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7-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-2-oxa-7-azaspiro[4.5]decan-8-one
(4aR,8aR)-7-[(3,4-dimethylphenyl)methyl]-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
4-{[4-(benzenesulfonyl)piperazin-1-yl]methyl}-1-ethyl-1H-pyrrole-2-carbonitrile
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)morpholine
2-(1H-imidazol-1-yl)-1-{2-[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}ethan-1-one
(3S,4R)-1-[2-(2,4-dimethyl-6-oxo-1,6-dihydropyrimidin-5-yl)acetyl]-4-(4-fluorophenyl)pyrrolidine-3-carboxylic acid
N-[1-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-[5-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-({1-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanoyl]piperidin-3-yl}methyl)-4-fluorobenzamide
1-[(1-methyl-1H-imidazol-2-yl)methyl]-N-[4-(1,3-thiazol-4-yl)phenyl]pyrrolidine-2-carboxamide
1-(3-methoxyphenyl)-4-[(3R)-1,2,3,4-tetrahydroisoquinoline-3-carbonyl]piperazin-2-one
1-(1H-indazole-3-carbonyl)-4-(2-methyl-1H-imidazol-1-yl)piperidine-4-carboxylic acid
(2S)-N-[2-methyl-4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]oxolane-2-carboxamide
5-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
1-(methoxymethyl)-N-{1-[2-(trifluoromethyl)phenyl]ethyl}cyclobutane-1-carboxamide
1-methyl-2-{1-[2-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-imidazol-2-yl}-1H-imidazole
methyl 4-[(2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamido)methyl]benzoate
(1R,5R)-6-[3-(methylsulfanyl)propyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
ethyl 1-[5-(4-chloro-3,5-dimethylphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidine-3-carboxylate
3-(1-methyl-1H-pyrazol-5-yl)-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)propanamide
1-(furan-2-yl)-2-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethane-1,2-dione
1-cyclopropanecarbonyl-3-[2-(2,6-difluorophenyl)ethyl]piperidine
N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}-2-(2-oxopyrrolidin-1-yl)propanamide
2-[3-(2,3-dimethoxyphenyl)pyrrolidin-1-yl]-5-methyl-4-(1-methyl-1H-pyrazol-4-yl)pyrimidine
2-(1H-indol-3-yl)-1-[4-(3-methylpyridin-4-yl)-1,4-diazepan-1-yl]ethan-1-one
2-(1-{[2-fluoro-4-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)propan-2-ol
7-(cyclopropylmethyl)-2-(3-hydroxyazetidine-1-carbonyl)-6-(4-methoxyphenyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
2-(2-{[3-(4-methylpiperazine-1-carbonyl)piperazin-1-yl]methyl}phenoxy)acetic acid
N-{1-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]ethyl}-5-(morpholin-4-ylmethyl)furan-3-carboxamide
(1S,6R)-N-(2,2-difluoro-2H-1,3-benzodioxol-5-yl)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carboxamide
3-(1H-indol-3-yl)-1-{3-[3-(trifluoromethyl)benzoyl]piperidin-1-yl}propan-1-one
2-[1-(furan-2-ylmethyl)-4-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)piperazin-2-yl]ethan-1-ol
3-[4-(4-methoxyphenoxy)piperidin-1-yl]-5-(3-methoxyphenyl)-1,2,4-triazine
methyl 1-{[(1-cyclohexyl-1H-pyrazol-5-yl)carbamoyl]methyl}-1H-pyrazole-3-carboxylate
4-[(6-methylpyridin-3-yl)oxy]-1-[(3-methylthiophen-2-yl)methyl]piperidine-4-carboxylic acid
{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[(3-phenyl-1,2-oxazol-5-yl)methyl]amine
N4-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-methylpyrimidine-4,6-diamine
N-[2-(dimethylamino)ethyl]-4-(4,5,6-trimethylpyridin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-amine
3-{[2-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]methyl}-5-methyl-1,2-oxazole
3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-N-{2-[(pyridin-3-yl)amino]ethyl}propanamide
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,9-dioxaspiro[5.5]undecan-4-amine
{2,4,6-trimethyl-3-[({2-[(3-methylpyridin-2-yl)amino]ethyl}amino)methyl]phenyl}methanol
4-(4-chlorophenyl)-1-(2-methyl-1,3-thiazole-4-carbonyl)piperidin-4-ol
1-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-7-yl)methyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
2-[5-(1-methylazepan-2-yl)-1-(quinolin-8-yl)-1H-1,2,4-triazol-3-yl]acetamide
1-{1-[(3,4-difluorophenyl)methyl]piperidin-4-yl}-N-(2-methoxyethyl)piperidine-3-carboxamide
3-(2-{[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}ethyl)-2,3-dihydro-1,3-benzoxazol-2-one
1-{4-[(3-{1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carbonyl}-1,2-oxazol-5-yl)methoxy]phenyl}-1H-1,2,4-triazole
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-N-methylacetamide
5-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carbonitrile
3-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]-6-methylpyridazine