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N6-cyclopentyl-N5-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N5-methyl-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
(2R,6R)-4-[3-(pyrazin-2-yl)propanoyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
N,N-dimethyl-2-({1-[1-(2-phenylethyl)piperidin-4-yl]piperidin-3-yl}formamido)acetamide
N-(1-benzyl-1H-pyrazol-3-yl)-2-[4-(4,6-dimethylpyrimidin-2-yl)-1H-pyrazol-1-yl]acetamide
5-[({1,9-dioxaspiro[5.5]undecan-4-yl}amino)methyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-[(3-hydroxyphenyl)methyl]-N-[3-(1H-indol-2-yl)phenyl]piperidine-4-carboxamide
2-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-3-(1H-pyrazol-1-yl)propanamide
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(7-hydroxyquinolin-3-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-4-[5-(1H-pyrazol-3-yl)thiophen-2-yl]-3-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
{[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazol-4-yl]methyl}(1-methoxypropan-2-yl)amine
3-{[(1H-1,3-benzodiazol-2-ylmethyl)(methyl)amino]methyl}-1-(cyclopropylmethyl)-3-hydroxypiperidin-2-one
N-(cyclohex-1-en-1-ylmethyl)-2-[2-(1-methyl-1H-imidazol-4-yl)ethyl]-1-oxo-2,3-dihydro-1H-isoindole-4-carboxamide
(2S)-1-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(methylamino)pentan-1-one
1-(4-ethoxy-3-methylphenyl)-4-(4-hydroxy-1,2,3,4-tetrahydroisoquinolin-2-yl)butane-1,4-dione
2-{[6-(2,3-dimethoxy-5-methylphenyl)quinazolin-4-yl]amino}ethan-1-ol
2-{[(1-{[2-(trifluoromethoxy)phenyl]methyl}piperidin-4-yl)oxy]methyl}pyridine
1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pentan-1-one
1-[1-(cyclopropylmethyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-cyclopentyl-4-methoxy-N-{[4-methoxy-3-(thiophen-2-ylmethoxy)phenyl]methyl}benzene-1-sulfonamide
(3S,4S)-4-[4-(pyridin-2-yl)piperazin-1-yl]-1-{thieno[3,2-d]pyrimidin-4-yl}pyrrolidin-3-ol
1-({[2-(2-chlorophenyl)-2-hydroxyethyl]carbamoyl}methyl)piperidine-4-carboxamide
N-[2-(3-methylpyridin-2-yl)ethyl]-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
3-{1-[3-(hydroxymethyl)-8-methylquinolin-2-yl]piperidin-3-yl}-N,N-dimethylpropanamide
(4aR,7aS)-1-acetyl-4-[(5-hydroxy-2-methoxyphenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-{[(3S,4S)-1-[(3-chloro-4-ethoxyphenyl)methyl]-3-hydroxypiperidin-4-yl]methyl}acetamide
propan-2-yl 4-[(3-methoxyphenyl)methyl]-1-methyl-1,4,9-triazaspiro[5.5]undecane-9-carboxylate
N-[(4-fluorophenyl)methyl]-N-(pyridin-4-ylmethyl)morpholine-2-carboxamide
5-{[(3-cyclopropyl-1,2,4-oxadiazol-5-yl)methyl](methyl)amino}-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
(butan-2-yl)[(2-methyl-2H-indazol-3-yl)methyl](pyridin-4-ylmethyl)amine
2-[4-(5-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]acetic acid
N-[(2-chlorophenyl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N,N-diethyl-1-{1-[(2-hydroxy-5-methoxyphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-3-(pyridin-2-yl)-1H-pyrazole-5-carboxamide
1-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-3-(1,3,6-trimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)urea
N,N-diethyl-5-methyl-4-{[(6-methylpyridin-2-yl)methyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
ethyl 4-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazine-1-carboxylate
3-[(3S,7S,8aS)-3-[(4-chlorophenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-chlorophenyl)urea
(3aS,6aS)-2-[(5-methylthiophen-2-yl)methyl]-5-(pyridin-3-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-benzyl-3-ethyl-1-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one
N-{[5-(cyclohexylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}-2-methoxyacetamide
4-hydroxy-N-(4-methoxy-2-methylphenyl)-4-(5-methylpyridin-2-yl)piperidine-1-carboxamide
1-(3-fluoro-5-methylphenyl)-3-{[1-(4-methylpiperazin-1-yl)cyclopentyl]methyl}urea
methyl 2-(cyclopropylsulfamoyl)-6-[(3,4-dimethylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2,3-dimethyl-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-2-(5-methyl-1,2-oxazol-3-yl)piperidine-1-carboxamide
4-chloro-5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-1,3-dimethyl-1H-pyrazole
2-cyclopropyl-9-(6-oxo-1,6-dihydropyridine-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-benzyl-N-[(6-methylpyridin-2-yl)methyl]-5-propyl-1,2-oxazole-3-carboxamide
[2-(2-ethylphenoxy)ethyl][2-(1H-imidazol-4-yl)ethyl]amine
N-{[4-(cyclobutylmethoxy)phenyl]methyl}-N-cyclopropyl-2-(pyridin-2-ylsulfanyl)acetamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(phenylsulfanyl)ethan-1-one