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N-(cyclopropylmethyl)-N-propyl-5-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]pyridin-2-amine
1-[(4aR,8aR)-7-[3-(4-fluorophenoxy)propyl]-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]-2-methoxyethan-1-one
1-cyclopropyl-N-methyl-6-oxo-N-{[4-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
3-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-1-[3-(thiophene-2-carbonyl)piperidin-1-yl]propan-1-one
N-({2-[(dimethylamino)methyl]phenyl}methyl)-1-(5-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
2-{4-[4-methyl-5-(morpholin-4-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine-4-carbonitrile
(1S,6R)-9-[5-(2-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-methyl-3,9-diazabicyclo[4.2.1]nonane
6-fluoro-2-{[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]methyl}quinoline
1-{4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyridin-4-ylsulfanyl)ethan-1-one
5-{1-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-1H-imidazol-2-yl}-1-ethyl-1H-1,2,4-triazole
2-(2,4-dichlorophenoxy)-1-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]ethan-1-one
(4S)-1-[(4-fluoro-3-methoxyphenyl)methyl]-4-(methoxymethyl)-3,3-dimethylpiperidin-4-ol
1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-2-(methylsulfanyl)ethan-1-one
4-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}-1,4-oxazepan-6-ol
N-{1-[(cyclopropylcarbamoyl)methyl]piperidin-4-yl}-2-(2,3-dihydro-1H-inden-1-yl)acetamide
N-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)-1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazole-5-carboxamide
1,5,6-trimethyl-N-{1-[5-methyl-1-(2-methylphenyl)-1H-pyrazol-4-yl]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
2-(4-fluorophenyl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]morpholine
N-[3-(pyridin-4-yl)propyl]-4-sulfamoylbenzamide
6-methyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
5-(1-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
(2S)-2-amino-1-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-3-hydroxypropan-1-one
5-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-{1-[5-(3-benzyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]piperidin-4-yl}ethan-1-ol
(4aS,7aR)-1-(6-methyl-4-oxo-1,4-dihydropyridine-3-carbonyl)-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-ethyl-N-{[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]methyl}pyrimidin-4-amine
2-[3-(2-fluorophenyl)-1,2,4-oxadiazol-5-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(furan-3-ylmethyl)(methyl)[(1-phenylpyrrolidin-3-yl)methyl]amine
1-(piperidin-3-ylmethyl)-N-[2-(pyrazin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
1-[1-({1-[(2-aminopyridin-3-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]cyclopentan-1-ol
1-(2-cyclopentylacetyl)-4-(cyclopropylmethyl)-1,4-diazepan-5-one
5-methyl-4-[(2-methylpyridin-3-yl)oxy]-6-[3-(pyrrolidine-1-carbonyl)piperazin-1-yl]pyrimidine
3-{4-[5-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl]phenyl}prop-2-yn-1-ol
(3S,7S)-5-(1,2-oxazole-3-carbonyl)-9-oxa-5-azatricyclo[8.4.0.03,7]tetradeca-1(10),11,13-triene-3-carboxylic acid
5-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
6-(4-hydroxyphenyl)-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}pyridine-3-carboxamide
3-({1-[4-(1H-pyrazol-1-yl)butanoyl]pyrrolidin-3-yl}methyl)benzamide
1-methyl-4-{[5-(4-methyl-1H-imidazol-5-yl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-3-yl]methyl}piperidine
6-methyl-5-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
methyl 1-ethoxy-8-[3-(furan-2-yl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylate
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
N-[2-(dimethylamino)-2-(pyridin-2-yl)ethyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
8-methyl-4-[2-(pyridin-3-yl)piperidine-1-carbonyl]-2-(pyrimidin-5-yl)quinoline
3-({[4-(pyridin-3-yl)phenyl]methyl}amino)propan-1-ol
N-ethyl-2,6-dihydroxy-N-[2-(4-methylphenoxy)ethyl]benzamide
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-1-methyl-2-oxo-1,2-dihydroquinoline-3-carboxamide
7-(3-methyl-1H-pyrazole-5-carbonyl)-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-[(2S)-1-hydroxybutan-2-yl]acetamide
5-acetyl-N,2,4-trimethyl-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrrole-3-carboxamide
2-[(1R,5R)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-3-yl]-5H,6H,7H-cyclopenta[b]pyridine-3-carboxamide