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1-(2-phenylethyl)-4-[3-(piperidine-1-carbonyl)pyridin-2-yl]piperazine
N-pentyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
N-{4-[3-(hydroxymethyl)-4-methoxyphenyl]phenyl}methanesulfonamide
N-(3-hydroxypropyl)-N-[(2-methoxyphenyl)methyl]-3,6-dimethyl-1-benzofuran-2-carboxamide
3-(1-methanesulfonylpiperidin-3-yl)benzoic acid
2-amino-6-(3,5-dimethyl-1H-pyrazol-4-yl)-4-(3,4,5-trimethoxyphenyl)pyridine-3-carbonitrile
2-fluoro-N-(2-{4-methyl-5-[(2-methylpropyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
4-methyl-2-(1-{5-methylpyrazolo[1,5-a]pyrimidin-7-yl}piperidin-3-yl)-1H-1,3-benzodiazole
N-(2-chloro-4-{2-[4-(propan-2-yl)morpholin-2-yl]acetamido}phenyl)propanamide
2-({methyl[3-(oxolan-2-yl)propyl]amino}methyl)quinolin-4-ol
N-{1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}-3-(thiophen-2-yl)propanamide
(1-{3-[1-(furan-3-ylmethyl)-1H-1,2,3-triazol-4-yl]phenyl}ethyl)dimethylamine
5-{4-[(8-methoxyquinolin-2-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-3-fluoro-2-methoxy-N-methylbenzamide
ethyl 4-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamido}piperidine-1-carboxylate
N-(4-{4-[(2,3-dihydro-1H-inden-2-yl)amino]piperidin-1-yl}phenyl)-3-phenylpropanamide
N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
(3R,4S)-1-(3-methoxy-2-methylbenzoyl)-4-propylpyrrolidin-3-amine
2-{1-[(4-ethylphenyl)methyl]-5-[(4-methyl-1,4-diazepan-1-yl)methyl]-1H-1,2,4-triazol-3-yl}acetamide
9-(1,2-dimethyl-1H-pyrrole-3-carbonyl)-2-[2-(pyridin-3-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[(1-cyclopropanecarbonylpiperidin-3-yl)methyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-1-[4-(pyridin-2-ylmethyl)piperazin-1-yl]ethan-1-one
1-(4-{[3-(propan-2-yloxy)propyl]amino}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl)ethan-1-one
3-(1,3-benzothiazol-2-yl)-N-[(1-ethylpiperidin-3-yl)methyl]propanamide
N3-(cyclopropylmethyl)-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-N3-propyl-1,4-dihydropyridine-3,5-dicarboxamide
6-ethyl-N-[(1-methylpiperidin-4-yl)methyl]-2-oxo-N-(2-phenylethyl)-1,2-dihydropyridine-4-carboxamide
6-({2-methyl-5-oxo-5H-[1,3]thiazolo[3,2-a]pyrimidin-7-yl}methyl)-5,6-dihydro-1,6-naphthyridin-5-one
1-[3-(1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-2-(benzyloxy)ethan-1-one
N-[(4-chlorophenyl)methyl]-N-[2-(cyclohex-1-en-1-yl)ethyl]-2-(morpholin-2-yl)acetamide
2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]acetamide
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-methyl-3-(pyrrolidin-1-yl)propan-1-one
5-ethyl-2-methyl-N-({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)pyrimidin-4-amine
N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
7-(2-methoxyethyl)-2-(1H-pyrrole-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
(3aR,6aR)-2-cyclopentyl-N-{[1-(methoxymethyl)cyclopropyl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-propanamidobenzamide
N-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
{2-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]-2-oxoethyl}urea
2-(4-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrazine
9-{[4-(difluoromethoxy)phenyl]methyl}-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
[(2S)-1-{2-phenylimidazo[1,2-a]pyridine-6-carbonyl}pyrrolidin-2-yl]methanol
5-[2-(2-aminoethyl)morpholin-4-yl]-2-[3-(pyridin-3-yl)propyl]-2,3-dihydropyridazin-3-one
2-{2-[(dimethylamino)methyl]phenyl}-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-cyclohexyl-N-[2-(1H-indol-3-yl)ethyl]-2-methyl-1,3-thiazole-4-carboxamide
3-{4-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl}propanoic acid
N-[3-(1H-indazol-1-yl)propyl]-2,6-dioxo-1,2,3,6-tetrahydropyrimidine-4-carboxamide
3-{[1-(2-chlorobenzoyl)pyrrolidin-3-yl]methyl}benzamide
2-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-ylmethyl]-3H,4H-thieno[3,2-d]pyrimidin-4-one
7-chloro-4-hydroxy-N-[(1S,2R)-2-[(oxan-4-yl)amino]cyclobutyl]quinoline-3-carboxamide
N-cyclopentyl-N'-(3,4-dihydro-2H-1,5-benzodioxepin-7-ylmethyl)butanediamide