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3-[ethyl({[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl})amino]-1λ6-thiolane-1,1-dione
2-(2-methoxyethyl)-N-[3-(2-methoxyphenyl)phenyl]morpholine-4-carboxamide
(3S,4R)-1-(1-tert-butyl-1H-pyrrole-3-carbonyl)-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
1-(8-acetamidoquinolin-5-yl)-5-methyl-1H-pyrazole-3-carboxylic acid
N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1-benzofuran-5-carboxamide
1-[(5-{furo[3,2-c]pyridin-4-yloxy}-2-methoxyphenyl)methyl]pyrrolidine
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-amine
(3E)-2-{methyl[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]amino}-4-phenylbut-3-enoic acid
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-[2-(pyrrolidine-1-sulfonyl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
4-(4-methanesulfonylphenyl)-2-methylquinazoline
4-{[(2,3-dimethoxyphenyl)methyl]amino}-N-(2-hydroxypropyl)-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-{5H,6H,7H,8H-imidazo[1,5-a]pyrazin-7-yl}ethan-1-one
1-(2-benzyl-1,3-thiazole-4-carbonyl)-4-(furan-2-carbonyl)-1,4-diazepane
3-(1-benzyl-1H-imidazol-2-yl)-1-(5-methoxyfuran-2-carbonyl)piperidine
ethyl 4-(4-{4-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]piperidin-1-yl}benzoyl)piperazine-1-carboxylate
1,2-dimethyl-4-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazine
2-methyl-N-[2-(2-oxo-5,5-diphenylpiperidin-1-yl)ethyl]propanamide
3-[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]-1-(5-phenyl-1,2-oxazole-3-carbonyl)piperidine
N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-2-[2,6,6-trimethyl-1-(2-methylpropyl)-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamide
(1R,5R)-3-{6-chloroimidazo[1,2-a]pyridine-2-carbonyl}-6-propyl-3,6-diazabicyclo[3.2.2]nonane
5-[3-(4-ethyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]-6-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
[3-(methylsulfanyl)propyl][(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amine
ethyl 2-{4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazin-1-yl}-1,3-oxazole-4-carboxylate
1-[4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidin-1-yl]-2-(morpholin-3-yl)ethan-1-one
2-{[4-(2H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-1,2,3,4-tetrahydroisoquinolin-4-ol
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-3-phenyl-3-(pyridin-2-yl)propanamide
3-[(3R,4S)-4-(dimethylamino)-1-[4-(2-fluorophenyl)benzoyl]piperidin-3-yl]propanoic acid
N-methyl-1-(3-phenylpropyl)-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
N,N,4-trimethyl-3-{[(prop-2-en-1-yl)(propyl)carbamoyl]methyl}-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-[4-(oxolan-2-yl)butyl]-1-(6-phenoxypyridin-3-yl)urea
2-amino-4-[4-(pyridin-2-ylmethoxy)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
1-methyl-4-{1-[1-(4-methyl-1,2,5-oxadiazole-3-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}piperazine
5-[3-(4-methoxyphenyl)-1H-pyrazol-5-yl]-1,3-dimethyl-1H-1,2,4-triazole
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-(4-methyl-1,3-oxazole-5-carbonyl)piperazine
4-(4-chlorophenyl)-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]butanamide
1-[2-(dimethylamino)ethyl]-6-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-2-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
ethyl (4aS,8aR)-6-{[(4-methylphenyl)methyl]carbamoyl}-decahydro-1,6-naphthyridine-4a-carboxylate
1-[2-(4-fluorophenyl)acetyl]-3-(3-methoxypropyl)piperidine-3-carboxylic acid
3-chloro-N-(2-methoxyethyl)-4-({1-[(2E)-4-methylpent-2-en-1-yl]piperidin-4-yl}oxy)benzamide
5-{3-butyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-3-(5-methylfuran-2-yl)-1H-pyrazole
N-(9H-fluoren-9-yl)-1,9-dioxaspiro[5.5]undecan-4-amine
3-(methylsulfanyl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)propanamide
{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}({2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl})amine
2-(3-methoxypropyl)-9-[2-methyl-3-(1H-pyrazol-1-yl)propanoyl]-2,9-diazaspiro[5.5]undecan-3-one
5-[1-(4-chlorophenyl)cyclohexyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
ethyl 1-{[2-(2,4-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine-4-carboxylate
N,1-dimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[5-methoxy-2-({[2-(pyridin-4-yl)ethyl]amino}methyl)phenoxy]-3-(4-methylpiperazin-1-yl)propan-2-ol
N-butyl-N-[(2E)-3-phenylprop-2-en-1-yl]-4-(1H-1,2,4-triazol-5-yl)benzamide