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4-{3-[(3S,4S)-3,4-bis(hydroxymethyl)pyrrolidine-1-carbonyl]phenyl}-2-methylbutan-2-ol
7-cyclohexyl-2-[3-(1H-pyrazol-1-yl)propanoyl]-2,7-diazaspiro[4.5]decan-6-one
(1S,5R)-3-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
3-[2-(3-methoxyphenyl)ethyl]-1-(1,3-thiazol-2-ylmethyl)piperidine
1-[1'-(1-ethyl-3-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]propan-1-one
5-(3-{1-[(1-ethyl-1H-imidazol-2-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrimidine
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-hydroxypropan-1-one
N-cyclopropyl-3-[4-({[(dimethyl-1,2-oxazol-4-yl)methyl](methyl)carbamoyl}amino)phenyl]propanamide
6-(quinolin-8-yl)pyridin-2-ol
4-[2-(3-hydroxypiperidin-1-yl)acetyl]-1-(4-methylphenyl)piperazin-2-one
1-[1-({2-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidin-4-yl]pyrrolidin-2-one
(2-ethoxy-5-{[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)amino]methyl}phenyl)methanol
4-amino-2-(morpholin-4-yl)-5-{pyrazolo[1,5-a]pyrimidin-3-yl}-5H,6H,7H,8H-pyrido[2,3-d]pyrimidin-7-one
2-methyl-4-(2-methylphenyl)-1-[5-(1H-pyrazol-1-ylmethyl)furan-2-carbonyl]piperazine
(3S,4R)-1-(3-methylpyridine-2-carbonyl)-4-(3-methylthiophen-2-yl)piperidin-3-ol
N,N-dimethyl-4-(4-phenyl-1,4-diazepane-1-carbonyl)piperidine-1-carboxamide
N-[3-(1H-indol-2-yl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidine-4-carboxamide
N-ethyl-1-methyl-N-(2-methylprop-2-en-1-yl)-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-1-(3-hydroxyphenyl)-5-oxopyrrolidine-3-carboxamide
4-(3-{1H-pyrazolo[3,4-b]pyridin-1-yl}phenyl)-4H-1,2,4-triazole
N-{2-[9-hydroxy-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-oxoethyl}acetamide
1-{3,7-dimethyl-3,7,11-triazaspiro[5.6]dodecan-11-yl}-2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]ethan-1-one
5-[1-(4-chlorophenyl)cyclobutanecarbonyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-6-carboxylic acid
N-[2-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]-3-(1H-indol-3-yl)propanamide
5-[methyl(2-phenylethyl)amino]-2-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-2,3-dihydropyridazin-3-one
9-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
[1-(5-{[(2E)-3-phenylprop-2-en-1-yl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-yl]methanol
1-(3-methyl-1H-pyrazole-4-carbonyl)-3-(4-phenylbenzoyl)piperidine
(1S,5R)-6-(2-methoxyethyl)-3-(pyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
2-{4-[(dimethyl-1,2-oxazol-4-yl)methyl]morpholin-3-yl}acetic acid
(2-aminoethyl)({[3-(methylsulfanyl)phenyl]methyl})(propan-2-yl)amine
[(3R,4R)-1-(2,6-difluoro-3-methoxybenzoyl)-4-{[(2-methoxyethyl)(methyl)amino]methyl}pyrrolidin-3-yl]methanol
N3-tert-butyl-1-cyclohexyl-4-oxo-N5-[phenyl(pyridin-4-yl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[(2,3-difluorophenyl)methyl]-3-hydroxy-3-({[(5-methylfuran-2-yl)methyl]amino}methyl)piperidin-2-one
7-[5-ethyl-4-(pyrrolidin-1-ylmethyl)furan-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-[1-(3-methylphenyl)-1H-imidazol-2-yl]-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]-4-{5-methylthieno[2,3-d]pyrimidin-4-yl}piperazine
1-{4-[(2-ethoxybutyl)amino]-2-(pyridin-2-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
N,1-dimethyl-N-[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]-5-(thiophen-2-yl)-1H-pyrazole-3-carboxamide
(1R,9aR)-1-({[2-(1H-indol-3-yl)ethyl]amino}methyl)-octahydro-1H-quinolizin-1-ol
N-[(2-chlorophenyl)methyl]-N-(prop-2-en-1-yl)pyridine-3-carboxamide
3-(5-chloro-2-methoxybenzoyl)-1-(1H-imidazol-2-ylmethyl)piperidine
2-(4-chlorophenyl)-N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
6-[2,4-bis(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
7-chloro-4-[1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
5-{[3-(4-methoxyphenoxy)phenyl]methyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine
N-[1-(1-{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]acetamide
N-(isoquinolin-5-ylmethyl)-N,2-dimethyl-5-sulfamoylbenzamide
8-(3-methylbutanoyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one