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4-{[1-tert-butyl-3-(pyridin-3-yl)-1H-1,2,4-triazol-5-yl](pyridin-3-yl)methyl}morpholine
9-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(thiophen-2-yl)acetamide
N-(2,2-dimethyloxan-4-yl)-2-oxo-6-[(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)methyl]-1,2-dihydropyridine-3-carboxamide
N-(furan-2-ylmethyl)-5,6-dimethyl-N-{[2-(morpholin-4-yl)-6H,7H,8H-cyclopenta[g]quinolin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
4-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(3S,7S,8aS)-7-(benzylamino)-3-[(4-hydroxyphenyl)methyl]-octahydropyrrolo[1,2-a]piperazine-1,4-dione
4-[(2-methoxynaphthalen-1-yl)methyl]-11-[(2-methylpropyl)amino]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
8-methoxy-3-(5-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-3,4-dihydroquinazolin-4-one
2-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-N,6-dimethylpyrimidin-4-amine
4-[3-(acetamidomethyl)phenyl]-N,N-diethylbenzamide
1-(2,3-difluoro-4-methoxybenzoyl)-3-(3-ethylphenoxy)azetidine
3-{methyl[3-oxo-3-(3-oxo-4-phenylpiperazin-1-yl)propyl]amino}-1λ6-thiolane-1,1-dione
N-[(4-fluorophenyl)(pyridin-4-yl)methyl]-2-(methylamino)-1,3-thiazole-4-carboxamide
2-(4-methoxynaphthalen-1-yl)-5-methyl-4-({1-methyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}methyl)-1,3-oxazole
1-phenyl-4-{[(5-propyl-1,3,4-oxadiazol-2-yl)amino]methyl}pyrrolidin-2-one
2,6-difluoro-4-methoxy-N-(oxolan-3-yl)benzamide
8-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-[3-(4-{[4-(2-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]oxolane-2-carboxamide
N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-4-(1H-pyrazol-1-ylmethyl)piperidine-1-carboxamide
2-[1-(2,3-dihydro-1H-inden-2-yl)-3-oxopiperazin-2-yl]-N-[2-(3-methoxyphenyl)ethyl]acetamide
(4S)-3,3,4-trimethyl-1-{[4-(pyridin-2-ylmethoxy)phenyl]methyl}piperidin-4-ol
N-[(2-{2-[(dimethylsulfamoyl)amino]phenyl}-5-methyl-1,3-oxazol-4-yl)methyl]thiophene-2-carboxamide
2-[(3,4-dimethoxyphenyl)methyl]-N-[3-(pyridin-3-yloxy)propyl]-1,3-benzoxazole-6-carboxamide
N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
3-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-6,8-dimethyl-3,4-dihydroquinazolin-4-one
N-[2-(1H-indol-1-yl)ethyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
3-benzyl-5-(2-ethoxyphenyl)-1H-1,2,4-triazole
2-{4-[(2,4-dimethoxy-3-methylphenyl)methyl]piperazin-1-yl}pyridine-3-carboxamide
7-cyclopentyl-2-[2-(2H-1,2,3-triazol-2-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
4-(2-methoxyphenoxy)-1-{[5-(oxan-2-yl)furan-2-yl]methyl}piperidine
2-[5-(methoxymethyl)-4-(4-propylpiperazine-1-carbonyl)-1H-pyrazol-1-yl]-4-(thiophen-2-yl)pyrimidine
10-[4-(4-chlorophenyl)piperazine-1-carbonyl]-1-azatricyclo[6.3.1.04,12]dodeca-4(12),5,7,10-tetraen-9-one
[1-ethyl-5-(1H-imidazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl]methanol
methyl[2-(3-{[(2S,5R)-5-(thiomorpholin-4-ylmethyl)oxolan-2-yl]methyl}phenoxy)ethyl]amine
N-cyclobutyl-3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)benzene-1-sulfonamide
3-(oxolan-3-yl)-5-[4-(1H-pyrazol-3-yl)phenyl]-1,2,4-oxadiazole
1-ethyl-3-[1-(2-hydroxyethyl)-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl]-4,6-dimethyl-1,2-dihydropyridin-2-one
4-[(2,4-dimethyl-1H-imidazol-1-yl)methyl]-2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazole
1-(2-methoxyacetyl)-N-{[1-(2-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-3-carboxamide
4-{[4-(4-ethyl-1H-pyrazol-5-yl)piperidin-1-yl]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-(4-fluoro-2-methylphenyl)-3-(1-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}piperidin-3-yl)propanamide
2-(4-fluorophenyl)-4-[3-(pyrrolidine-1-carbonyl)pyridin-2-yl]morpholine
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-(naphthalen-1-ylmethyl)pyrrolidin-3-yl]methanol
1-{4-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidine-1-carbonyl]thiophen-2-yl}ethan-1-one
N-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}thiophene-2-sulfonamide
3-{1-[3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carbonyl]piperidin-2-yl}pyridine
(3S,4R)-1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
N4-{3-[(pyridin-3-yl)amino]propyl}-5,6,7,8-tetrahydroquinazoline-2,4-diamine
methyl 5-{2-[(dimethyl-1H-1,2,4-triazol-1-yl)methyl]propanoyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate