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1-[4-benzyl-4-(hydroxymethyl)piperidin-1-yl]-2-(3-methoxyphenoxy)ethan-1-one
4-{[1-(3-methylpyrazin-2-yl)piperidin-4-yl]oxy}-N-(pyridin-2-ylmethyl)benzamide
(1S,5R)-3-benzyl-6-[(2-cyclohexylpyrimidin-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2-chlorophenoxy)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-(3-benzoylpiperidin-1-yl)pyridine-3-carboxylic acid
N-cyclopropyl-4-methoxy-2-({1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-(hexahydro-1H-pyrrolizin-7a-ylmethyl)-4-(4-methylpiperazin-1-yl)benzamide
1-(adamantan-2-yl)-4-[(2S,4S)-1-[(2-fluorophenyl)methyl]-4-[(4-methoxyphenyl)sulfanyl]pyrrolidine-2-carbonyl]piperazine
1-(5-ethyl-1,3-oxazole-4-carbonyl)-4-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
3-(3,4-dimethoxyphenyl)-N-ethyl-N-(pyridin-4-ylmethyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
2-ethoxy-5-[2-({pyrazolo[1,5-a]pyrimidin-3-ylmethyl}amino)pyrimidin-4-yl]benzoic acid
2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]({[4-(methylsulfanyl)phenyl]methyl})amino}ethan-1-ol
2-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyridine-3-carbonitrile
4-methyl-2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
methyl({[2-(2-methylphenyl)pyrimidin-5-yl]methyl})(pyrazin-2-ylmethyl)amine
3-(1H-1,3-benzodiazol-2-yl)-1-[4-(pyridin-4-ylmethyl)-1,4-diazepan-1-yl]propan-1-one
N-(5-chloro-2-methoxyphenyl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
4-{6-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl}thiomorpholine
4-(2-methoxyphenyl)-1-(oxolan-3-ylmethyl)piperidine
N-(2,3-dihydro-1H-inden-2-yl)-5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2-(4-fluorophenyl)-N-(2-hydroxy-2-phenylethyl)imidazo[1,2-a]pyridine-6-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-({[5-(trifluoromethyl)pyridin-2-yl]amino}methyl)pyridin-2-amine
1-[(1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
N-{[1-(1H-indol-2-ylmethyl)pyrrolidin-3-yl]methyl}-3-methyl-1H-pyrazole-5-carboxamide
1-{2-[({2-[2-hydroxy-3-(4-methylpiperazin-1-yl)propoxy]-4-methoxyphenyl}methyl)amino]ethyl}piperidin-2-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-(6-oxo-1,4,5,6-tetrahydropyridazine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-amino-2-(3,5-dimethyl-1H-pyrazol-4-yl)-1-(4-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-yl}piperidin-1-yl)ethan-1-one
(4aR,8aS)-1-[2-(3,4-dimethoxyphenyl)ethyl]-6-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-decahydro-1,6-naphthyridin-2-one
2-(4-ethoxyphenyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}acetamide
2-[4-(3-methyl-1H-indole-2-carbonyl)piperazin-1-yl]-1,3-benzothiazole
1-(2-methyloxane-2-carbonyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
(3S,7S,8aS)-7-{[(2,5-difluorophenyl)methyl]amino}-3-propyl-octahydropyrrolo[1,2-a]piperazine-1,4-dione
6-methoxy-2-{[5-(oxan-2-yl)furan-2-yl]methyl}-1,2,3,4-tetrahydroisoquinoline
N-(3-methoxyphenyl)-3-(4-phenylbenzoyl)piperidine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(pyrrolidin-1-yl)pyridine-3-carboxamide
2,5-dimethyl-N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)pyrazolo[1,5-a]pyrimidin-7-amine
5-acetyl-N-[2-(dimethylamino)ethyl]-6-methyl-N-[(5-methylthiophen-2-yl)methyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[4-(3,5-dimethoxyphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]propan-2-one
9-(dimethyl-1,2-oxazole-4-carbonyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-(6-aminopyridin-3-yl)-5,6-dimethylpyridine-3-carboxamide
N-[(2,3-difluoro-4-methoxyphenyl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide
2-phenyl-N-[2-(pyrrolidin-1-yl)ethyl]imidazo[1,2-a]pyridine-6-carboxamide
(3R)-3,4,4-trimethyl-1-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)pyrrolidin-3-ol
N,1-dimethyl-2-oxo-N-[1-(pyridin-3-yl)propyl]-1,2-dihydroquinoline-4-carboxamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-2-(dimethyl-1,3-thiazol-5-yl)-N-methylacetamide
9-[(1-methyl-1H-indol-6-yl)methyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecan-9-yl}-4-[4-(propan-2-yl)phenyl]butan-1-one
1-methyl-N-[1-(5,6,7,8-tetrahydronaphthalen-2-yl)ethyl]-1H-pyrazole-5-carboxamide
2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]-N-(1-propylcyclopropyl)acetamide
4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]-1-{thieno[3,2-d]pyrimidin-4-yl}piperidine