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1-[5-(3,4-difluorophenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-ol
N-[2-(1H-imidazol-4-yl)ethyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
(1R,5R)-6-benzyl-N-ethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(2-methoxyethyl)-4-({[1-(3-methylphenyl)cyclopropyl]carbamoyl}amino)benzamide
2-(2-hydroxyethyl)-8-[6-(propan-2-yl)pyridin-2-yl]-2,8-diazaspiro[5.5]undecan-3-one
N-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-8-fluoroquinoline-2-carboxamide
N-ethyl-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-5-[(4H-1,2,4-triazol-3-ylsulfanyl)methyl]furan-2-carboxamide
N-[(4-methylphenyl)(phenyl)methyl]-2-(4-oxo-1,4-dihydropyridin-1-yl)acetamide
N-[(3S,4R)-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-(2-{[(2-methoxyethyl)(pyridin-4-ylmethyl)carbamoyl]amino}phenyl)-N,N-dimethylacetamide
dimethyl({[(3S,4R)-1-(6-methylpyridazin-3-yl)-4-(propan-2-yl)pyrrolidin-3-yl]sulfamoyl})amine
(2S,4S)-4-amino-N-methyl-1-[(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)sulfonyl]pyrrolidine-2-carboxamide
2-hydroxy-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
N-(6-phenoxypyridin-3-yl)-1-(pyridine-4-carbonyl)piperidine-4-carboxamide
1-[4-(2-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
1-{1'-[(3-methyl-1,2-oxazol-5-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}propan-1-one
1-[1-(6-methylquinolin-4-yl)piperidin-4-yl]piperidin-4-ol
5-tert-butyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1,3,4-oxadiazol-2-amine
2-[4-(3,4-diethoxyphenyl)-1H-imidazol-2-yl]pyridine
1-(2-methoxyacetyl)-N,4-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]piperazine-2-carboxamide
N4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N4,N6,N6-trimethylpyrimidine-4,6-diamine
2-[(dimethylcarbamoyl)amino]-N-[2-(1,3-thiazol-4-yl)ethyl]acetamide
1-[3-(1-benzothiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4-methylpiperazine
5-benzyl-N-(2-hydroxyethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
(2S,4S)-4-cyclobutaneamido-1-methyl-N-(naphthalen-1-ylmethyl)pyrrolidine-2-carboxamide
N-cyclopropyl-N-[(3-methylthiophen-2-yl)methyl]-4-sulfamoylbenzamide
4-(2-phenylphenyl)-3-(1H-pyrazol-1-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1,3-dimethyl-6-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
1-(azepan-1-yl)-3-(3-{[ethyl(pyridin-4-ylmethyl)amino]methyl}phenoxy)propan-2-ol
N,N-dimethyl-1-(2-phenoxybenzoyl)azepan-4-amine
4-chloro-3-{1-[3-(1H-imidazol-1-yl)propyl]-1H-imidazol-2-yl}-1-methyl-1H-indazole
1-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-yl]-2-(5-amino-1,3,4-thiadiazol-2-yl)ethan-1-one
1-(3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-1-yl)ethan-1-one
2-[1-(naphthalen-2-ylmethyl)-3-oxopiperazin-2-yl]-N-(prop-2-en-1-yl)acetamide
N-(furan-3-ylmethyl)-5-oxo-1-(pyridin-4-ylmethyl)pyrrolidine-3-carboxamide
4-[1-(2-methoxyphenyl)-1H-pyrazole-4-carbonyl]-3,4-dihydro-2H-1,4-benzoxazine
7-[(2-ethylpyrimidin-4-yl)methyl]-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
N1-{4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}pentane-1,5-diamine
N-[2-(4-fluorophenyl)ethyl]-2-[(pyridin-3-ylmethyl)amino]acetamide
N-[(2R,4R,6S)-2-tert-butyl-6-[2-methyl-4-(1H-pyrazol-1-yl)phenyl]oxan-4-yl]acetamide
N-{1-oxaspiro[4.5]decan-3-yl}furan-2-carboxamide
1-methyl-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
methyl 2-{[5-(2-fluorophenoxymethyl)-1H-pyrazol-3-yl]formamido}butanoate
4-chloro-N-[(3S,5S)-5-(ethylcarbamoyl)-1-(4-methylpent-3-en-1-yl)pyrrolidin-3-yl]-1H-pyrazole-3-carboxamide
ethyl 3-[(3-chlorophenyl)methyl]-1-(thiophene-2-carbonyl)piperidine-3-carboxylate
1-[(1R,5R)-6-(2-phenylethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
(4aR,7aS)-1-[2-(dimethylamino)acetyl]-4-(3-ethoxypropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[2-(propan-2-yloxy)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]-5,6-dimethylthieno[2,3-d]pyrimidin-4-amine
2-(4-{[3-(2-hydroxyethyl)-4-(thiophen-2-ylmethyl)piperazin-1-yl]methyl}phenoxy)ethan-1-ol