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4-(propan-2-yl)-2-[4-(pyrazin-2-yl)piperazin-1-yl]-6-(trifluoromethyl)pyrimidine
3-{[3-methyl-1-(3-methylphenyl)-1H-1,2,4-triazol-5-yl]methyl}-2,3-dihydro-1,3-benzoxazol-2-one
(2S,4S,5R)-5-(4-chlorophenyl)-4-[(1,3-dihydroxypropan-2-yl)carbamoyl]-1,2-dimethylpyrrolidine-2-carboxylic acid
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(thian-4-yl)piperidin-4-yl]oxy}benzamide
[(3R,4S)-1-[(5-fluoro-2-methoxyphenyl)methyl]-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
2-[(3S)-3-hydroxypyrrolidin-1-yl]-N,1-dimethyl-N-(thian-4-yl)-1H-1,3-benzodiazole-5-carboxamide
2-methyl-4-{methyl[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}butan-2-ol
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-3-(2-ethyl-1H-imidazol-1-yl)propan-1-one
1-[1,3-dioxo-2-(quinolin-3-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-[2-(3-fluorophenyl)ethyl]piperidine-4-carboxamide
5-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-[1-(1H-imidazol-1-yl)butan-2-yl]-1H-pyrazole-3-carboxamide
1-(3-{5-methyl-2-[(pyridin-2-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-2-(morpholin-4-yl)propan-1-one
N-butyl-N-[(4-fluorophenyl)methyl]-2-(pyridin-4-yl)acetamide
{[1-(2,5-dimethylphenyl)-3-phenyl-1H-pyrazol-4-yl]methyl}(oxan-4-ylmethyl)amine
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-{1-[2-(trifluoromethyl)phenyl]ethyl}acetamide
4-(1H-imidazol-1-yl)-1-(4-phenyl-1,3-thiazol-2-yl)piperidine-4-carboxylic acid
8-[(1-ethyl-1H-pyrazol-4-yl)methyl]-2-(3-methylbutyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[(dimethylamino)methyl]-1-[2-(morpholin-4-yl)pyrimidine-5-carbonyl]pyrrolidin-3-ol
2-{4-[(3,3-difluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
3-[1-(1-benzofuran-2-ylmethyl)piperidin-3-yl]-N-(4-methoxy-2-methylphenyl)propanamide
1-methyl-N-(2-propoxyethyl)-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
2-(4-fluorophenyl)-1-(thiophene-3-carbonyl)pyrrolidine
2-(1,3-benzoxazol-2-yl)-7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
N-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}-5-oxopyrrolidine-2-carboxamide
(1R,5R)-6-(2-methoxyethyl)-3-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
4-[3-(2-methylpropyl)-1,2-oxazole-5-carbonyl]-1λ6-thiomorpholine-1,1-dione
3-methyl-7-(quinolin-4-ylmethyl)-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
2-(2-aminoethyl)-N-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}quinazolin-4-amine
1-{[5-(1-benzyl-1H-1,2,4-triazol-5-yl)furan-2-yl]methyl}-4-methylpiperazine
1-[2-(cyclohex-1-en-1-yl)ethyl]-5-(4-methyl-1H-imidazol-5-yl)-4-phenyl-1H-imidazole
5-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-2-ethylpyrimidine
4-[2-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]thiomorpholine
5-(2-ethylpyrimidine-5-carbonyl)-N-phenyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[2-(4-cyclopropyl-4-methyl-2-oxopyrrolidin-1-yl)acetyl]-4-phenylpiperidine-4-carbonitrile
5-[3-(naphthalene-2-carbonyl)piperidine-1-carbonyl]-4-propylpyrimidine
2-(dimethylamino)-2-(3-fluorophenyl)-1-[4-(4-hydroxyphenyl)piperazin-1-yl]ethan-1-one
N-ethyl-2-{3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}pyrimidin-4-amine
N-[2-(1H-imidazol-1-yl)ethyl]-3-(5-methylfuran-2-yl)benzamide
4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
2-{3-[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]propyl}phenol
4-[2-(dimethyl-1,2-oxazol-4-yl)pyrrolidine-1-carbonyl]-6-ethyl-2-methylquinoline
N-[(3R,4S)-1-(5-methyl-1,2,4-oxadiazol-3-yl)-4-propylpyrrolidin-3-yl]-3-(morpholin-4-yl)propanamide
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1,2,3,4-tetrahydronaphthalene-2-carboxamide
N-methyl-N-[(5-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
5-chloro-2-[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]-1H-1,3-benzodiazole
propan-2-yl (4aS,7aR)-6,6-dioxo-4-(pyridine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
2-[4-(adamantan-2-yl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-(4-methoxyphenyl)-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carboxamide
3,3,3-trifluoro-2-methoxy-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-phenylpropanamide
1-methyl-5-{4-[(3-methylphenyl)methyl]piperazine-1-carbonyl}-1,2-dihydropyridin-2-one