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1-(2-{[(1-phenylpiperidin-4-yl)amino]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)ethan-1-one
1-(2-fluoro-4-hydroxybenzoyl)-4-methylpiperidine-4-carbonitrile
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-[4-(1H-pyrazol-1-yl)phenyl]piperidine-2-carboxamide
3-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)-N-[1-(pyridin-3-yl)propyl]propanamide
4-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl]pyrrolidin-2-one
1-[3-methyl-1-(pyridin-3-yl)butyl]-3-[3-(methylsulfamoyl)phenyl]urea
2-{[4-(1H-imidazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-(4-methoxyphenyl)-1H-imidazole
1-(3-chlorophenyl)-4-(3-methanesulfonylpropanoyl)piperazin-2-one
7-{imidazo[1,2-a]pyridine-3-carbonyl}-2-phenyl-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-methoxy-8-(2-methyl-1-phenyl-1H-1,3-benzodiazole-5-carbonyl)-1,8-diazaspiro[4.5]decan-2-one
1-(6-methyl-2H-1,3-benzodioxol-5-yl)-3-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)urea
8-fluoro-N-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]quinoline-2-carboxamide
N,1-dimethyl-N-[2-(oxan-2-yl)ethyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
[(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)({1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}methyl)amine
2-(7-chloro-2,3-dihydro-1,4-benzodioxin-6-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N5-[(4-chlorophenyl)(phenyl)methyl]-N3-methyl-N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
N,1-dimethyl-N-(2-phenyl-1-{1-[3-(thiophen-2-yl)propanoyl]piperidin-4-yl}ethyl)-1H-pyrazole-3-carboxamide
1-methyl-4-{2-[3-(1-methyl-1H-pyrazol-3-yl)phenyl]pyridine-4-carbonyl}piperazine
N2,N2,6-trimethyl-N4-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyrimidine-2,4-diamine
1-[(1-{1-[1-(1-methylcyclopropyl)propan-2-yl]piperidin-4-yl}-1H-1,2,3-triazol-4-yl)methyl]azepane
2-{4-[(2-chloro-6-fluorophenyl)methyl]-1-(3-methylbutyl)piperazin-2-yl}ethan-1-ol
[(3,5-dichloropyridin-4-yl)methyl][2-(2-ethoxyphenoxy)ethyl]methylamine
7-[4-(1H-pyrazol-4-yl)butanoyl]-1-oxa-3,7-diazaspiro[4.5]decan-2-one
3-(dimethyl-1,2-oxazol-4-yl)-N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)propanamide
N-[2-(4-methoxyphenyl)ethyl]-2-[1-(naphthalen-1-ylmethyl)-3-oxopiperazin-2-yl]acetamide
N-[3-(dimethylamino)propyl]-1-[(2,5-dimethylthiophen-3-yl)sulfonyl]-N-methylpiperidin-3-amine
1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]-3-[4-(methylsulfanyl)benzoyl]piperidine
1-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-3-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}urea
N-[(2-aminopyridin-3-yl)methyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
{1-[3-(1H-1,3-benzodiazol-6-yl)phenyl]ethyl}dimethylamine
N-(1,3-benzothiazol-2-ylmethyl)-5-(4-fluorophenyl)-1,2,4-triazin-3-amine
(3aS,6aS)-5-[4-(cyclopropylcarbamoyl)pyridin-2-yl]-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-(4-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-2-yl)-1H-indole
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-3-(1-methylpiperidin-2-yl)propanamide
2-(2H-1,2,3-benzotriazol-2-yl)-1-[1-(2-hydroxyethyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl]ethan-1-one
2-(4-fluoro-3-methylphenyl)-2-[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]acetic acid
2-{4-[2-(2-chloro-6-fluorophenyl)acetyl]-2-oxopiperazin-1-yl}benzonitrile
(1S,5R)-6-[(1-phenyl-1H-pyrazol-4-yl)methyl]-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-methyl-4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carboxamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-[(2-fluorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(5-chlorothiophen-2-yl)methyl]-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
N-[3-(propan-2-yloxy)propyl]-5-(3,4,5-trimethoxyphenyl)-1,2,4-triazin-3-amine
3-methyl-2-{3-[1-(propan-2-yl)-1H-pyrazol-3-yl]phenyl}pyridine
1-cyclopentyl-N-(2-methylpropyl)-4-oxo-5-{1,3,3-trimethyl-6-azabicyclo[3.2.1]octane-6-carbonyl}-1,4-dihydropyridine-3-carboxamide
4-({2,5-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-N-phenylpiperidine-1-carboxamide
2-(4,4-dimethyl-2,5-dioxoimidazolidin-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
4-hydroxy-1-[3-(trifluoromethyl)pyridin-2-yl]piperidine-4-carboxylic acid
N-cyclopentyl-3-{methyl[2-(1H-pyrazol-1-yl)ethyl]sulfamoyl}benzamide
2-(1H-1,3-benzodiazol-1-yl)-N-methyl-N-(quinolin-5-ylmethyl)propanamide
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(3-methylpyridin-2-yl)ethyl]acetamide