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[1-(dimethyl-1,3-thiazole-4-carbonyl)piperidin-2-yl]methanamine
1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}urea
2-(pyridin-3-yloxy)-1-[2-(trifluoromethyl)morpholin-4-yl]ethan-1-one
4,6-dimethyl-2-oxo-N-{2-[3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1,2-dihydropyridine-3-carboxamide
2-[1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)pyrrolidin-3-yl]benzoic acid
N-[(1-ethylcyclobutyl)methyl]-3-[(2-oxopyrrolidin-3-yl)sulfamoyl]benzamide
6-(morpholin-4-yl)-N-{[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-4-amine
2-[1-(cyclohexylmethyl)-4-[1-(2,3-dihydro-1H-inden-5-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
2-[2-(2,4-difluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-1-(propan-2-yl)-1H-pyrrole
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-3-(1H-1,2,4-triazol-1-yl)propanamide
5-phenyl-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}-1,2-oxazole-3-carboxamide
(1S,5R)-3-(8-fluoroquinoline-2-carbonyl)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-butyl-1'-{6-methylthieno[2,3-d]pyrimidin-4-yl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-(methylsulfanyl)-1-{4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidin-1-yl}ethan-1-one
4-(3-hydroxy-3-methylbutyl)-N-(2-methoxy-2-methylpropyl)benzamide
N-(2-methylphenyl)-4-(4-oxo-4,5,6,7-tetrahydro-1-benzofuran-3-carbonyl)morpholine-2-carboxamide
N,N-dimethyl-3-{4-[2-(pyrrolidin-1-yl)ethoxy]phenyl}benzamide
2-(2-{1-[2-(dimethylamino)-5,6-dimethylpyrimidin-4-yl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazin-1-yl]-2-(2H-1,2,3,4-tetrazol-2-yl)ethan-1-one
[(3S,5R)-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(5-propylfuran-2-yl)methyl]piperidin-3-yl]methanol
4-({1-[(5-chloro-2,4-dimethoxyphenyl)methyl]piperidin-2-yl}methyl)morpholine
1-(2-methoxyphenyl)-N-{[5-(4-methoxyphenyl)-1,2-oxazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
2,2,2-trifluoro-N-{2-[(6-methyl-2-oxo-1,2-dihydropyridin-3-yl)formamido]ethyl}acetamide
2,4-dimethoxy-N-{[1-(propan-2-yl)piperidin-4-yl]methyl}benzamide
1-[(3-cyclopropyl-1H-pyrazol-5-yl)methyl]-4-(4-methoxyphenyl)piperazine
N-[4-(4-methylpyridin-3-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
3-methyl-5-(1-{2-[2-(methylsulfanyl)phenyl]-1H-imidazol-1-yl}propyl)-1,2,4-oxadiazole
2-amino-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)-4-[5-(oxan-2-yl)furan-2-yl]pyridine-3-carbonitrile
3-[(3-hydroxypiperidin-1-yl)methyl]-7-methyl-1,2-dihydroquinolin-2-one
5-{[4-(4-methoxybenzoyl)piperazin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
1-[2-butyl-5-oxo-4-(3-phenylphenyl)piperazin-1-yl]pentane-1,4-dione
N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-3-(1H-1,2,4-triazol-3-yl)benzamide
3-(propan-2-yl)-5-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)pyrrolidin-2-yl]-1,2,4-oxadiazole
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
6-[(diethylamino)methyl]-N-(1,2-oxazol-5-ylmethyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N,2-dimethyl-6-oxo-1,6-dihydropyrimidine-5-carboxamide
N-{[7-(2,3-difluorobenzoyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-1-phenylmethanesulfonamide
N4-(2,5-difluorophenyl)morpholine-2,4-dicarboxamide
[1-(5-fluoro-1H-indole-2-carbonyl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
(2R,3R)-1'-[(2,6-dimethoxyphenyl)methyl]-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-benzothiazole
(2-methoxyethyl)[(3-methyl-1H-pyrazol-5-yl)methyl](thiophen-2-ylmethyl)amine
8-[4-(1H-imidazol-1-yl)butanoyl]-2-(3-methoxypropyl)-2,8-diazaspiro[4.5]decan-3-one
(3R,5R)-N-{1-[(3-methylphenyl)methyl]cyclopropyl}-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
2-(propan-2-yl)-9-[(2,3,4-trifluorophenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
5-(1H-imidazol-1-yl)pyridine-3-carboxamide
2-{1-[(2-chloro-6-fluorophenyl)methyl]-3-oxopiperazin-2-yl}acetamide
5-(propan-2-yl)-N-[2-(pyrrolidin-1-yl)ethyl]-1,2-oxazole-3-carboxamide
(2S,4R)-4-(dimethylamino)-1-(1,3-thiazol-4-ylmethyl)pyrrolidine-2-carboxylic acid
N-[(5-ethylpyridin-2-yl)methyl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]acetamide