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N-(1,3-dihydroxypropan-2-yl)-1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-3-carboxamide
4-{[2-(3,4-difluorophenyl)-8-methoxy-2,3,4,5-tetrahydro-1,5-benzothiazepin-5-yl]methyl}-2,6-dimethoxyphenol
methyl 2-{[(3-fluorophenyl)methyl]sulfamoyl}-6-(1-methyl-1H-pyrazole-5-carbonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
5-[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]-1-[2-(morpholin-4-yl)ethyl]piperidin-2-one
2-{5-[4-(4-chlorophenoxy)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
(3R,5S)-5-(morpholine-4-carbonyl)-N-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]ethyl}piperidine-3-carboxamide
ethyl 1-(4-phenyl-1,3-thiazol-2-yl)-5-{[(pyridin-3-ylmethyl)amino]methyl}-1H-pyrazole-4-carboxylate
5,6-dichloro-2-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-1H-1,3-benzodiazole
5-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methylpyridin-2-amine
1-(4-methoxy-3,5-dimethylphenyl)-5-oxopyrrolidine-3-carboxylic acid
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(2-methoxyphenyl)methyl]-N-(prop-2-en-1-yl)propanamide
4-{1-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]piperidin-3-yl}benzoic acid
1-[(2R,3S,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(dimethylamino)ethan-1-one
9-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]-2-[2-(pyridin-2-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
7-({7-hydroxy-2-methyl-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)-3-methyl-1-oxa-3,7-diazaspiro[4.4]nonan-2-one
3,5-dimethyl-1-(3-{1-[(1-methyl-1H-pyrazol-4-yl)methyl]-1H-imidazol-2-yl}phenyl)-1H-pyrazole
2-(morpholin-3-yl)-N-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}acetamide
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-3-phenyl-1H-pyrazole-4-carboxamide
3-[(4aS,7aR)-4-(2-methylpropanoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carbonyl]-5-fluorobenzonitrile
2-[(3S,4R)-4-amino-3-methoxypiperidin-1-yl]-6-(1-benzothiophen-2-yl)pyridine-3-carboxylic acid
N-{2-[2-(trifluoromethoxy)phenyl]ethyl}oxolane-3-carboxamide
3-methyl-8-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-(1H-imidazol-4-yl)-2-{[4-(piperidin-1-ylmethyl)phenyl]formamido}propanoic acid
2-{3-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]piperidin-1-yl}-5-methyl-4-(1-methyl-1H-pyrazol-5-yl)pyrimidine
1-{4-[4-({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)piperazin-1-yl]phenyl}ethan-1-one
N,N-dimethyl-4-(1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperazine-1-carboxamide
4-hydroxy-N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]benzamide
4-cyclobutyl-6-methyl-N-[1-(pyrazin-2-yl)propan-2-yl]pyrimidin-2-amine
5-chloro-N-{[1-(2-methylpropyl)piperidin-3-yl]methyl}-6-oxo-1,6-dihydropyridine-3-carboxamide
2-{[(7-methoxynaphthalen-2-yl)oxy]methyl}-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]-1,3-oxazole-4-carboxamide
5-{[2-(2-methoxyethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-3-(pyrrolidine-1-carbonyl)pyridine
4-{3-[1-(1,4-dioxan-2-ylmethyl)-1H-pyrazol-3-yl]phenyl}-2-(methylsulfanyl)pyrimidine
5-[(5-chloro-2-methylphenyl)carbamoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylic acid
N-[2-(3-benzyl-1,2,4-oxadiazol-5-yl)ethyl]imidazo[2,1-b][1,3]thiazole-6-carboxamide
1-[(4-methoxy-2,3-dimethylphenyl)methyl]-3-(pyrrolidin-1-yl)piperidine
1-{[3-(2H-1,3-benzodioxol-5-yl)-1-phenyl-1H-pyrazol-4-yl]methyl}-3-(pyrrolidin-1-ylmethyl)piperidine
(3aS,6aR)-5-[(5-ethylfuran-2-yl)methyl]-3-[2-(pyridin-2-yl)ethyl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
methyl 5-{[2-(pyridin-2-yl)pyrimidin-5-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
7-methyl-N-[(5-methylpyrazin-2-yl)methyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
(1S)-2-phenyl-1-[1-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]ethan-1-ol
4-[6-oxo-1-(3-phenylpropyl)piperidine-3-carbonyl]-1λ6-thiomorpholine-1,1-dione
N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-2-(1,3-thiazol-2-yl)pyrrolidine-1-carboxamide
4-hydroxy-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-2-(pyridin-2-yl)pyrimidine-5-carboxamide
N-cyclopropyl-3-{4-[2-(3,4-dihydroxyphenyl)-1H-imidazol-1-yl]phenyl}propanamide
5-[(methylsulfanyl)methyl]-3-(oxan-4-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
N-(2-{4-methyl-5-[(pyridin-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)-2-[3-(trifluoromethyl)phenyl]acetamide
N-(furan-2-ylmethyl)-N-(2-phenylethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-3-carboxamide
5-cyclohexaneamido-1-(2-methoxyethyl)-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]-1H-1,3-benzodiazole-7-carboxamide
3-methyl-7-(2-propyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-3,4-dihydroquinazolin-4-one