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3-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}amino)methyl]-1-[(2-fluorophenyl)methyl]-3-hydroxypiperidin-2-one
2-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
(3S,4R)-1-[1-(difluoromethyl)-1H-pyrazole-3-carbonyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
5-{[(5-chloropyridin-3-yl)oxy]methyl}-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1,2-oxazole-3-carboxamide
1-(2-{1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
(3S,4R)-1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
{3-[4-(4-chlorophenoxy)piperidine-1-carbonyl]phenyl}methanol
ethyl 4-[3-(2-{[(2-fluorophenyl)methyl]carbamoyl}ethyl)piperidin-1-yl]piperidine-1-carboxylate
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-2-(pyrrolidin-3-yl)benzamide
(2R)-2-[({4-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)amino]propanamide
2-{2-oxo-2-[(2S)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl]ethyl}-2,3-dihydro-1,2-benzothiazol-3-one
3-[5-(2-methyl-1,3-thiazol-4-yl)-3-(oxan-4-yl)-1H-1,2,4-triazol-1-yl]benzoic acid
(2S,4R)-N,N-diethyl-4-{4-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-1H-1,2,3-triazol-1-yl}pyrrolidine-2-carboxamide
4-(3-chloro-4-fluorophenyl)-6-(methoxymethyl)pyrimidine
4-[(2,3-difluorophenyl)methyl]-3-(2-oxo-2-{4-[2-(pyrrolidin-1-yl)ethyl]piperidin-1-yl}ethyl)piperazin-2-one
3-{4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-1-yl}-1,2-benzothiazole
N-cyclohexyl-3-({1H-pyrrolo[2,3-b]pyridin-6-yl}amino)propanamide
methyl 1-{[5-methyl-2-(4-methylphenyl)-1,3-oxazol-4-yl]methyl}piperidine-2-carboxylate
1-ethyl-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
N-{2-[4-(4-fluorophenyl)-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl]ethyl}-4-methoxybenzamide
10-methoxy-5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
N-ethyl-2-(2-methoxy-5-methylphenyl)-N-methylpyrimidin-4-amine
5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole
N-[cyclopropyl(3-methylpyridin-2-yl)methyl]-4-hydroxy-2-phenylpyrimidine-5-carboxamide
(1R,5R)-3-[4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)benzoyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-methyl-5-[4-(3-phenylpropyl)piperazin-1-yl]-2,3-dihydropyridazin-3-one
N-{4-[1-(cyclohex-3-en-1-ylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}acetamide
(3S,4R)-1-(2,5-dimethylfuran-3-carbonyl)-4-(2-methoxyphenyl)pyrrolidine-3-carboxylic acid
3-[1-(pyridin-3-ylmethyl)piperidin-3-yl]-N-[4-(trifluoromethyl)phenyl]propanamide
1-[(2E)-3-(4-fluorophenyl)prop-2-en-1-yl]-N-phenylpiperidin-3-amine
2-{[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)amino}-N-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)acetamide
(1S,5R)-6-(cyclopropylmethyl)-3-{2-[(3-methoxyphenyl)sulfanyl]acetyl}-3,6-diazabicyclo[3.2.2]nonan-7-one
1-cyclopentyl-N-methyl-6-oxo-N-(quinolin-8-ylmethyl)piperidine-3-carboxamide
2-({1-[(4-methanesulfonylphenyl)methyl]piperidin-3-yl}methyl)-1H-1,3-benzodiazole
N-[4-(2,2-dimethylpropanamido)-3-methylphenyl]-2,3-dihydro-1,4-benzodioxine-2-carboxamide
2-(dimethylamino)-1-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]ethan-1-one
2-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
4-[2-(2-amino-4,6-dimethylpyrimidin-5-yl)acetyl]-1-(3-methoxyphenyl)-5-methylpiperazin-2-one
2-({[(3R,4R)-1-(3-chloro-5-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(ethyl)amino)ethan-1-ol
N-[(5-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
ethyl 1-[2-(4-methoxyphenyl)ethyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
4-[4-(3-fluorophenoxy)piperidine-1-carbonyl]-1,2,3,4-tetrahydroquinolin-2-one
(2-methoxyethyl)({2-phenyl-1-[1-(thiophen-2-ylmethyl)piperidin-4-yl]ethyl})(pyridin-3-ylmethyl)amine
1-[(3aR,7aS)-5-methyl-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-3-(1H-1,2,3-benzotriazol-1-yl)propan-1-one
(4aR,7aS)-1-methyl-4-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-benzyl-5-{[3-(3-methyl-1H-1,2,4-triazol-5-yl)piperidin-1-yl]methyl}pyrimidin-2-amine
N-[cyclopropyl(4-methoxyphenyl)methyl]-3-(3,5-dimethyl-1H-pyrazol-4-yl)propanamide
(3R,4R)-3-[ethyl({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)amino]-4-hydroxy-1λ6-thiolane-1,1-dione
4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-1-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}piperidine
N3-{[2-(2-fluorophenyl)-3-methyl-1H-indol-5-yl]methyl}piperidine-1,3-dicarboxamide