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3-[(3R,4S)-1-(isoquinolin-1-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(3-chloro-1,2-oxazol-5-yl)-N-[(1-cyclopentylpiperidin-3-yl)methyl]propanamide
8-cyclopropanecarbonyl-2-(2-phenylethyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}cyclopropanecarboxamide
2-(2,2-dimethylpropanamido)-5-methyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]thiophene-3-carboxamide
4-(pyridine-4-carbonyl)-2-{[3-(trifluoromethyl)phenyl]methyl}morpholine
(2-chloro-6-fluorophenyl)(4-{[5-(methoxymethyl)furan-2-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methanol
4-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-11-{[(3,4,5-trifluorophenyl)methyl]amino}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
1-[(3-fluorophenyl)methyl]-4-{2-[3-(methylsulfanyl)phenyl]acetyl}piperazin-2-one
4-(furan-3-carbonyl)-9-methoxy-7-[4-(methylsulfanyl)phenyl]-2,3,4,5-tetrahydro-1,4-benzoxazepine
2-{[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrol-5-yl]methyl}-6-methylquinolin-4-ol
N-benzyl-N-(3-hydroxy-2-methylpropyl)-6-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
N,N-dimethyl-6-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyrazin-2-amine
4-{[2-(2-methoxyphenyl)pyrrolidin-1-yl]methyl}-5-methyl-2-(thiophen-3-yl)-1,3-oxazole
1-{1-[(3-chlorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperidin-3-ol
3-{4-methyl-2-[2-(morpholin-4-ylmethyl)phenyl]phenyl}-1,3-oxazolidin-2-one
3-[2-(3-{[3-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-2-oxoethyl]-3,4-dihydroquinazolin-4-one
N-{2-[4-(4-methoxyphenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]ethyl}-2H-1,3-benzodioxole-5-carboxamide
5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
N'-(2,4-dimethylphenyl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]propanediamide
N-(butan-2-yl)-2,7-dimethyl-N-(pyridin-3-ylmethyl)pyrazolo[1,5-a]pyrimidine-5-carboxamide
2-(4-methylphenoxy)-N-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}acetamide
N-cycloheptyl-3-[methyl({[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]propanamide
N-{2-[(2S)-2-hydroxy-2-phenylacetamido]-4-methylphenyl}pentanamide
1-(1'-{[3-(2-hydroxyethoxy)phenyl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl)ethan-1-one
3-butyl-1-methyl-4-[2-(phenylamino)pyrimidine-5-carbonyl]piperazin-2-one
N-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-5-(pyrrolidin-2-yl)thiophene-2-carboxamide
(3R,4R)-3-cyclopropyl-4-methyl-1-(1-phenylpiperidin-4-yl)pyrrolidin-3-ol
2-{[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-3-yl]methyl}-1H-1,3-benzodiazole
2-{[3-(3-methoxyphenyl)-1H-pyrazol-4-yl]formamido}-N-methyl-2-phenylacetamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
[1-({1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
1-cyclohexyl-4-(5-ethylpyrimidin-2-yl)piperazin-2-one
2-(4-chloro-2-methylphenoxy)-N-methyl-N-[1-(pyridin-3-yl)ethyl]acetamide
4-{[3-(2,6-dimethylphenoxy)azetidin-1-yl]methyl}pyridine
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-6-methoxy-N-methylpyrimidin-4-amine
4-[(5,6-dimethoxy-1-oxo-1,2-dihydroisoquinolin-2-yl)methyl]benzamide
ethyl 1-(cyclohex-3-en-1-ylmethyl)-4-{[3-(trifluoromethyl)phenyl]methyl}piperidine-4-carboxylate
N-[3-(2-chlorophenoxy)propyl]-N,5-dimethyl-1,3-oxazole-4-carboxamide
N-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-4-(1H-pyrrole-2-carbonyl)piperazine-1-carboxamide
3-[(2R,3R,6R)-5-(2,4-dimethylpyrimidine-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-3-yl]phenol
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridine-4-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-4-(piperidin-1-ylmethyl)benzamide
2-amino-4-(2,1,3-benzoxadiazol-4-yl)-6-(pyrimidin-2-yl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-(4-hydroxyphenyl)-2-[methyl(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)amino]acetic acid
4-{3-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}-1H-pyrazolo[3,4-d]pyrimidin-6-amine
2-(5-tert-butyl-2H-1,2,3,4-tetrazol-2-yl)-N-{1,4,6-trimethyl-1H-pyrazolo[3,4-b]pyridin-3-yl}acetamide
1-{[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-indole
N-{[(2S,4S)-4-fluoropyrrolidin-2-yl]methyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
4-{[2-(2-fluorophenyl)-2-hydroxyethyl]amino}pyrimidine-5-carboxylic acid