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N-({2-[2-(3-fluorobenzenesulfonamido)phenyl]-5-methyl-1,3-oxazol-4-yl}methyl)-2-methoxyacetamide
1-methyl-N-{[2-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
3-(4-{2-[benzyl(methyl)carbamoyl]ethyl}piperidine-1-carbonyl)piperidine-1-carboxamide
1-[3-(diphenylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]cyclobutan-1-amine
N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)-5-(morpholin-4-ylmethyl)furan-3-carboxamide
N-[2-(pyridin-2-yl)ethyl]-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}(3-phenylpropyl)amine
[(3,4-dimethoxyphenyl)methyl]({[2-(4-methoxyphenyl)-7-methylquinolin-3-yl]methyl})amine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-amine
2-[3-benzyl-1-(2-methoxyphenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(propan-2-yl)acetamide
2-(2,5-dimethoxyphenyl)-N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
3-[1-(2,1,3-benzothiadiazol-5-ylmethyl)piperidin-3-yl]-N-(2-fluorophenyl)propanamide
N-[2-(dimethylamino)ethyl]-N-[(5-methylthiophen-2-yl)methyl]-5-phenyl-1,2-oxazole-4-carboxamide
[(5-methoxy-3-methyl-1H-indol-2-yl)methyl](methyl)[3-(oxolan-2-yl)propyl]amine
1-(cyclohexylmethyl)-N-(furan-2-ylmethyl)-6-oxo-N-propylpiperidine-3-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-7-oxo-7H-[1,3]thiazolo[3,2-a]pyrimidine-5-carboxamide
8-chloro-N-(2-hydroxyethyl)-2-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]quinoline-4-carboxamide
ethyl 4-{2-[3-(2-methylphenyl)-2,5-dioxo-1-(pyridin-4-ylmethyl)pyrrolidin-3-yl]acetyl}piperazine-1-carboxylate
1-(6-{3-[1-(2-methylpropyl)piperidin-4-yl]pyrrolidin-1-yl}pyridin-3-yl)ethan-1-one
2-[1-({2-phenylimidazo[1,2-a]pyrimidin-3-yl}methyl)pyrrolidin-2-yl]pyridine
1-methyl-8-[(5-methylfuran-2-yl)methyl]-3-[3-(pyridin-4-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-chloro-N-methyl-N-(1,2-oxazol-3-ylmethyl)-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
2-amino-7-(4-chloro-1H-pyrazole-3-carbonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
ethyl 1-(2-chlorophenyl)-5-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)-1H-pyrazole-4-carboxylate
1-[4-hydroxy-4-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-2-(1H-pyrazol-1-yl)butan-1-one
[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
3-({[2-(4-phenylpyrimidin-2-yl)ethyl]amino}methyl)pyrrolidin-3-ol
1-[1-(2-chlorobenzoyl)piperidine-4-carbonyl]azepan-4-amine
4-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-6-methylpyrimidin-2-amine
4-{[6-(3-fluoro-4-methoxyphenyl)pyridin-3-yl]methyl}morpholine
methyl 2-(4-{[3-(3-methylphenyl)piperidine-1-carbonyl]amino}phenoxy)acetate
4-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-oxobutanamide
1-methyl-3-propyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
2-[(1-cyclobutanecarbonylpiperidin-4-yl)formamido]-2-(2-fluorophenyl)acetic acid
2-(1-benzofuran-2-yl)benzamide
8-[2-(dimethylamino)acetyl]-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
(3S,4S)-N-(3-cyclopentaneamidophenyl)-3-hydroxy-4-(propan-2-yloxy)pyrrolidine-1-carboxamide
1-(4-{[1,2,4]triazolo[4,3-a]pyridin-3-ylmethoxy}phenyl)ethan-1-one
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-4-(piperidin-1-yl)-N-(pyridin-4-ylmethyl)benzamide
1-methanesulfonyl-4-[2-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)phenoxy]piperidine
2-[8-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1,1-dioxo-1λ6-thiane-4-carboxamide
2-(2-methyl-1,3-thiazol-4-yl)-N-[1-(pyridine-4-carbonyl)piperidin-4-yl]acetamide
4-(3-chloro-4-methoxyphenyl)-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
3,5-dimethoxy-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decane
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(3-methylthiophen-2-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-fluoro-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-5-sulfamoylbenzamide
(2-ethoxy-5-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}phenyl)methanol
{[4-methoxy-3-(1H-1,2,4-triazol-1-ylmethyl)phenyl]methyl}(methyl)(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amine