{2-[2-(2-methoxyphenyl)acetamido]ethyl}-1H-1,2,3-triazole-4-carboxamide
3-(4-fluorophenyl)-N-[(1R,2S)-2-phenylcyclopropyl]-1H-pyrazole-5-carboxamide
(1S,6R)-9-(4-phenyl-1,3-thiazole-2-carbonyl)-3,9-diazabicyclo[4.2.1]nonan-4-one
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
N-[4-(2-methyl-1H-imidazol-1-yl)phenyl]-1-(thian-4-yl)piperidine-3-carboxamide
[(1-methylpiperidin-4-yl)methyl](2-phenylethyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
3-[4-(2-carboxyethyl)phenyl]-5-(pyrrolidine-1-sulfonyl)benzoic acid
1-(1-benzofuran-5-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
1-benzyl-5-(cyclohexylamino)-N,N-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
5,7-dimethyl-N-{1-oxaspiro[4.4]nonan-3-yl}pyrido[2,3-d]pyrimidin-4-amine
(4aS,7aR)-1-{[4-(propan-2-yl)phenyl]methyl}-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-cyclopropyl-N-{[2-(3-methoxyphenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}furan-2-carboxamide
5-(4-methylpiperazine-1-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
1-cyclopentyl-3-(2-methylphenyl)-3-{2-[4-(morpholin-4-yl)piperidin-1-yl]-2-oxoethyl}pyrrolidine-2,5-dione
3-(hydroxymethyl)-1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
3-[(cyclobutylamino)methyl]-1-[(4-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
1-methyl-4-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
N-[(3-fluorophenyl)methyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-4-(5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carbonyl)piperazine
(3S,4S)-1-({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)-4-methylpiperidine-3,4-diol
2-methyl-N-{1-[1-(3-methylbut-2-en-1-yl)piperidin-4-yl]-1H-pyrazol-5-yl}benzamide
5-amino-4-chloro-N-[2-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide
1-[5-(ethanesulfonyl)thiophen-2-yl]-1H-1,3-benzodiazole
2-{1-[(4-ethoxyphenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[2-(2-methoxyphenyl)ethyl]-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-3-(5-fluoro-1H-1,3-benzodiazol-2-yl)propanamide
1-{5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(1H-pyrazol-1-yl)ethan-1-one
N-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}methanesulfonamide