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N-[2-(2,3-dihydro-1,4-benzodioxin-2-yl)ethyl]-1-(propan-2-yl)piperidine-4-carboxamide
2-(4-{2-[3-(furan-2-yl)phenyl]-1H-imidazol-1-yl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
1-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-hydroxyethan-1-one
7-chloro-3-[4-(1H-imidazol-2-yl)piperidine-1-carbonyl]quinolin-4-ol
7-[2-(1H-pyrazol-1-yl)benzoyl]-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
1-{5-[(3-propoxypiperidin-1-yl)methyl]imidazo[2,1-b][1,3]thiazole-6-carbonyl}azocane
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-2-(3-methyl-1,2-oxazol-5-yl)acetamide
9-{[4-(propan-2-yl)phenyl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
(3aS,6aS)-2-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]acetyl}-5-(2-methylpropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
2-ethyl-4-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-imidazol-2-yl)pyrimidine
2-({1-[(5-chlorothiophen-2-yl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
N-({5-[(2,3-difluoro-4-methylphenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)cyclobutanecarboxamide
1-[3-(furan-2-yl)propanoyl]-4-phenoxypiperidine-4-carboxylic acid
N-methyl-5-{[methyl({3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-yl})amino]methyl}pyrimidin-2-amine
(4aR,8aS)-1-(2H-1,3-benzodioxol-5-ylmethyl)-6-{[4-(2-methylphenyl)phenyl]methyl}-decahydro-1,6-naphthyridin-2-one
1-[(2R,3R,6R)-3-(4-fluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3-(2-methyl-1H-imidazol-1-yl)propan-1-one
6-amino-N-[2-(5-methoxy-1H-1,3-benzodiazol-2-yl)ethyl]-N-methylpyridine-3-carboxamide
N-[2-(ethanesulfonyl)ethyl]-5-ethyl-1,2-oxazole-3-carboxamide
1-{4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(pyrimidin-2-ylsulfanyl)ethan-1-one
3-(1-methyl-1H-pyrazol-5-yl)-1-[2-(pyridin-3-yloxy)propyl]urea
3-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-1-(1-propyl-1H-1,3-benzodiazol-5-yl)urea
2-(4-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepine-9-carbonyl}piperazin-1-yl)pyrimidine
(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)methanol
4-[4-(2-chlorophenyl)piperidin-4-yl]-N-[(5-methylfuran-2-yl)methyl]pyrimidin-2-amine
1-cyclohexyl-5-[(3,4-dimethoxyphenyl)methyl]-1H-1,2,4-triazole
(2S,4S)-4-amino-N-methyl-1-{2-[(4-methyl-1,3-thiazol-2-yl)sulfanyl]acetyl}pyrrolidine-2-carboxamide
1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N,N-bis(prop-2-en-1-yl)piperidine-3-carboxamide
1-ethyl-N-methyl-N-{[2-(trifluoromethyl)phenyl]methyl}-1H-pyrazole-3-carboxamide
1-amino-N-[1-benzyl-4-(pyridin-3-yloxy)-1H-indazol-3-yl]cyclopropane-1-carboxamide
2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}-N-(pyridin-2-ylmethyl)acetamide
2-{4-[(2-aminopyrimidin-5-yl)methyl]-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-ethyl-3-(piperidin-4-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl 1-(2-{[(3-chlorophenyl)methyl]carbamoyl}ethyl)piperidine-4-carboxylate
2-{2-[1-(cyclopropylmethyl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]-1H-pyrrol-1-yl}-1,3-thiazole
N-{1-[6-(methoxymethyl)-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl]piperidin-4-yl}methanesulfonamide
N-(2-chloro-6-methylphenyl)-2-(methoxymethyl)piperidine-1-carboxamide
2-(5-chloro-6-methyl-1-benzofuran-3-yl)-N-(3-hydroxypropyl)-N-(pyridin-4-ylmethyl)acetamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]acetamide
methyl({[2-(morpholin-4-yl)pyrimidin-5-yl]methyl})[(3-phenyl-1H-pyrazol-5-yl)methyl]amine
1-(3-chloro-2,6-dimethylphenyl)-3-[(3S,4S)-4-methoxy-1-methylpyrrolidin-3-yl]urea
5-(propan-2-yl)-N-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}ethyl)-1,2-oxazole-3-carboxamide
4-acetyl-N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}benzamide
N,N-dimethyl-2-[2-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]carbamoyl}amino)phenyl]acetamide
4-(3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}phenyl)phenol
2-(5-chloro-2-ethoxyphenyl)-2-(pyrrolidin-1-yl)acetic acid
4-(3-methylphenyl)-3-(3,4,5-trimethoxyphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(benzenesulfonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
2-{3-[({imidazo[1,2-a]pyridin-3-ylmethyl}(methyl)amino)methyl]phenyl}-3H,4H,5H,6H,7H-cyclopenta[d]pyrimidin-4-one
2-{[5-(4-methoxyphenyl)furan-2-yl]methyl}-octahydro-1H-pyrido[1,2-a]piperazine
3-({[(6-chloropyridin-3-yl)methyl](methyl)amino}methyl)-1-methyl-1,2-dihydroquinolin-2-one