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1-[4-(4-ethylpiperazine-1-carbonyl)phenyl]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-amine
N-(2-phenylethyl)-N-(pyridin-2-ylmethyl)oxane-2-carboxamide
4-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]piperazine-1-sulfonamide
{[5-(methoxymethyl)furan-2-yl]methyl}({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
1-(4-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-ylmethyl}phenyl)-1H-imidazole
N,4,6-trimethyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}pyrimidin-2-amine
2-[3-({[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]amino}methyl)-2-methyl-1H-indol-1-yl]acetamide
2-(2-ethyl-1H-imidazol-1-yl)-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}ethan-1-one
N-[(1S,6R)-6-carbamoylcyclohex-3-en-1-yl]-3-cyclopropaneamido-4-methylbenzamide
1-(3-{4-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]piperidine-1-carbonyl}piperidin-1-yl)ethan-1-one
5-{6-chloro-1H,2H,3H,4H,5H-pyrido[4,3-b]indole-2-carbonyl}-2-cyclopropyl-4-methylpyrimidine
3-chloro-N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-4-fluoro-1-benzothiophene-2-carboxamide
2-chloro-N-{2-[4-(cyclohex-3-en-1-yl)-1H-1,2,3-triazol-1-yl]ethyl}benzamide
3-[(3R,4S)-1-(3-chlorothiophene-2-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(pyridin-2-ylsulfanyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
dimethyl({[1-methyl-2-(2-methylpropyl)-7-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)-1H-1,3-benzodiazol-5-yl]sulfamoyl})amine
2-[2-(methylsulfanyl)acetyl]-7-(oxan-4-yl)-2,7-diazaspiro[4.5]decan-6-one
11-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecane
2-methyl-6-{1-[(4-phenylphenyl)methyl]piperidin-4-yl}pyrimidin-4-ol
1-[(3S,4R)-3-(dimethylamino)-4-(4-methylphenyl)pyrrolidin-1-yl]-2-hydroxyethan-1-one
1-{4-[(3-chlorophenyl)methyl]piperazin-1-yl}-2-(pyridin-3-yl)ethan-1-one
3-(pyrrolidin-3-yl)-N-{5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-ylmethyl}benzamide
(2R,3R,6R)-3-(2,3-difluorophenyl)-5-[(3-fluorophenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-1-(6-ethyl-2-methylpyrimidin-4-yl)piperidin-4-amine
1-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)benzoyl]-4-[(2-methylphenyl)methyl]piperazine
N-[2-(4-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(pyridin-3-yl)acetamide
5-{3-[2-(2-methoxyphenyl)pyrrolidin-1-yl]-3-oxopropyl}-5-[(4-methylphenyl)methyl]pyrrolidin-2-one
N-[(4-hydroxy-3-methoxyphenyl)methyl]-2-methyl-4-phenyl-1,3-thiazole-5-carboxamide
N-[2-(2-chlorophenyl)-2-(dimethylamino)ethyl]-3-cyclohexyl-1H-pyrazole-4-carboxamide
5-(2-{[butyl(methyl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carbonyl)-4-methyl-2-oxo-1,2-dihydropyridine-3-carbonitrile
[3-({1-[(6-methoxy-2H-chromen-3-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[1-(3-ethyl-1,2-oxazol-5-yl)ethyl]-8-fluoroquinoline-2-carboxamide
8-(2-methylpyridine-3-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
2,6,6-trimethyl-3-[2-oxo-2-(5-oxo-1,4-diazepan-1-yl)ethyl]-1-(propan-2-yl)-4,5,6,7-tetrahydro-1H-indol-4-one
3-hydroxy-S-[2-(1-methylcyclopropanecarbonyl)-1,2,3,4-tetrahydroisoquinolin-6-yl]butane-1-sulfonamido
N-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2,8-diazaspiro[4.5]decane-3-carboxamide
N-[2-(4-fluorobenzenesulfonyl)ethyl]-2-[(propan-2-yl)amino]pyrimidine-5-carboxamide
3-[2-(3-chloro-4-hydroxyphenyl)acetyl]-3,9-diazaspiro[5.6]dodecan-10-one
1-[(4-hydroxy-3-methoxyphenyl)methyl]-5-oxopyrrolidine-3-carboxylic acid
4-(1H-1,2,3,4-tetrazol-5-ylmethyl)-8-thia-4,6-diazatricyclo[7.5.0.02,7]tetradeca-1(9),2(7),5-trien-3-one
5-{3-cyclopropyl-1-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-yl}-2-methyl-1,4-dihydropyridin-4-one
3-(2-acetylphenyl)-5-(morpholine-4-sulfonyl)benzoic acid
1-(4-benzylpiperazin-1-yl)-3-[1-(thiophen-3-ylmethyl)piperidin-3-yl]propan-1-one
N-ethyl-4-hydroxy-2-(4-methylphenyl)-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
3-methyl-5-{2-oxo-2-[3-(pyrimidin-4-yl)piperidin-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2S)-2-amino-3-methoxy-1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)propan-1-one
3-[5-({[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}methyl)thiophen-3-yl]prop-2-yn-1-ol
(3S,4R)-3-ethyl-4-methyl-1-(5-phenyl-1H-pyrrole-2-carbonyl)piperidin-4-ol
3-(4,5-dimethyl-1H-pyrazol-3-yl)-N-(2-methoxyethyl)-N-(pyridin-3-ylmethyl)propanamide
3-({[1-(2,3-dihydro-1H-indene-1-carbonyl)piperidin-4-yl]oxy}methyl)pyridine