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3-[2-(1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}piperidin-2-yl)ethyl]phenol
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-4-methyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]benzamide
1-[(3R,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-4-phenylbutan-1-one
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
ethyl 2-(2-{5-[(pyridin-4-ylmethyl)carbamoyl]thiophen-2-yl}pyrrolidin-1-yl)acetate
N-{[4-methoxy-3-(thiophen-3-ylmethoxy)phenyl]methyl}-4-methyl-N-(pyridin-2-ylmethyl)benzamide
N-[1-(4-chlorophenyl)ethyl]-3-{5-[2-(4-methoxyphenyl)ethyl]-1,3,4-oxadiazol-2-yl}propanamide
6-{[benzyl(1,3-thiazol-2-ylmethyl)amino]methyl}-1,4-oxazepan-6-ol
N-(3-fluorophenyl)-4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidine-1-carboxamide
(3R,5S)-N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-5-(pyrrolidine-1-carbonyl)piperidine-3-carboxamide
3-[(1S,9aR)-octahydro-1H-quinolizin-1-yl]-1-[4-(pyridin-4-yl)piperazin-1-yl]propan-1-one
N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)piperidin-4-yl]methyl}-4-(pyrrolidin-1-yl)butanamide
1-[(2S)-2-[3-(2,3-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]pyrrolidin-1-yl]ethan-1-one
5-methyl-N-(3-methylbutyl)-4-(4-methylpiperazin-1-yl)thieno[2,3-d]pyrimidine-6-carboxamide
3-hydroxy-3-({methyl[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
(2R,3R)-2-hydroxy-3-(morpholin-4-yl)-N-propyl-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-carboxamide
1-[(3-{[1-(benzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
(2R,3R)-3-{[2-(1,3-benzothiazol-2-yl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{[5-(3-chlorophenyl)furan-2-yl]methyl}-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)-N-{[1-(piperidin-1-yl)cyclohexyl]methyl}acetamide
2-(2,3-dihydro-1,4-benzodioxin-6-yl)-6,7-dimethoxyquinazolin-4-amine
5-({5-methyl-2-[4-(methylsulfanyl)phenyl]-1,3-oxazol-4-yl}methyl)-4H,5H,6H,7H-[1,3]thiazolo[5,4-c]pyridin-2-amine
N-cyclopentyl-4-(2,4-dimethoxypyrimidin-5-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-1,2-dihydroquinoxalin-2-one
N-(3-cyclopentylpropyl)-5-[(4-hydroxypiperidin-1-yl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
2-[4-(4-benzyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]pyrazine
4-(piperidin-1-yl)-N-[1-(pyridin-4-yl)propyl]butanamide
3-(5-methylfuran-2-yl)-N-[1-(thiophen-2-ylmethyl)piperidin-4-yl]-1H-pyrazole-5-carboxamide
1-[(4aR,8aS)-1-(1H-indole-2-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-3-(pyridin-3-yl)propan-1-one
3-[3-(4-fluorophenyl)pyrrolidine-1-carbonyl]-1-methyl-6-(propan-2-yl)-1,2-dihydropyridin-2-one
N-(6-methoxy-2H-1,3-benzodioxol-5-yl)-2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carboxamide
N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
5-(2-methylpropyl)-1-(2-phenylethyl)-N-(pyridin-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
5-(3-propoxypiperidine-1-carbonyl)-2-(pyridin-2-yl)pyrimidin-4-ol
(2S,4R)-4-{4-[(1-furan-2-yl-N-methylformamido)methyl]-1H-1,2,3-triazol-1-yl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl](methyl)[(2-methyl-2,3-dihydro-1H-isoindol-5-yl)methyl]amine
2-[3-(dimethylamino)pyrrolidin-1-yl]-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
1-(2-oxo-2-{5-propanoyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}ethyl)imidazolidine-2,4-dione
(3R,5S)-5-{[(6-methylpyridin-3-yl)oxy]methyl}-N-[2-(1-methylpyrrolidin-2-yl)ethyl]-1-(naphthalen-2-ylmethyl)piperidine-3-carboxamide
2-{5-cyclopropyl-4-[4-(propan-2-yl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-4-(3-methoxyphenyl)pyrimidine
1-(1,3-thiazol-4-ylmethyl)-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-cyclohexyl-5-{[4-(3-methoxybenzoyl)piperazin-1-yl]methyl}pyrimidine
5-chloro-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-1,3-dimethyl-1H-pyrazole-4-sulfonamide
ethyl 4-[(1-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)amino]piperidine-1-carboxylate
4-(hydroxymethyl)-1-[(4-methyl-1H-imidazol-5-yl)methyl]azepan-4-ol
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-2-(ethylamino)-N-methylpyrimidine-5-carboxamide
8-[(3-methyl-1,2-oxazol-5-yl)methyl]-1-oxa-8-azaspiro[4.6]undecan-9-one
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-(3-hydroxypiperidin-1-yl)acetamide
4-hydroxy-1-(3-methoxypyrazin-2-yl)piperidine-4-carboxylic acid
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-pyrrole-2-carboxamide