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1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]azetidine-2-carboxylic acid
2-(3-{[3-(2-hydroxyethyl)-4-(3-methylbut-2-en-1-yl)piperazin-1-yl]methyl}-1H-indol-1-yl)acetamide
(2R)-2-amino-1-[7-(5-chloropyridin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propan-1-one
2-[2-(1,4-oxazepan-4-yl)-2-oxoethyl]-1,2-dihydroisoquinolin-1-one
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-[9-hydroxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-(propan-2-yl)acetamide
2-amino-6-(4-hydroxy-3-methoxyphenyl)-4-(2-methoxypyrimidin-5-yl)pyridine-3-carbonitrile
3-(cyclobutylmethyl)-5-[(3-methoxyphenyl)methyl]-5-(piperidin-4-yl)imidazolidine-2,4-dione
(3aS,6aS)-2-(ethanesulfonyl)-5-[(3-ethoxyphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-(benzylamino)butanamide
N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
2-(3-fluoro-4-hydroxyphenyl)-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[(1R,2R)-2-(dimethylamino)-2,3-dihydro-1H-inden-1-yl]-1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(5-methylthiophen-2-yl)-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1H-pyrazole-5-carboxamide
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1-(2-methoxyphenyl)-1H-pyrazole-4-carboxamide
N-cycloheptyl-N-[(3-methoxyphenyl)methyl]morpholine-2-carboxamide
N-methyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-7H-pyrrolo[2,3-d]pyrimidin-4-amine
2-{4-[(4-fluoropiperidin-1-yl)methyl]phenyl}-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
1-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-amine
4-[4-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)piperidin-1-yl]-N-(propan-2-yl)pyridine-2-carboxamide
1-[4-(4-{5-fluoro-2-[(2-methoxyphenyl)methyl]-1H-1,3-benzodiazol-1-yl}piperidine-1-carbonyl)piperidin-1-yl]ethan-1-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(3-fluoro-4-methoxybenzoyl)pyrrolidin-3-yl]methanol
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(3-ethylphenyl)urea
N-(3-hydroxy-2,2-dimethylpropyl)-2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}acetamide
N-(propan-2-yl)-3-(1H-pyrazol-1-ylmethyl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]benzamide
2-[2-(1-methylpiperidin-2-yl)ethyl]-5-(pyrrolidin-1-yl)-2,3-dihydropyridazin-3-one
N-[2-(propan-2-yl)-1H-1,3-benzodiazol-5-yl]-3-(pyridin-2-yl)azetidine-1-carboxamide
2-[1-(2,2-dimethylpropyl)-3-oxopiperazin-2-yl]-N-{[3-(trifluoromethoxy)phenyl]methyl}acetamide
2-{[4-(2-chloro-6-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-imidazole
4-{4-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]piperazin-1-yl}phenol
2-methoxy-5-{2-[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]-1H-imidazol-1-yl}pyridine
4-(4-chlorophenyl)-1-[4-(pyridin-4-ylmethyl)piperazin-1-yl]butan-1-one
1-(4-methoxyphenyl)-6,6-dimethyl-N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-(4-{[4-(trifluoromethoxy)phenyl]methyl}piperazin-1-yl)-2,3-dihydro-1H-isoindole-1,3-dione
N-(2-phenoxyphenyl)-3-(pyridin-3-yl)azetidine-1-carboxamide
1-[1-(3-{2-methyl-1H-imidazo[4,5-b]pyridin-6-yl}phenyl)ethyl]pyrrolidine
2-[(dimethyl-1,2-oxazol-4-yl)methyl]-8-(3,6-dimethylpyrazin-2-yl)-2,8-diazaspiro[4.5]decan-3-one
2-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
1-methyl-2-oxo-8-(pyridazine-3-carbonyl)-1,8-diazaspiro[4.5]decane-4-carboxylic acid
2-[2-({3-[(dimethylamino)methyl]-3-hydroxypiperidin-1-yl}methyl)phenoxy]-N,N-dimethylacetamide
8-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[3-methyl-1-(propan-2-yl)-1H-pyrazol-5-yl]-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
N5,N5-diethyl-N2-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2,5-dicarboxamide
1-(2H-1,3-benzodioxol-5-yl)-5-(dimethyl-1,2-oxazol-4-yl)-3-(2-methylpropyl)-1H-1,2,4-triazole
4-(5-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-pyrazol-3-yl)pyridine
ethyl 3-(3-phenylpropyl)-1-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}piperidine-3-carboxylate
1-{3,5-dimethyl-4-[2-(4-methylpiperazine-1-carbonyl)piperazine-1-carbonyl]-1H-pyrrol-2-yl}ethan-1-one
N-benzyl-3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
methyl 5-[(7-methyl-1H-indol-3-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
N-[4-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-4-(3-methyl-1H-1,2,4-triazol-5-yl)piperidine-1-carboxamide