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3-{5-[2-(2H-1,3-benzodioxol-5-ylmethyl)propyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl}pyridine
(3S,4R)-N,N-dimethyl-4-(4-methylphenyl)-1-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidin-3-amine
1-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]urea
1-(4-{[(cyclopropylmethyl)(methyl)amino]methyl}-2-methoxyphenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
3-(2H-1,3-benzodioxole-5-carbonyl)-1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)piperidine
1-[(2-fluoro-5-methoxyphenyl)methyl]-4-(1-methylpiperidin-4-yl)piperidine
N-{1-[1-(4-tert-butylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
methyl 6-(1-methoxypropan-2-yl)-2-[(3-methylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-[(2R,3R,6R)-5-[(3-hydroxy-4-methoxyphenyl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
2-ethyl-4-methyl-N-[2-(4-phenylpyrimidin-2-yl)ethyl]-1,3-oxazole-5-carboxamide
4-[(2-fluorophenyl)methyl]-1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidine
2-{4-[(4-methylphenyl)methyl]-1-(thiophen-2-ylmethyl)piperazin-2-yl}ethan-1-ol
8-(5-methylpyrazine-2-carbonyl)-2-(3-phenylpropyl)-2,8-diazaspiro[4.5]decan-3-one
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-3-(morpholin-4-yl)benzamide
6,8-dimethyl-2-({4-[2-(pyrrolidin-1-yl)ethyl]piperazin-1-yl}methyl)quinolin-4-ol
[(3R,4R)-1-[1-(4-chlorophenyl)cyclobutanecarbonyl]-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-1,2,3-thiadiazole-4-carboxamide
4,6-dimethyl-N-[1-(morpholin-4-yl)propan-2-yl]pyrimidin-2-amine
5-benzyl-4-[(1-methyl-1H-imidazol-2-yl)methyl]-1-(4-methylphenyl)piperazin-2-one
4-(4-tert-butylbenzoyl)-1-(2-chlorophenyl)piperazin-2-one
[(3R,4R)-1-(6-chloro-1,3-benzothiazol-2-yl)-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
1-{2-[(2,3-dihydro-1-benzofuran-2-ylmethyl)(methyl)amino]pyrimidin-4-yl}piperidin-4-ol
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-{[1-(pyrimidin-2-yl)piperidin-3-yl]methyl}propanamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-2-ethyl-4-methyl-1,3-oxazole-5-carboxamide
5,6-dimethyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-cyclopropyl-1-[2-(1H-1,2,4-triazol-3-yl)benzoyl]piperazine-2-carboxamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-1,4,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[3-chloro-2-(propan-2-yloxy)phenyl]-3-(pyridin-2-yl)azetidine-1-carboxamide
{[5,8-dimethoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}dimethylamine
N-{1-[(4-chlorophenyl)methyl]cyclopropyl}-1-ethyl-3-methyl-1H-pyrazole-4-carboxamide
3-methyl-1-{4-[5-(piperidine-1-carbonyl)furan-2-yl]phenyl}urea
N-[(2-methoxyphenyl)methyl]-3-[2-(trifluoromethyl)morpholin-4-yl]propanamide
3-[(dimethylamino)methyl]-1-[4-(4-methylpiperazine-1-carbonyl)pyridin-2-yl]pyrrolidin-3-ol
3-(4-methoxy-3,5-dimethylphenyl)-1-{3-[(pyridin-3-yl)amino]propyl}urea
methyl 3-{4-[2-amino-3-cyano-5-methyl-6-(5-methylfuran-2-yl)pyridin-4-yl]-1H-pyrazol-1-yl}propanoate
1-(2,5-dimethylphenyl)-3-methyl-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-1,2,4-triazole
(3S,4S)-1-[(5-ethylpyridin-2-yl)methyl]-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
6-methyl-2-[4-(pyridin-3-ylmethoxy)piperidin-1-yl]pyridine-3-carboxylic acid
2-ethyl-4-{[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyrimidine
N-methyl-N-(1-methylpiperidin-4-yl)-1-[2-(naphthalen-1-ylmethyl)-1,3-dioxo-2,3-dihydro-1H-isoindol-4-yl]piperidine-4-carboxamide
2-methoxy-3-[6-(thiomorpholin-4-yl)pyridazin-3-yl]quinoline
1-(2-chloropyridin-3-yl)-3-(2,2-dimethyloxan-4-yl)-3-ethylurea
1-(3-phenylphenyl)-N-(3,3,3-trifluoropropyl)piperidin-4-amine
methyl (2S,4R)-1-[1-(2-fluorophenyl)cyclopropanecarbonyl]-4-hydroxypyrrolidine-2-carboxylate
N-[(1,3-dimethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazol-5-yl)methyl]-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-{[2-(2-methylpropanamido)ethyl]sulfamoyl}-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylic acid
2-[(4aR,7aS)-4-{[(4-methylphenyl)methyl]carbamoyl}-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]acetic acid
2-(1-{[2-cyclopropylmethanesulfonyl-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-2-yl)ethan-1-ol
3-(3-cyano-4-ethoxyphenyl)-1-[(4,6-dimethylpyridin-2-yl)methyl]-1-methylurea