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2-{4-[(3-chlorophenyl)methyl]piperazine-1-carbonyl}-N,N-dimethylaniline
1-(morpholin-2-ylmethyl)-3-[4-(1H-pyrazol-1-yl)phenyl]urea
3-[2-(piperidin-2-yl)ethyl]-5-[5-(pyrrolidine-1-carbonyl)furan-2-yl]phenol
N-[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
5-chloro-6-[2-(dimethylamino)phenyl]-2-methylpyrimidin-4-ol
(1R,7S)-3-(2-ethylbutyl)-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
{5-[1-(6-phenoxypyridin-3-yl)-1H-imidazol-2-yl]furan-2-yl}methanol
1-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}-4-(methoxymethyl)piperidine
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(5-methylpyrazine-2-carbonyl)-2,7-diazaspiro[4.5]decane
5-{3-[3-(4-fluorophenyl)oxolan-3-yl]-1,2,4-oxadiazol-5-yl}-4-propylpyrimidine
(1R,2R,6S,7S)-N-(2-fluoro-5-methanesulfonamidophenyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane-4-carboxamide
3-[1-(2,3-dimethylphenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methylbut-3-enamide
N-benzyl-2-(morpholin-4-yl)-2-oxo-N-(prop-2-en-1-yl)acetamide
2-(3-methoxy-2-oxo-1,2-dihydropyridin-1-yl)-N-methyl-N-(piperidin-4-yl)acetamide
N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-3-(piperidin-3-yl)benzamide
5-(2,3-dihydro-1,4-benzodioxine-5-carbonyl)-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}-3-methyl-1-(pyridin-2-yl)-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1,4-diazepan-5-one
5-({2-[5-(hydroxymethyl)furan-2-yl]-1H-imidazol-1-yl}methyl)-N,N-dimethylfuran-2-carboxamide
8-(3-methyl-1H-pyrazole-5-carbonyl)-2-[(2E)-3-phenylprop-2-en-1-yl]-2,8-diazaspiro[4.5]decan-3-one
N,N-dimethyl-2-[4-phenyl-5-(thiophen-3-yl)-1H-imidazol-1-yl]propanamide
9-(4-chloro-1,5-dimethyl-1H-pyrazole-3-carbonyl)-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[3-(3-fluorophenyl)benzoyl]-4-(2-methoxyethyl)-1,4-diazepan-5-one
2-(1H-imidazol-4-yl)-1-methyl-5-(pyrrolidine-1-sulfonyl)-1H-1,3-benzodiazole
3-{4-[(pyridin-2-yl)amino]piperidine-1-carbonyl}piperidine-1-carboxamide
3-(1-benzyl-5-oxopyrrolidin-3-yl)-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(1S,2S)-1,3-dihydroxy-1-phenylpropan-2-yl]-5-[(4-methylpiperazin-1-yl)methyl]furan-2-carboxamide
3,3,3-trifluoro-1-[(3R,5R)-3-(hydroxymethyl)-5-{[(2-methoxyethyl)(methyl)amino]methyl}piperidin-1-yl]propan-1-one
1-[2-amino-4-(pyridin-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl]-3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propan-1-one
{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[4-(morpholin-4-yl)butyl]amine
N'-(3-fluorophenyl)-N-(thiolan-3-yl)butanediamide
3-methyl-5-[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-pyrazole
1-[4-(3-methoxyphenyl)phenyl]-N-(pyrimidin-4-ylmethyl)piperidin-4-amine
N-{[1-(naphthalen-1-yl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
N,1,3-trimethyl-N-(pyrazin-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
[3-(2-methoxyethyl)-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-3-yl]methanol
[(4-methyl-1H-imidazol-5-yl)methyl]({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)amine
N-cyclopropyl-2-[(3S,4S)-3-hydroxy-4-(naphthalen-2-yl)piperidin-1-yl]pyridine-4-carboxamide
N-(cyclobutylmethyl)-2-(ethylamino)-N-(oxolan-2-ylmethyl)pyrimidine-5-carboxamide
1-{2-[2-(4-methoxyphenyl)acetamido]ethyl}-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
2-[4-(6-methoxypyridin-3-yl)-1H-pyrazol-1-yl]-N-[3-methyl-1-(pyridin-2-yl)-1H-pyrazol-5-yl]acetamide
1-[(2,6-difluorophenyl)methyl]-N-[2-methyl-1-(1-methyl-1H-imidazol-2-yl)propyl]-1H-1,2,3-triazole-4-carboxamide
2-chloro-N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-5-acetamidobenzamide
1-(azocan-1-yl)-3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propan-1-one
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
N-[(5-methylfuran-2-yl)methyl]-3-{1-[(2E)-3-(pyridin-2-yl)prop-2-enoyl]piperidin-3-yl}propanamide
3-{[4-(thiophen-2-ylmethyl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
3-amino-1-(2-phenylethyl)pyrrolidine-3-carboxylic acid