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N-[(3R,4R)-4-(pyrrolidin-1-yl)oxolan-3-yl]-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
1-benzyl-N-ethyl-5-[(prop-2-en-1-yl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
3-(2,4-dimethoxybenzoyl)-1-(1-propylpiperidin-4-yl)piperidine
3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[2-(7-methyl-1H-1,3-benzodiazol-2-yl)ethyl]benzamide
2-(1H-indol-3-yl)-1-[2-(piperidin-1-ylmethyl)-1,4-oxazepan-4-yl]ethan-1-one
N-{[5-(4-fluorophenyl)furan-2-yl]methyl}-1-(2-methoxyacetyl)piperidine-3-carboxamide
N-[(2-methoxyphenyl)methyl]-5-methyl-6-(4-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
2-(4-cyclobutyl-6-methylpyrimidin-2-yl)-2,7-diazaspiro[4.5]decan-6-one
1-methyl-2-[1-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]propanamide
5-methyl-1-(4-{4-[(1-propylcyclopropyl)amino]piperidin-1-yl}phenyl)pyrrolidin-2-one
4-chloro-N-[(1-methanesulfonylpiperidin-3-yl)methyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
2-(1-{[4-(difluoromethoxy)phenyl]methyl}piperidin-3-yl)-1,2,3,4-tetrahydroisoquinoline
1-{2-[(2-methylpropyl)amino]ethyl}-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-{1-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
N-[(1-benzylpiperidin-4-yl)methyl]-N,1-dimethyl-2-oxoimidazolidine-4-carboxamide
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-1-(2-fluorophenyl)cyclopropane-1-carboxamide
5-({[2-(3,4-dimethoxyphenyl)propan-2-yl]carbamoyl}amino)-2-fluoro-N-methylbenzamide
5-(4-benzyl-3-ethyl-5-oxo-1,4-diazepane-1-carbonyl)-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
4-(3,3-diphenylpiperidine-1-carbonyl)imidazolidin-2-one
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-(1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)acetamide
3,7-dimethyl-2-{5-[(1-methyl-1H-imidazol-2-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-1H-indole
1-(cyclopropylmethyl)-4-[4-(propan-2-yl)-1,3-thiazol-2-yl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
3-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazole
4-{[2-(1-benzylpyrrolidin-3-yl)ethyl]amino}pyrimidine-5-carboxylic acid
(3aR,6aR)-2-methanesulfonyl-N-[(5-methylpyrazin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
2-(oxolan-2-ylmethyl)-9-(trimethyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-{1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)quinoxaline
1-(cyclopropylmethyl)-5-(1-ethyl-3-methylpiperidine-3-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-({1-[4-(1H-1,2,4-triazol-3-yl)benzoyl]pyrrolidin-3-yl}methyl)benzoic acid
2-({[1-(1-benzoxepine-4-carbonyl)piperidin-3-yl]oxy}methyl)pyridine
3-{[6-(4-methoxyphenyl)-7-methyl-8-oxo-7H,8H-imidazo[1,2-a]pyrazin-2-yl]formamido}propanamide
N-cyclopentyl-N-[(4-methoxynaphthalen-1-yl)methyl]-2-(methylamino)pyrimidine-5-carboxamide
2-(cyclohex-1-en-1-yl)-N-(1,2-oxazol-3-ylmethyl)acetamide
N-[(7-fluoro-2-oxo-1,2-dihydroquinolin-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
N-[3-({ethyl[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]carbamoyl}amino)-4-fluorophenyl]acetamide
2-(4-{1-cyclopentyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
2-[(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}phenyl)formamido]acetamide
2-[4-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-6-methoxyphenol
4-{[3-ethyl-1-(1-methylpiperidin-4-yl)-1H-1,2,4-triazol-5-yl](pyridin-3-yl)methyl}morpholine
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-4-(2-fluoro-5-methylphenoxy)piperidine-4-carboxylic acid
(4S,6R)-6-methyl-2-sulfanylidene-N-({7-[2-(trifluoromethyl)phenyl]-2,3-dihydro-1-benzofuran-2-yl}methyl)-1,3-diazinane-4-carboxamide
2-{1-[(3,4-difluorophenyl)methyl]-4-[(4-ethynylphenyl)methyl]piperazin-2-yl}ethan-1-ol
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-2-methylimidazo[1,2-a]pyridine-6-carboxamide
2-{9-[4-(dimethylamino)benzoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
4-{1-[1-(5,6-dimethylpyrimidin-4-yl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
1-(1H-imidazol-2-ylmethyl)-4-{[5-(methylsulfanyl)-4-phenyl-4H-1,2,4-triazol-3-yl]methyl}piperidine
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)-1,3-dimethyl-1H-pyrazole-5-carboxamide