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8-(2-hydroxyethyl)-2-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-3-one
3-[(1R,5R)-6-benzyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-4,6-dimethyl-1,2-dihydropyridin-2-one
N-{2-[cyclopentyl(methyl)amino]ethyl}-1-(4-methoxyphenyl)-N,2,2-trimethylcyclopropane-1-carboxamide
N-[3-(oxolan-3-yl)propyl]-1-(pyrimidin-2-yl)piperidin-4-amine
9-(dimethyl-1,3-oxazole-5-carbonyl)-2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecane
2-[(3-cyclohexyl-1H-pyrazol-4-yl)methyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decane
4-{[(2,3-dimethoxyphenyl)methyl]amino}-N-(2-methoxyethyl)-N,5-dimethylthieno[2,3-d]pyrimidine-6-carboxamide
N-[(5-chloro-2-propoxyphenyl)methyl]-5-methoxy-4-oxo-1,4-dihydropyridine-2-carboxamide
N-{1-[1-(1,4-dithiepan-6-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2H-1,3-benzodioxole-5-carboxamide
2-fluoro-N-[4-(4-{[2-(1H-indol-1-yl)ethyl]amino}piperidin-1-yl)phenyl]benzamide
(4S,4aS,8aR)-4-hydroxy-4-phenyl-N-(1,3,4-thiadiazol-2-yl)-decahydroquinoline-1-carboxamide
(1R,9aR)-1-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-octahydro-1H-quinolizin-1-ol
(2S,4R)-1-[(2-aminopyridin-3-yl)methyl]-N-ethyl-4-(furan-3-amido)pyrrolidine-2-carboxamide
8-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
(3aR,6aR)-2-cyclobutanecarbonyl-5-(3-methylbenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-methyl-9-(prop-2-en-1-yl)-4-(9H-purin-6-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
4-ethyl-6-(4-{[5-(1H-1,2,4-triazol-5-ylsulfanyl)furan-2-yl]methyl}piperazin-1-yl)pyrimidine
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
ethyl 3-{[(1-cycloheptyl-5-oxopyrrolidin-3-yl)carbamoyl]amino}propanoate
N-{1-[2-(3-chlorophenyl)ethyl]-5-oxopyrrolidin-3-yl}-2-(2-methyl-1,3-thiazol-4-yl)acetamide
5-methyl-N-{[3-(oxolan-3-ylmethoxy)phenyl]methyl}-N-(pyridin-2-ylmethyl)thiophene-2-carboxamide
N-{[5-(5-acetylthiophen-2-yl)-7-chloro-2,3-dihydro-1-benzofuran-2-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
4-[3-({[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}amino)propyl]-1,3-thiazol-2-amine
[(3R,4R)-1-(3,5-dichloropyridin-2-yl)-4-[(4-ethylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
N-[(3S,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-bromobenzamide
(oxolan-2-ylmethyl)[(1-phenyl-1H-1,2,3-triazol-4-yl)methyl](pyridin-2-ylmethyl)amine
N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-2-(pyridin-2-yl)acetamide
2-{5-[3-(2-phenylethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazol-1-yl}ethan-1-ol
3-cyclopropyl-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-1H-pyrazole-5-carboxamide
8-(5-propylpyrimidin-4-yl)-2-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-(2-phenyl-1H-imidazol-1-yl)acetamide
1-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
1-{4-[(1,3-dihydroxypropan-2-yl)amino]-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
5-methyl-N-[(2-methylphenyl)(thiophen-2-yl)methyl]-1,3,4-oxadiazole-2-carboxamide
4-[1-(2-ethoxyethyl)-3-methyl-1H-pyrazole-5-carbonyl]-1-(4-methylphenyl)piperazin-2-one
6-methyl-4-oxo-N-(oxolan-2-ylmethyl)-N-(pyridin-2-ylmethyl)-4H-pyran-2-carboxamide
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-fluoro-4-methylquinoline
3-benzyl-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
4-(1H-1,3-benzodiazol-1-yl)-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-4-carboxylic acid
2-methoxy-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)acetamide
2-[4-(2-chloro-6-fluoro-3-methylbenzamido)-3,5-dimethyl-1H-pyrazol-1-yl]acetic acid
4-methyl-2-[4-(3-methylpyridin-4-yl)piperazin-1-yl]quinazoline
N-[3-({methyl[1-(1,3-thiazol-2-yl)ethyl]carbamoyl}methoxy)phenyl]propanamide
N-[(2S)-1-methoxypropan-2-yl]-3-{[2-oxo-2-(pyrrolidin-1-yl)ethyl]sulfamoyl}benzamide
(2S,4R)-1-(cyclohexylmethyl)-N-(2-methylpropyl)-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carboxamide
3-(dimethyl-1,2-oxazol-4-yl)-1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-methylurea
2-cyclohexyl-N-methyl-N-[3-(1-methyl-1H-imidazol-2-yl)propyl]-1,3-benzoxazole-6-carboxamide
3-{[1-(3-fluorophenyl)-3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}morpholine
N-{1-[(4-methylphenyl)methyl]cyclopropyl}-2-(thiophen-2-yl)acetamide
4-acetyl-N-{1-[(2-chlorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzamide