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7-(5-chloropyridin-2-yl)-4-(4-methylpyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3R,4R)-1-(cyclopropanesulfonyl)-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
2-methoxy-4-[6-(methylamino)-1H-pyrrolo[2,3-b]pyridin-4-yl]phenol
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl({[1-(piperidin-1-yl)cyclohexyl]methyl})(pyridin-2-ylmethyl)amine
2-({[(3R,4R)-1-[(5-fluoro-1-methyl-1H-indol-2-yl)methyl]-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine
(1R,5R)-6-(cyclopropylmethyl)-3-[6-(4H-1,2,4-triazol-4-yl)pyridine-3-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperidin-3-yl)methyl]acetamide
1-{4-[4-(2-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropane-1-carboxamide
2-(1-methylpyrrolidine-3-carbonyl)-7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinoline
2-{2-ethyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-6-(4-fluorophenyl)pyridine-3-carboxylic acid
6-fluoro-3-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}quinolin-4-ol
ethyl 2-(4-{[4-(3-hydroxyphenyl)piperidine-1-carbonyl]amino}phenyl)acetate
2-{[6-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyrazin-2-yl]sulfanyl}acetic acid
4-[4-(1,3-dimethyl-1H-pyrazol-5-yl)-4H-1,2,4-triazol-3-yl]phenol
1-cyclopropyl-4-[4-(pyridin-3-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
1-({6-methylimidazo[2,1-b][1,3]thiazol-5-yl}methyl)-4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine
1-[1-(3,5-dimethylfuran-2-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N,N,6,8-tetramethyl-2-[1-(2,2,2-trifluoroethyl)-1H-pyrazol-4-yl]quinoline-4-carboxamide
2-(azocan-1-yl)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]acetamide
4-[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]-1-[4-(1H-pyrazol-1-yl)phenyl]piperidine
1-{3-[benzyl(methyl)amino]piperidin-1-yl}-2-(2-chlorophenoxy)ethan-1-one
ethyl (4aS,8aR)-6-({2-methyl-7-oxo-4H,7H-pyrazolo[1,5-a]pyrimidin-5-yl}methyl)-decahydro-1,6-naphthyridine-4a-carboxylate
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]acetamide
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-N-methyl-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)isoquinoline
[4-({5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)phenyl]methanol
4-(6-methoxypyridin-2-yl)-2-({4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}methyl)phenol
N-{[4-(pyrrolidine-1-carbonyl)phenyl]methyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-(4-acetylphenyl)-6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[1-(cyclopropylmethyl)-4-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperazin-2-yl]ethan-1-ol
5-{[(3,4-difluorophenyl)methyl]amino}-N-(furan-2-ylmethyl)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-phenyl-4-(1H-1,2,3-triazole-5-amido)piperidine-1-carboxamide
1,6-dimethyl-N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-1H-indole-2-carboxamide
N-[1-(4-fluorophenyl)-4-(propan-2-yloxy)-1H-indazol-3-yl]-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
4-(1-{[2-(7-methoxy-2H-1,3-benzodioxol-5-yl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-4-yl)thiomorpholine
(1S,5R)-6-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
1,2-dimethyl-5-{1-[1-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
3-benzyl-3-[2-(1,4-diazepan-1-yl)-2-oxoethyl]-1-methyl-2,3-dihydro-1H-indol-2-one
2,6-difluoro-N,3-dimethyl-N-[1-(pyridin-3-yl)ethyl]benzamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}piperidine
methyl[(1-phenylpyrrolidin-3-yl)methyl]{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}amine
1-{2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidin-4-yl}piperidin-4-ol
3-(4-hydroxyphenyl)-5-[(4-methylpiperazin-1-yl)sulfonyl]benzoic acid
2-(pyridin-4-yl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]quinoline-4-carboxamide
6-(thian-4-yl)-N-(thiophen-2-ylmethyl)-6-azaspiro[2.5]octane-1-carboxamide
5-(2-chloro-4-methoxyphenoxymethyl)-N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1,2-oxazole-3-carboxamide
(3S,4R)-4-methyl-3-(2-methylpropyl)-1-(2-propylpyridine-4-carbonyl)piperidin-4-ol