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methyl (2S)-1-{3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanoyl}pyrrolidine-2-carboxylate
3-[(3S,7S,8aS)-3-(4-aminobutyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2-fluorophenyl)urea
5-{[4-(2-methoxyethoxy)piperidin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
5-(1-acetylpiperidine-3-carbonyl)-N-methyl-4H,5H,6H,7H-thieno[3,2-c]pyridine-2-carboxamide
(2S,4R)-4-amino-N-ethyl-1-[1-(4-methoxyphenyl)cyclopentanecarbonyl]pyrrolidine-2-carboxamide
4-[3-(propan-2-yl)-1H-pyrazol-5-yl]-1-[3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carbonyl]piperidine
4-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
2-[4-(2H-1,3-benzodioxol-5-yl)-2-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)phenoxy]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethan-1-one
3-(2-hydroxyethyl)-4-{6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperazin-2-one
1-{[2-(4-methoxy-2,3-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1,4-diazepan-5-one
1-(4-ethoxybenzoyl)-4-(1-ethyl-1H-imidazol-2-yl)piperidine
4-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-2-(pyridin-3-yl)morpholine
3-(3-methoxybenzoyl)-1-[(2,3,4-trimethoxyphenyl)methyl]piperidine
(2R,3R)-1'-(1H-1,3-benzodiazol-2-yl)-3-[ethyl(methyl)amino]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
N,N-dimethyl-2-[(1S,5R)-3-[2-(3-methyl-1,2-oxazol-5-yl)acetyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
4-(cyclopropylmethyl)-1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}-3-(propan-2-yl)-1,4-diazepan-5-one
{[3-(2-chlorophenyl)-1-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}(oxolan-2-ylmethyl)amine
(4aS,8aR)-6-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-1-propyl-decahydro-1,6-naphthyridin-2-one
4-benzyl-1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperidin-4-ol
ethyl 2-{1-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]piperidin-2-yl}acetate
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-3-ol
3-{2-[(4-fluoro-3-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(thiophen-3-yl)propan-2-yl]propanamide
2-(4,6-dimethyl-1-benzofuran-3-yl)-1-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]ethan-1-one
2,6-dimethyl-4-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidine-1-carbonyl}quinoline
2-(2-{[4-(pyridin-3-yloxy)piperidin-1-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl)acetic acid
2-(3-phenylpropyl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]-1,3-benzoxazole-5-carboxamide
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-5-propyl-1,2-oxazole-3-carboxamide
3-(2-amino-1,3-thiazol-4-yl)-1-[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]propan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
N-ethyl-2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrimidin-4-amine
4-[3-(1H-1,3-benzodiazol-1-yl)propanoyl]-1-(3,5-dimethylphenyl)piperazin-2-one
7-(2-hydroxyethyl)-2-(2-methoxy-4-methylbenzoyl)-2,7-diazaspiro[4.5]decan-6-one
2-methyl-N4-{[1-(phenoxymethyl)cyclopropyl]methyl}pyrimidine-4,6-diamine
2-{2-[(2-ethylmorpholin-4-yl)methyl]phenoxy}ethan-1-ol
4-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-N,N-dimethylpiperazine-1-sulfonamide
4-[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]-N-propylbenzene-1-sulfonamide
N-(5-cyclopropyl-1,3,4-thiadiazol-2-yl)-3-{[1-(furan-2-yl)ethyl]amino}propanamide
1-[4-({[(4-chlorophenyl)methyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
5-cyclopropyl-1-[4-(2,5-dimethylthiophen-3-yl)pyrimidin-2-yl]-N-(2-methoxyethyl)-N-methyl-1H-pyrazole-4-carboxamide
5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]-3-(propan-2-yl)-1,2,4-oxadiazole
N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(5-methylthiophene-2-carbonyl)piperidine
1-amino-N-(2-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}ethyl)cyclopentane-1-carboxamide
1-(4-tert-butylphenyl)-4-[(1R,3S)-1-hydroxy-3-methoxy-7-azaspiro[3.5]nonan-7-yl]butan-1-one
4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidine
2-{4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-5-methyl-1H-pyrazol-1-yl}-4-(3-methoxyphenyl)pyrimidine
6-(hydroxymethyl)-N-[6-(3-methoxyphenoxy)pyridin-3-yl]-1,4-oxazepane-4-carboxamide
N-methyl-3-(2-methyl-1H-imidazol-1-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]butanamide
N-{[4-(methylsulfanyl)phenyl]methyl}-2-oxo-N-propyl-2,3-dihydro-1H-imidazole-4-carboxamide
(3aR,6aS)-N-[4-(difluoromethoxy)phenyl]-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-2-carboxamide