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(2R,3S,6R)-5-benzoyl-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
[(4-ethynylphenyl)methyl]({1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl})amine
N,5-dimethyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-4-[(oxolan-2-ylmethyl)amino]thieno[2,3-d]pyrimidine-6-carboxamide
2-benzyl-9-[(dimethyl-1,3-thiazol-5-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(2-cyclopentylethyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
4-[(2E)-3-phenylprop-2-en-1-yl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-[2-methoxy-4-({[2-(4-methylphenyl)ethyl]amino}methyl)phenoxy]-3-[methyl(propan-2-yl)amino]propan-2-ol
N-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-2-(pyridin-3-yloxy)acetamide
(3aS,7aR)-5-methyl-2-(5-methyl-4-phenylthiophene-3-carbonyl)-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
N-(3-cyanophenyl)-3-{[4-(2-hydroxyethyl)piperazin-1-yl]methyl}benzamide
{4-[(4-phenylphenyl)methyl]-1,4-oxazepan-6-yl}methanol
3-(1H-1,2,3-benzotriazol-4-yl)-1-benzyl-1-(oxolan-2-ylmethyl)urea
N-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]-3-(2-fluorophenyl)-1H-pyrazole-5-carboxamide
3-(5-{[3-(4-methylphenoxymethyl)piperidin-1-yl]methyl}thiophen-3-yl)prop-2-yn-1-ol
5-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[1-(thiophen-3-yl)propan-2-yl]pyridin-2-amine
1-{6-chloro-2-methylimidazo[1,2-a]pyridine-3-carbonyl}-4-methanesulfonyl-1,4-diazepane
3-({5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}amino)butan-1-ol
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2-(thiophen-3-yl)acetamide
N-[1-(3-cyclopentyl-1,2,4-oxadiazol-5-yl)butyl]acetamide
2-[(2,6-dichlorophenyl)methyl]-5-(3-methoxypiperidine-1-carbonyl)pyrimidin-4-ol
5-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridine-6-carbonyl]-2-methylpyrimidine
2-{[3-fluoro-2-(trifluoromethyl)phenyl]methyl}-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
(3S,4R)-1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-(hydroxymethyl)piperidin-3-ol
2-(3-{1-[(1R,2S)-2-phenylcyclopropyl]-1H-1,2,3-triazol-4-yl}phenoxy)acetamide
6-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-ylmethyl]-N-({2-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)-2-oxo-1,2-dihydropyridine-3-carboxamide
3-({1-[3-(3-fluorophenyl)phenyl]piperidin-4-yl}amino)-2,2-dimethylpropan-1-ol
2-[4-(1-benzofuran-2-ylmethyl)morpholin-3-yl]-1-(4-ethylpiperazin-1-yl)ethan-1-one
4-{[4-(1,5-dimethyl-1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}-5-(hydroxymethyl)-2-methylpyridin-3-ol
N-(3-aminopropyl)-2-[(3-methoxyphenyl)amino]butanamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(2-methoxy-2-methylpropyl)piperidine-3-carboxamide
5-(pyrrolidin-1-ylmethyl)-N-[1-(thian-4-yl)piperidin-4-yl]furan-2-carboxamide
N-[(3R,4R)-1-[(2E)-3,7-dimethylocta-2,6-dien-1-yl]-3-hydroxypiperidin-4-yl]pyridine-2-carboxamide
2-amino-6-(2-amino-4-methyl-1,3-thiazol-5-yl)-4-(2-chloro-4-hydroxyphenyl)pyridine-3-carbonitrile
(3S,4S)-1-{[5-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
(1R,9S)-5-amino-3-{2-[2-(dimethylamino)ethoxy]phenyl}-12-methyl-6,12-diazatricyclo[7.2.1.02,7]dodeca-2,4,6-triene-4-carbonitrile
4-[(4-hydroxy-6,8-dimethylquinolin-2-yl)methyl]piperazin-2-one
N-[(3S,4R)-1-{[1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-propylpyrrolidin-3-yl]acetamide
[3-(3-methylbut-2-en-1-yl)-1-(oxan-4-ylmethyl)piperidin-3-yl]methanol
[4-(6-methoxy-3-methyl-1-benzofuran-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methanol
5-[3-(thiophen-3-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)cyclopropanecarboxamide
9-(2,4-dimethylbenzoyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
[1-(oxolane-3-carbonyl)piperidin-4-yl]diphenylmethanol
N-(3,4-difluorophenyl)piperidin-3-amine
3-[(dimethylamino)methyl]-1-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)pyrrolidin-3-ol
N-cyclopropyl-5-phenyl-N-(thiophen-3-ylmethyl)-1H-pyrazole-3-carboxamide
4-benzyl-3-[2-(4-benzylpiperidin-1-yl)-2-oxoethyl]piperazin-2-one
8-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}quinoline-2-carboxamide
(3aR,6aR)-2-(2-methoxyacetyl)-N-[2-(3-methylpyridin-2-yl)ethyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
1'-[3-(trimethyl-1H-pyrazol-4-yl)propanoyl]-3,4-dihydrospiro[1-benzopyran-2,3'-pyrrolidine]-4-one