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N-{[2-(1H-1,3-benzodiazol-1-yl)pyridin-3-yl]methyl}-2-(phenylsulfanyl)acetamide
1-(furan-2-ylmethyl)-N-[3-(pyridin-4-yl)propyl]piperidine-3-carboxamide
1-cyclohexyl-N-methyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
1-[(3,4-dihydroxyphenyl)methyl]-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
1-(1-butyl-1H-pyrazol-5-yl)-3-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]urea
methyl (3aS,6aS)-2-({3-[(dimethylamino)methyl]-4-hydroxyphenyl}methyl)-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylate
1'-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
3-({3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
N-{2-[methyl(phenyl)amino]ethyl}-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
4-{3-[(3-chlorophenyl)methyl]-1-(2-hydroxyethyl)-1H-1,2,4-triazol-5-yl}-1-oxaspiro[4.4]nonan-2-one
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[2-(pyridin-3-yl)pyrimidine-5-carbonyl]piperidin-3-ol
N-({8-[3-(1H-pyrazol-4-yl)benzoyl]-1-oxa-8-azaspiro[4.5]decan-2-yl}methyl)acetamide
1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-8-[5-(trifluoromethyl)pyridin-2-yl]-1,8-diazaspiro[4.5]decane
methyl 1-ethoxy-2-oxo-8-(thian-4-yl)-1,8-diazaspiro[4.5]decane-4-carboxylate
N-ethyl-N-[(3-ethyl-1,2,4-oxadiazol-5-yl)methyl]-1-methyl-1H-pyrazolo[1,5-a]imidazole-7-carboxamide
1-(4-fluorophenyl)-4-{1-[(2-methylphenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}piperazine
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(1-methoxy-2-methylpropan-2-yl)acetamide
3-(2-amino-1,3-thiazol-4-yl)-1-[(1R,5R)-3-methanesulfonyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
3-(prop-2-en-1-yl)-1-{[(pyridin-2-ylmethyl)carbamoyl]methyl}piperidine-3-carboxylic acid
2-{4-[4-(1H-pyrazol-5-yl)phenyl]-1H-pyrazol-1-yl}ethan-1-ol
(2S)-2-phenyl-2-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)ethan-1-ol
8-methoxy-2-oxo-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,2,3,4-tetrahydroquinoline-4-carboxamide
1-(1-benzylpiperidin-3-yl)-4-(2-fluorophenyl)piperazine
[(5-tert-butyl-1H-pyrazol-3-yl)methyl](ethyl)[2-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]amine
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-[(6-methylpyridin-2-yl)methyl]piperidin-3-amine
[(2-ethoxyphenyl)methyl]({[1-(2-methoxyethyl)piperidin-4-yl]methyl})(pyridin-4-ylmethyl)amine
N-(furan-2-ylmethyl)-3-(1-methyl-1H-pyrrol-2-yl)-N-(thiophen-2-ylmethyl)-1H-pyrazole-5-carboxamide
(2S)-2-phenyl-2-{[2-(pyridin-4-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethan-1-ol
5-(3-benzoylpiperidine-1-carbonyl)-2-methyl-4-phenylpyrimidine
4-chloro-N,N-dimethyl-5-{1-[(4-methyl-1,3-thiazol-2-yl)methyl]-1H-imidazol-2-yl}-1,3-thiazol-2-amine
N-[(3R,4S)-1-(5-cyanopyridin-2-yl)-4-cyclopropylpyrrolidin-3-yl]-2-(propan-2-yloxy)acetamide
N-[1-(1-{[5-(hydroxymethyl)furan-2-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]-2H-1,3-benzodioxole-5-carboxamide
9-(1-ethyl-1H-pyrazole-5-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
2-(5-{[(1S,5R)-6-(2-methoxyethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}furan-2-yl)benzonitrile
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-(hydroxymethyl)azepan-4-ol
2-[(cyclopropylmethyl)sulfanyl]-N-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]acetamide
3-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]propan-1-ol
N-[(3R,4R)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
2-{pyrazolo[1,5-a]pyridin-7-yl}-1,3-thiazole-4-carboxamide
3-[1-({2-[3-(dimethylamino)propoxy]phenyl}methyl)piperidin-4-yl]phenol
N-[(3-methoxyphenyl)methyl]-2-(morpholin-4-yl)-N-propyl-2-(pyridin-3-yl)acetamide
4-[4-(2,2-dimethylpropanoyl)piperazin-1-yl]-5-methylthieno[2,3-d]pyrimidine-6-carboxylic acid
2-butyl-4-{[2-(4-fluorophenyl)pyrrolidin-1-yl]methyl}-1H-imidazole
2-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-[1-(pyridin-4-yl)propyl]benzamide
3-(1H-1,3-benzodiazol-1-yl)-1-[2-(pyrrolidine-1-carbonyl)piperazin-1-yl]propan-1-one
2-(azepan-1-yl)-N-{[(1,3-thiazol-2-yl)carbamoyl]methyl}acetamide
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
4-{[1-(2-methoxyacetyl)piperidin-4-yl]oxy}-N-{[3-(methylsulfanyl)phenyl]methyl}benzamide