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1-{[4-(methylsulfanyl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)piperidin-4-ol
N-(cyclopropylmethyl)-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-(cyclopropylmethyl)-5-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2-[(4-chlorophenyl)methyl]-8-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-2,8-diazaspiro[4.5]decan-3-one
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-3,3-dimethylbutan-1-one
2-methyl-1-[2-(oxolan-3-yl)ethyl]-1,4-dihydroquinolin-4-one
N-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-N-(propan-2-yl)-4,5,6,7-tetrahydro-1,2-benzoxazole-3-carboxamide
3-[2-(4-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]-5-(propan-2-yl)-1,2-oxazole
N-[2-(ethanesulfonyl)ethyl]-1-ethyl-3,5-dimethyl-1H-pyrazole-4-carboxamide
2-[(2-fluoro-4,5-dimethoxyphenyl)methyl]-2-azaspiro[4.5]decan-3-one
1-[(3S,4S)-3,4-dihydroxy-4-methylpiperidin-1-yl]-2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]ethan-1-one
1-{5-methoxy-2-[({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}amino)methyl]phenoxy}-3-(4-methylpiperazin-1-yl)propan-2-ol
ethyl 4-(5-ethyl-1,3-oxazole-4-carbonyl)piperazine-1-carboxylate
N-[2-(dimethylamino)ethyl]-N-methyl-3-{[1-(4-methylbenzoyl)piperidin-4-yl]oxy}benzamide
(1S,9aR)-1-(4H-1,2,4-triazol-4-ylmethyl)-octahydro-1H-quinolizine
2-(2-{[4-(ethylamino)pyrimidin-2-yl]amino}ethyl)-6-methyl-3,4-dihydropyrimidin-4-one
(4aS,8aR)-1-(4-hydroxybutyl)-6-(isoquinolin-1-yl)-decahydro-1,6-naphthyridin-2-one
2-(dimethylamino)-4-methyl-N-(2-phenoxyethyl)pyrimidine-5-carboxamide
1-(4-methoxyphenyl)-4-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperazin-2-one
2-({methyl[2-(morpholin-4-yl)propyl]amino}methyl)quinolin-8-ol
N-{1-[2-(azocan-1-yl)-4-methylpyrimidin-5-yl]ethyl}-5-methyl-1,3-oxazole-4-carboxamide
(2S,4S,5R)-1-methyl-4-{[(1-methyl-1H-pyrazol-4-yl)methyl]carbamoyl}-2-(2-methylpropyl)-5-(pyridin-3-yl)pyrrolidine-2-carboxylic acid
(3aR,5R,6S,7aS)-2-[1-(4-chlorophenyl)cyclobutanecarbonyl]-octahydro-1H-isoindole-5,6-diol
2-(3-methoxypropyl)-8-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
{[(1R,5S,6S)-3-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl}dimethylamine
2-(2-{[3-(dimethylamino)pyrrolidin-1-yl]methyl}phenyl)-6-(3-methylpyrazin-2-yl)-3,4-dihydropyrimidin-4-one
6-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}pyridine-2-carboxylic acid
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2-methyl-6-(propan-2-yl)pyrimidin-4-amine
N-(1-benzylpyrrolidin-3-yl)-3-{1-[2-(methylsulfanyl)acetyl]piperidin-4-yl}propanamide
N-[(2-fluoro-4-methoxyphenyl)methyl]-7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
5-{[3-(2-methoxyphenoxy)azetidin-1-yl]methyl}-N,N-dimethylpyridin-2-amine
4-ethyl-5-methyl-2-{4-[(1-methylpiperidin-3-yl)methyl]piperazin-1-yl}pyrimidine
N-[(3S,4R)-1-(3,5-difluoropyridine-2-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
({3-[(2-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl)(oxan-2-ylmethyl)amine
propan-2-yl (4aR,7aS)-4-[(4-chlorophenyl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
3-(2-aminoethyl)-4-[4-(trifluoromethoxy)phenyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(5-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}-2-methylphenyl)imidazolidin-2-one
(3aS,7aR)-5-methyl-2-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
5-methyl-N-[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-[(2-fluorophenyl)formamido]-N-[2-(methylsulfamoyl)ethyl]propanamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-[2-(dimethylamino)ethyl]piperidine-3-carboxamide
N-(cyclohexylmethyl)-3-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidine-1-carboxamide
5-methyl-N-[4-(morpholine-4-carbonyl)phenyl]-1H-indazole-3-carboxamide
N-butyl-4-propyl-N-(pyridin-4-ylmethyl)pyrimidine-5-carboxamide
7-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-[2-(ethylamino)pyrimidin-4-yl]pyridine-4-carboxylic acid
9-{4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}-3-azaspiro[5.5]undecane
N-(1-{1-[(2-methyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenylpropanamide
3-(dimethylsulfamoyl)-5-[(furan-3-ylmethyl)amino]-N-methyl-N-[1-(pyridin-2-yl)ethyl]benzamide