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3-(2,2-diphenylethyl)-5-(oxolan-3-yl)-1,2,4-oxadiazole
5-{1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-1H-imidazol-2-yl}-2-(pyrrolidin-1-yl)pyrimidine
methyl[(5-phenyl-1,2-oxazol-3-yl)methyl]{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}amine
1-(2,6-dimethylpyridin-4-yl)-4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperazine
N-({5-[(3-fluoro-2-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)methanesulfonamide
1-{1-[1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carbonyl]azetidin-3-yl}piperidine
11-{[3-(propan-2-yloxy)propyl]amino}-4-{[3-(trifluoromethyl)phenyl]methyl}-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-methyl-N-(3-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetamido}phenyl)benzamide
1,3,6-trimethyl-N-{[1-(2-methylpropyl)piperidin-4-yl]methyl}-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-({[2-(2,5-difluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(2-hydroxyethyl)amino)ethan-1-ol
3-{[4-(2-hydroxypropan-2-yl)piperidin-1-yl]methyl}-7-methyl-1,2-dihydroquinolin-2-one
methyl N-{2-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]-2-oxoethyl}carbamate
6-(pyrrolidin-1-ylmethyl)-4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]-1,4-oxazepan-6-ol
N-(furan-2-ylmethyl)-6-methoxy-N-methyl-3,4-dihydro-2H-1-benzopyran-3-carboxamide
2-[2,4-bis(morpholin-4-yl)pyrimidin-5-yl]-2-methylpropanoic acid
8-hexanoyl-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
(3R,4S)-1-[4-(4-fluorophenyl)-1,3-thiazol-2-yl]-4-propylpyrrolidin-3-amine
5-{3-[({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)methyl]pyrrolidin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
(3R,4S)-4-[ethyl({[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amino]oxolan-3-ol
(4aS,8aR)-6-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-1-[2-(thiophen-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
1-propyl-4-(4-{[1-(pyridin-2-ylmethyl)piperidin-4-yl]oxy}benzoyl)piperazine
1-methyl-N-(propan-2-yl)-N-[(2,4,5-trimethoxyphenyl)methyl]-1H-pyrrole-2-carboxamide
5-(2-fluoro-4,5-dimethoxyphenyl)-1-phenyl-1H,4H-pyrazolo[3,4-d]imidazole
2-(dimethylamino)-1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
(3S,4S)-1-(3-carbamoylpyridin-2-yl)-4-cyclopropylpyrrolidine-3-carboxylic acid
6-fluoro-N-methyl-2-oxo-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1,2-dihydroquinoline-4-carboxamide
(4aS,8aR)-1-(3-methoxypropyl)-6-(3-methylfuran-2-carbonyl)-decahydro-1,6-naphthyridin-2-one
methyl 1-[(4-cyclopentanecarbonyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)methyl]piperidine-4-carboxylate
ethyl 2-[3-(2-hydroxyethyl)-4-[(6-methylpyridin-2-yl)methyl]piperazin-1-yl]-1,3-oxazole-4-carboxylate
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
2-methyl-N-(2-phenoxyethyl)-2,8-diazaspiro[4.5]decane-3-carboxamide
1-{4-[4-ethyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(propan-2-ylsulfanyl)ethan-1-one
1-(2,3-dihydro-1-benzofuran-7-carbonyl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-2-(7-fluoro-2-methyl-1H-indol-3-yl)acetamide
5-methyl-2-(4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}piperazin-1-yl)-1,3-benzoxazole
N-[3-(1H-indazol-1-yl)propyl]-2-oxo-6-phenyl-1,2-dihydropyridine-3-carboxamide
N-phenyl-3-{2-[1-(piperidin-4-yl)-1H-1,2,3-triazol-4-yl]-1H-imidazol-1-yl}propanamide
2-(ethoxymethyl)-N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
4-[4-(2,2-dimethylpropyl)piperazin-1-yl]-2-(3-methoxypropyl)-2,3-dihydro-1H-isoindole-1,3-dione
2-[4-(hydroxymethyl)phenyl]-1-[3-(4-methoxyphenoxymethyl)piperidin-1-yl]ethan-1-one
N-(3-methoxyphenyl)-1-{2-[(2-methylpropyl)amino]ethyl}-1H-1,2,3-triazole-4-carboxamide
5-(methoxymethyl)-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-N-{[1-(morpholin-4-yl)cyclopentyl]methyl}-1H-pyrazole-4-carboxamide
[(3R,4R)-4-(piperidin-1-ylmethyl)-1-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]pyrrolidin-3-yl]methanol
5-{2-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
3-{2-[4-(1H-imidazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
N-[3-(1H-1,3-benzodiazol-2-yl)propyl]-N'-(3-ethylphenyl)butanediamide
3-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-4,5,6-trimethyl-1,2-dihydropyridin-2-one
3-(2-fluorophenyl)-3-phenyl-1-(pyrrolidin-1-yl)propan-1-one
N-[(4-fluorophenyl)methyl]-3-[1-(1H-indol-2-ylmethyl)piperidin-4-yl]propanamide
3-{1-[(4-fluorophenyl)methyl]-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-5-yl}-5-(propan-2-yl)-1,2,4-oxadiazole