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4-chloro-1-methyl-N-(2-methylpropyl)-N-(pyridin-2-ylmethyl)-1H-pyrazole-3-carboxamide
[(3,5-dichloropyridin-4-yl)methyl][(4-fluorophenyl)methyl](pyridin-4-ylmethyl)amine
N-methyl-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
1-(3,5-difluorophenyl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-4-amine
4-(2-{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-2-yl}ethyl)morpholine
(1S,6R)-9-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-3,9-diazabicyclo[4.2.1]nonane
N-(2-{1-[2-(4-chloro-3,5-dimethylphenoxy)propanoyl]piperidin-4-yl}ethyl)acetamide
N,N-diethyl-N'-methyl-N'-[1-(pyridin-4-yl)ethyl]ethanediamide
5-{[4-(1-methyl-1H-imidazol-2-yl)piperidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
2-[2-(4-fluorophenyl)ethyl]-4-{4-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-{[1-(propan-2-yl)pyrrolidin-3-yl]methyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
2-(3,3,3-trifluoropropyl)-1H-1,3-benzodiazole-6-carboxylic acid
1-(4-cyclobutyl-6-methylpyrimidin-2-yl)-4-(hydroxymethyl)piperidin-4-ol
N-ethyl-6-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-N-[(1-methyl-1H-imidazol-2-yl)methyl]pyridine-3-carboxamide
1-(2-ethoxyethyl)-N-ethyl-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-phenyl-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]-1,4-diazepane
3-hydroxy-1-[(3-methylphenyl)methyl]-3-({[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]amino}methyl)piperidin-2-one
1-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-4-[2-(2-phenylethyl)-3H-imidazo[4,5-b]pyridin-3-yl]piperidine
6-methyl-3-(3-phenylpiperazine-1-carbonyl)-4H-pyrido[1,2-a]pyrimidin-4-one
2-(dimethylamino)-2-(2-fluorophenyl)-1-{1-oxa-7-azaspiro[3.5]nonan-7-yl}ethan-1-one
4-{6-[(diethylamino)methyl]pyrazolo[1,5-a]pyrimidine-3-carbonyl}-1-methylpiperazin-2-one
2-(adamantan-1-yl)-4-hydroxy-N-methyl-N-(1H-pyrazol-3-ylmethyl)pyrimidine-5-carboxamide
2-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-5,6,7,8-tetrahydroquinoline
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridin-2-amine
2-[(1S,5R)-3-{[(furan-2-ylmethyl)carbamoyl]methyl}-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-({4-methyl-5-[1-(1H-pyrrole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-(2,4-dimethoxyphenyl)-1-[(1R,5S,6S)-6-[(dimethylamino)methyl]-3-azabicyclo[3.1.0]hexan-3-yl]ethan-1-one
N-(dimethyl-1H-1,2,4-triazol-3-yl)-3-(dimethylamino)piperidine-1-carboxamide
1-[benzyl(methyl)amino]-3-{5-[(cyclopentylamino)methyl]-2-methoxyphenoxy}propan-2-ol
3-{4-[6-amino-2-(butylsulfanyl)pyrimidin-4-yl]piperazin-1-yl}-1,2-dihydropyrazin-2-one
1-(2-aminoethyl)-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-1H-1,2,3-triazole-4-carboxamide
5-(2-acetylbenzoyl)-1-(cyclopropylmethyl)-N-methyl-N-(1,3-thiazol-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-phenylpropan-1-one
3-(5-{1-[(4-chloro-3-methyl-1H-pyrazol-5-yl)methyl]piperidin-3-yl}-1,2,4-oxadiazol-3-yl)pyridine
2-(3,4-dichlorophenyl)-4-(1-ethyl-5-methyl-1H-pyrazole-4-carbonyl)morpholine
5-(2-methylpropyl)-3-{[4-phenyl-5-(1,3-thiazol-2-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazole
2-(2-{[3-(1H-imidazol-1-yl)pyrrolidin-1-yl]methyl}phenyl)-6-(methoxymethyl)-3,4-dihydropyrimidin-4-one
3-(dimethyl-1,2-oxazol-4-yl)-1-{[1-(oxan-4-yl)piperidin-3-yl]methyl}urea
2-amino-6-(3,4-dichlorophenyl)-4-(1,3-dimethyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
[(1-tert-butyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](methyl){[3-(3-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-[2-({2-cyclopropyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}amino)ethyl]piperidin-3-ol
(3E)-1-[(1S,5R)-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]pent-3-en-1-one
1-(2-methylphenyl)-3-{1-[1-(oxan-4-yl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
3-[3-(dimethylamino)propyl]-8-(quinoline-5-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-(1H-pyrazol-4-yl)butanamide
4-[3-(2-cyclohexylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-5-ethyl-1,3-oxazole
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)propan-2-yl]-1-methyl-3-(trimethyl-1H-pyrazol-4-yl)-1H-pyrazole-5-carboxamide
1-[3-(furan-2-yl)-5-[2-(1H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
7-[2-(3-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidin-5-yl)acetyl]-2,7-diazaspiro[4.4]nonane-1,3-dione
7-fluoro-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]quinazolin-4-amine