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4-methyl-N-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-1,4-diazepane-1-carboxamide
5-{1-[(2-methyl-1,3-thiazol-4-yl)methyl]-1H-imidazol-2-yl}-3-phenyl-1,2-oxazole
(3R,4S)-4-[ethyl({[4-(1H-imidazol-1-yl)phenyl]methyl})amino]oxolan-3-ol
1-[(5-chloro-2-propoxyphenyl)methyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
6-[1-benzyl-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-2-methyl-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
propan-2-yl 3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine-1-carboxylate
5-{1-[2-(4-methoxyphenyl)ethyl]-1H-pyrazol-3-yl}-4-methyl-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-1,3-thiazol-2-amine
N-[5-(2-ethoxypyridin-3-yl)quinolin-8-yl]acetamide
N-(3-ethylphenyl)-8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
(3aS,6aS)-2-(2,3-dihydro-1H-inden-2-yl)-5-[(4-methyl-1H-imidazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-tert-butyl-4-hydroxy-N-(2-methyl-4,5,6,7-tetrahydro-1,3-benzothiazol-4-yl)pyrimidine-5-carboxamide
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)acetamide
1-(cyclohexylmethyl)-5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-4-oxo-N-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
3-[(3S,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidine-1-carbonyl]-1,2-dihydroquinoxalin-2-one
2-[(3R,4R)-4-ethyl-3,4-dihydroxypiperidin-1-yl]-N-(1-methyl-1H-pyrazol-3-yl)acetamide
2-(cyclopentylmethyl)-6-methyl-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-4-oxo-1-(pyridin-3-ylmethyl)-1,4-dihydropyridine-3-carboxamide
1-methyl-5-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
2-{[3-(1H-1,3-benzodiazol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}-4-methyl-1,2-dihydrophthalazin-1-one
2-{2-[1-(7-fluoro-4-methylquinolin-2-yl)piperidin-4-yl]-1H-imidazol-1-yl}acetamide
4-(1H-imidazol-1-yl)-1-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}piperidine-4-carboxylic acid
N,1-dimethyl-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1H-indole-6-carboxamide
methyl 9-[2-(2-fluorophenyl)ethoxy]-7-oxo-3-[3-(1H-1,2,4-triazol-1-yl)propanoyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[2-oxo-2-(2-propyl-2,5-dihydro-1H-pyrrol-1-yl)ethyl]-3,4-dihydro-2H-1,4-benzoxazin-3-one
4-chloro-3-[({[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}carbamoyl)amino]-N-propylbenzamide
2-(2H-1,3-benzodioxol-5-yl)-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(dimethyl-1,3-thiazol-5-yl)-N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]acetamide
N-({2-[benzyl(methyl)amino]pyridin-3-yl}methyl)morpholine-2-carboxamide
N-(3-chloro-4-methoxyphenyl)-3-[4-(1-methyl-1H-pyrazol-4-yl)-1,2,3,6-tetrahydropyridin-1-yl]propanamide
(1R,5R)-3-(3-chloro-5-fluorobenzoyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-{1-[(4-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-methoxyethyl)acetamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-N'-[2-(propan-2-yl)phenyl]butanediamide
6-methyl-N-[3-(methylsulfanyl)propyl]-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N-(1H-indol-7-ylmethyl)-N-(pyridin-2-ylmethyl)cyclopropanamine
1-[5-(2-methoxypyridin-3-yl)thiophen-2-yl]-2-methylpropan-1-one
N-(1,3-benzothiazol-2-ylmethyl)-2-ethyl-N,4-dimethyl-1,3-oxazole-5-carboxamide
1-{[2-(cycloheptanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
1-(1-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}pyrrolidin-3-yl)-3,5-dimethyl-1H-pyrazole
2-(oxolane-3-carbonyl)-N-(pyridin-3-yl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
1-butyl-5-(thiophen-3-yl)-1H,4H-pyrazolo[3,4-d]imidazole
4-{[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenyl]methyl}-2-phenylmorpholine
(4aR,7aS)-1-acetyl-4-(4-methyl-1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
[1-(1H-imidazol-4-ylmethyl)piperidin-4-yl]diphenylmethanol
N-[(3-chlorophenyl)methyl]-N-methyl-2-{2-oxo-1-oxa-3,8-diazaspiro[4.5]decan-3-yl}acetamide
N-cyclopropyl-1-[3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanoyl]piperazine-2-carboxamide
(3S,4R)-4-(2,3-dimethoxyphenyl)-1-[3-(1H-imidazol-1-yl)propyl]pyrrolidine-3-carboxylic acid
N-cyclopentyl-N-{[3,5-dimethoxy-4-(oxolan-2-ylmethoxy)phenyl]methyl}-3-(2-oxopyrrolidin-1-yl)benzamide
4-({3-[4-(prop-2-en-1-yl)piperazine-1-carbonyl]-1,2-oxazol-5-yl}methyl)morpholine
N-(2-methoxyethyl)-4-[(1-methyl-6-oxopiperidin-3-yl)sulfamoyl]benzamide
N-{[4-(4-fluorophenyl)-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}-2,4-dimethoxybenzamide
N-(2-{3-methyl-7-oxo-7H-[1,3]thiazolo[3,2-b][1,2,4]triazin-6-yl}phenyl)-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide