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ethyl 4-{[(2,2-dimethyloxan-4-yl)(ethyl)carbamoyl]amino}benzoate
6-methoxy-N-(2-methylpropyl)-N-[(3-methylthiophen-2-yl)methyl]-4-oxo-1,4-dihydroquinoline-3-carboxamide
cyclopentyl 4-({[3-oxo-3-(pyrrolidin-1-yl)propyl]carbamoyl}amino)benzoate
3-(3-methoxyphenyl)-N-{2-[(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)amino]ethyl}-1H-pyrazole-4-carboxamide
2-(ethylamino)-4-methyl-N-[(2,3,6-trifluorophenyl)methyl]-1,3-thiazole-5-carboxamide
2-{[8-methyl-2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
1-ethyl-4-{4-[2-(3-methoxyphenoxy)ethyl]piperazine-1-carbonyl}pyrrolidin-2-one
4-chloro-1-methyl-3-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-indazole
N-[2-(dimethyl-1,3-thiazol-2-yl)ethyl]-5-(3-methoxyphenoxymethyl)-1,2-oxazole-3-carboxamide
2-(2-phenyl-1H-imidazol-1-yl)-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]acetamide
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-[1-(1,3-thiazol-2-yl)ethyl]piperidin-4-amine
3-{3-[cyclohexyl(methyl)amino]propyl}-8-[(2R)-2-hydroxypropanoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(3-aminopyrrolidine-1-carbonyl)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]benzene-1-sulfonamide
9-(2,1,3-benzothiadiazol-5-ylmethyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
3-({2-[1-(5-methylthiophene-2-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
3-[(4aR,7aS)-4-(3-hydroxy-4-methylbenzoyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-methyl-3-({methyl[(3-methyl-1,2-oxazol-5-yl)methyl]amino}methyl)-1,2-dihydroquinolin-2-one
9-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-2-(2-methylpropyl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carboxamide
4-[(4,5-dimethylfuran-2-yl)methyl]-1-[(3-methoxyphenyl)methyl]piperazin-2-one
(1R,3S)-3-{ethyl[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]carbamoyl}cyclopentane-1-carboxylic acid
2-methyl-N-{[3-(pyridin-3-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}aniline
1-(5-chloro-2-methoxybenzoyl)-3-(1-ethyl-1H-imidazol-2-yl)piperidine
2-[5-(4-methoxyphenyl)furan-2-carbonyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl][(8-methoxyquinolin-5-yl)methyl]methylamine
{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}({[2-(3-methylphenyl)pyrimidin-5-yl]methyl})amine
2-[3-(2H-1,3-benzodioxol-5-yl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]acetamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(pyridine-4-carbonyl)pyrrolidin-3-amine
1-{4-[2-(methoxymethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidin-1-yl}-2-phenoxypropan-1-one
N-(1,2-oxazol-3-ylmethyl)-2-[(quinolin-8-yloxy)methyl]-1,3-oxazole-4-carboxamide
2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-[(4-methoxyphenyl)methyl]-N-propylacetamide
N-(5-fluoro-2-methylphenyl)-2-({1-methyl-1H-pyrazolo[1,5-a]imidazol-7-yl}formamido)propanamide
N-({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)-N,2-dimethylpyrimidine-5-carboxamide
1-methyl-4-({5-[2-(1H-1,2,4-triazol-3-yl)phenyl]-1,2,4-oxadiazol-3-yl}methyl)piperidine
(1S,4S)-2-(3,4-difluorophenyl)-5-[2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)acetyl]-2,5-diazabicyclo[2.2.1]heptan-3-one
3-tert-butyl-1-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]urea
(2S,4R)-N-ethyl-4-[2-(2-methyl-1H-imidazol-1-yl)acetamido]-1-[(5-methylfuran-2-yl)methyl]pyrrolidine-2-carboxamide
N-[1-(1-cyclopropylethyl)-4-methyl-1H-pyrazol-5-yl]pyridine-4-carboxamide
[(3R,4R)-4-{[4-(hydroxymethyl)piperidin-1-yl]methyl}-1-[6-methyl-2-(methylamino)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
(4aS,7aR)-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-N-(1,1-dioxo-1λ6-thiolan-3-yl)-1-[(3-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carboxamide
(4aS,7aR)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-3-(3-hydroxy-1,2-oxazol-5-yl)propan-1-one
N-cyclohexyl-4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
1-[3-(2-{[benzyl(ethyl)amino]methyl}-4-methoxyphenoxy)-2-hydroxypropyl]piperidin-4-ol
(1R,5R)-3-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
9-methanesulfonyl-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
1-[1-(2,6-dimethylhept-5-en-1-yl)piperidin-4-yl]-N-(2-methoxyethyl)-1H-1,2,3-triazole-4-carboxamide
N-[(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)methyl]ethane-1-sulfonamide
N-[1-(naphthalen-1-ylmethyl)-5-oxopyrrolidin-3-yl]-3-(pyrazin-2-yl)propanamide